NO20083005L - Anvendelse av benzofuserte heterocykliske sulfamidderivater for behandling av smerte - Google Patents

Anvendelse av benzofuserte heterocykliske sulfamidderivater for behandling av smerte

Info

Publication number
NO20083005L
NO20083005L NO20083005A NO20083005A NO20083005L NO 20083005 L NO20083005 L NO 20083005L NO 20083005 A NO20083005 A NO 20083005A NO 20083005 A NO20083005 A NO 20083005A NO 20083005 L NO20083005 L NO 20083005L
Authority
NO
Norway
Prior art keywords
pain
treatment
formula
sulfamide derivatives
benzofused heterocyclic
Prior art date
Application number
NO20083005A
Other languages
English (en)
Inventor
Allen B Reitz
Virginia L Smith-Swintosky
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of NO20083005L publication Critical patent/NO20083005L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D321/00—Heterocyclic compounds containing rings having two oxygen atoms as the only ring hetero atoms, not provided for by groups C07D317/00 - C07D319/00
    • C07D321/02—Seven-membered rings
    • C07D321/10—Seven-membered rings condensed with carbocyclic rings or ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/357—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)

Abstract

Det beskrives en fremgangsmåte for behandling av smerte omfattende administrering til et individ som trenger det, av en terapeutisk effektiv mengde av et eller flere nye benzofuserte heterosykelsulfamidderivater med formel (I) eller formel (II) som beskrevet her. Det beskrives videre metoder for behandling av smerte omfattende ko-terapi med et eller flere analgetiske midler og en forbindelse med formel (i) eller formel (II) som beskrevet her.
NO20083005A 2005-12-19 2008-07-03 Anvendelse av benzofuserte heterocykliske sulfamidderivater for behandling av smerte NO20083005L (no)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US75168605P 2005-12-19 2005-12-19
US77381206P 2006-02-15 2006-02-15
US11/612,071 US8716231B2 (en) 2005-12-19 2006-12-18 Use of benzo-fused heterocycle sulfamide derivatives for the treatment of pain
PCT/US2006/048539 WO2007075752A1 (en) 2005-12-19 2006-12-19 Use of benzo-fused heterocycle sulfamide derivatives for the treatment of pain

Publications (1)

Publication Number Publication Date
NO20083005L true NO20083005L (no) 2008-09-16

Family

ID=38007332

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20083005A NO20083005L (no) 2005-12-19 2008-07-03 Anvendelse av benzofuserte heterocykliske sulfamidderivater for behandling av smerte

Country Status (27)

Country Link
US (1) US8716231B2 (no)
EP (1) EP1973540B1 (no)
JP (1) JP5190377B2 (no)
KR (1) KR20080077025A (no)
CN (1) CN101378746B (no)
AT (1) ATE447948T1 (no)
AU (1) AU2006331734B2 (no)
BR (1) BRPI0620018A2 (no)
CA (1) CA2634115C (no)
CR (1) CR10167A (no)
CY (1) CY1109732T1 (no)
DE (1) DE602006010442D1 (no)
DK (1) DK1973540T3 (no)
EA (1) EA016302B1 (no)
ES (1) ES2335699T3 (no)
HK (1) HK1125039A1 (no)
HR (1) HRP20100007T1 (no)
IL (1) IL192100A0 (no)
MY (1) MY150903A (no)
NI (1) NI200800169A (no)
NO (1) NO20083005L (no)
NZ (1) NZ569040A (no)
PL (1) PL1973540T3 (no)
PT (1) PT1973540E (no)
RS (1) RS51249B (no)
SI (1) SI1973540T1 (no)
WO (1) WO2007075752A1 (no)

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US8497298B2 (en) 2005-12-19 2013-07-30 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels
US8937096B2 (en) 2005-12-19 2015-01-20 Janssen Pharmaceutica Nv Use of benzo-fused heterocyle sulfamide derivatives for the treatment of mania and bipolar disorder
US20070155827A1 (en) * 2005-12-19 2007-07-05 Smith-Swintosky Virginia L Use of benzo-fused heterocycle sulfamide derivatives for the treatment of depression
US8691867B2 (en) 2005-12-19 2014-04-08 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for the treatment of substance abuse and addiction
TW200812573A (en) 2006-05-19 2008-03-16 Janssen Pharmaceutica Nv Co-therapy for the treatment of epilepsy and related disorders
US20090247617A1 (en) * 2008-03-26 2009-10-01 Abdel-Magid Ahmed F Process for the preparation of benzo-fused heteroaryl sulfamates
US20090247616A1 (en) * 2008-03-26 2009-10-01 Smith-Swintosky Virginia L Use of benzo-fused heterocyle sulfamide derivatives for the treatment of anxiety
MX2010011498A (es) * 2008-04-29 2010-11-12 Nsab Af Neurosearch Sweden Ab Moduladores de neurotransmision de dopamina.
JP2011519839A (ja) * 2008-04-29 2011-07-14 エヌエスエイビー、フィリアル アヴ ノイロサーチ スウェーデン エービー、スヴェーリエ ドーパミン神経伝達のモジュレーター
WO2009133107A1 (en) * 2008-04-29 2009-11-05 Nsab, Filial Af Neurosearch Sweden Ab, Sverige Modulators of dopamine neurotransmission
US8809385B2 (en) 2008-06-23 2014-08-19 Janssen Pharmaceutica Nv Crystalline form of (2S)-(-)-N-(6-chloro-2,3-dihydro-benzo[1,4]dioxin-2-ylmethyl)-sulfamide
US8815939B2 (en) * 2008-07-22 2014-08-26 Janssen Pharmaceutica Nv Substituted sulfamide derivatives
EP2760851A1 (en) 2011-09-29 2014-08-06 Janssen Pharmaceutica, N.V. Process for the preparation of sulfamide derivatives
JP2014528399A (ja) 2011-09-29 2014-10-27 ヤンセン ファーマシューティカ エヌ．ベー． スルファミド誘導体の改善された調製プロセス
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CA2634115A1 (en) 2007-07-05
IL192100A0 (en) 2009-08-03
PL1973540T3 (pl) 2010-04-30
CN101378746B (zh) 2013-07-17
JP5190377B2 (ja) 2013-04-24
KR20080077025A (ko) 2008-08-20
CR10167A (es) 2009-01-16
US8716231B2 (en) 2014-05-06
NI200800169A (es) 2012-05-28
DK1973540T3 (da) 2010-02-01
BRPI0620018A2 (pt) 2011-10-25
PT1973540E (pt) 2010-01-28
CY1109732T1 (el) 2014-09-10
HRP20100007T1 (hr) 2010-02-28
SI1973540T1 (sl) 2010-03-31
NZ569040A (en) 2011-04-29
EP1973540B1 (en) 2009-11-11
US20070155822A1 (en) 2007-07-05
CA2634115C (en) 2014-11-18
EA016302B1 (ru) 2012-04-30
DE602006010442D1 (de) 2009-12-24
EA200870091A1 (ru) 2009-12-30
JP2009520035A (ja) 2009-05-21
ES2335699T3 (es) 2010-03-31
HK1125039A1 (en) 2009-07-31
CN101378746A (zh) 2009-03-04
EP1973540A1 (en) 2008-10-01
RS51249B (sr) 2010-12-31
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MY150903A (en) 2014-03-14
ATE447948T1 (de) 2009-11-15

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