CR10167A - "uso de derivados de sulfamida heterociclica benzo-fusionada para el tratamiento de dolor" - Google Patents

"uso de derivados de sulfamida heterociclica benzo-fusionada para el tratamiento de dolor"

Info

Publication number
CR10167A
CR10167A CR10167A CR10167A CR10167A CR 10167 A CR10167 A CR 10167A CR 10167 A CR10167 A CR 10167A CR 10167 A CR10167 A CR 10167A CR 10167 A CR10167 A CR 10167A
Authority
CR
Costa Rica
Prior art keywords
formula
benzo
fusioned
sulfamide derivatives
pain treatment
Prior art date
Application number
CR10167A
Other languages
English (en)
Inventor
L Smith-Swintosky Virginia
B Reitz Allen
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of CR10167A publication Critical patent/CR10167A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D321/00—Heterocyclic compounds containing rings having two oxygen atoms as the only ring hetero atoms, not provided for by groups C07D317/00 - C07D319/00
    • C07D321/02—Seven-membered rings
    • C07D321/10—Seven-membered rings condensed with carbocyclic rings or ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/357—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having two or more oxygen atoms in the same ring, e.g. crown ethers, guanadrel
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Rheumatology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Pyrane Compounds (AREA)

Abstract

La presente invención es un método para el tratamiento de dolor que comprende la administración a un sujeto que lo necesita de una cantidad terapéuticamente efectiva de uno o más derivados de sulfamida heterocíclica benzo-fusionada novedosos de fórmula (I) o fórmula (II) como se definen aquí; la presente invención se refiere además a métodos para el tratamiento de dolor que comprende la co-terapia con agente o agentes analgésicos y un compuesto de fórmula (I) o fórmula (II) como se definen aquí.
CR10167A 2005-12-19 2008-07-21 "uso de derivados de sulfamida heterociclica benzo-fusionada para el tratamiento de dolor" CR10167A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US75168605P 2005-12-19 2005-12-19
US77381206P 2006-02-15 2006-02-15
US11/612,071 US8716231B2 (en) 2005-12-19 2006-12-18 Use of benzo-fused heterocycle sulfamide derivatives for the treatment of pain

Publications (1)

Publication Number Publication Date
CR10167A true CR10167A (es) 2009-01-16

Family

ID=38007332

Family Applications (1)

Application Number Title Priority Date Filing Date
CR10167A CR10167A (es) 2005-12-19 2008-07-21 "uso de derivados de sulfamida heterociclica benzo-fusionada para el tratamiento de dolor"

Country Status (27)

Country Link
US (1) US8716231B2 (es)
EP (1) EP1973540B1 (es)
JP (1) JP5190377B2 (es)
KR (1) KR20080077025A (es)
CN (1) CN101378746B (es)
AT (1) ATE447948T1 (es)
AU (1) AU2006331734B2 (es)
BR (1) BRPI0620018A2 (es)
CA (1) CA2634115C (es)
CR (1) CR10167A (es)
CY (1) CY1109732T1 (es)
DE (1) DE602006010442D1 (es)
DK (1) DK1973540T3 (es)
EA (1) EA016302B1 (es)
ES (1) ES2335699T3 (es)
HK (1) HK1125039A1 (es)
HR (1) HRP20100007T1 (es)
IL (1) IL192100A0 (es)
MY (1) MY150903A (es)
NI (1) NI200800169A (es)
NO (1) NO20083005L (es)
NZ (1) NZ569040A (es)
PL (1) PL1973540T3 (es)
PT (1) PT1973540E (es)
RS (1) RS51249B (es)
SI (1) SI1973540T1 (es)
WO (1) WO2007075752A1 (es)

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CA2609185A1 (en) * 2005-05-20 2006-11-30 Ahmed F. Abdel-Magid Process for preparation of sulfamide derivatives
US8497298B2 (en) 2005-12-19 2013-07-30 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for lowering lipids and lowering blood glucose levels
US8937096B2 (en) 2005-12-19 2015-01-20 Janssen Pharmaceutica Nv Use of benzo-fused heterocyle sulfamide derivatives for the treatment of mania and bipolar disorder
US8691867B2 (en) 2005-12-19 2014-04-08 Janssen Pharmaceutica Nv Use of benzo-fused heterocycle sulfamide derivatives for the treatment of substance abuse and addiction
US20070155827A1 (en) * 2005-12-19 2007-07-05 Smith-Swintosky Virginia L Use of benzo-fused heterocycle sulfamide derivatives for the treatment of depression
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US20090247617A1 (en) * 2008-03-26 2009-10-01 Abdel-Magid Ahmed F Process for the preparation of benzo-fused heteroaryl sulfamates
US20090247616A1 (en) * 2008-03-26 2009-10-01 Smith-Swintosky Virginia L Use of benzo-fused heterocyle sulfamide derivatives for the treatment of anxiety
MX2010011498A (es) * 2008-04-29 2010-11-12 Nsab Af Neurosearch Sweden Ab Moduladores de neurotransmision de dopamina.
JP2011519839A (ja) * 2008-04-29 2011-07-14 エヌエスエイビー、フィリアル アヴ ノイロサーチ スウェーデン エービー、スヴェーリエ ドーパミン神経伝達のモジュレーター
MX2010011724A (es) * 2008-04-29 2010-11-30 Nsab Af Neurosearch Sweden Ab Moduladores de neurotransmision de dopamina.
MX2011000090A (es) 2008-06-23 2011-03-02 Janssen Pharmaceutica Nv Forma cristalina de (2s)-(-)-n-(6-cloro-2,3-dihidro-benzo[1,4]diox in-2-ilmetil)sulfamida.
US8815939B2 (en) * 2008-07-22 2014-08-26 Janssen Pharmaceutica Nv Substituted sulfamide derivatives
JP2014528953A (ja) 2011-09-29 2014-10-30 ヤンセン ファーマシューティカ エヌ．ベー． スルファミド誘導体の調製プロセス
CA2850015A1 (en) 2011-09-29 2013-04-04 Janssen Pharmaceutica Nv Improved process for the preparation of sulfamide derivatives
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GB2591937B (en) 2018-09-04 2023-06-07 Minerva Neurosciences Inc Methods of using a phenoxypropylamine compound to treat pain
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CA2634115A1 (en) 2007-07-05
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EP1973540B1 (en) 2009-11-11
PT1973540E (pt) 2010-01-28
ATE447948T1 (de) 2009-11-15
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CY1109732T1 (el) 2014-09-10
US20070155822A1 (en) 2007-07-05
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CN101378746A (zh) 2009-03-04
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IL192100A0 (en) 2009-08-03
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EP1973540A1 (en) 2008-10-01
EA016302B1 (ru) 2012-04-30
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AU2006331734A1 (en) 2007-07-05
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