NO20073367L - Makrolider - Google Patents

Makrolider

Info

Publication number
NO20073367L
NO20073367L NO20073367A NO20073367A NO20073367L NO 20073367 L NO20073367 L NO 20073367L NO 20073367 A NO20073367 A NO 20073367A NO 20073367 A NO20073367 A NO 20073367A NO 20073367 L NO20073367 L NO 20073367L
Authority
NO
Norway
Prior art keywords
compounds
methods
macrolides
intermediates
antibacterial
Prior art date
Application number
NO20073367A
Other languages
English (en)
Norwegian (no)
Inventor
Thomas Victor Magee
Mark Edward Flanagan
Louis Stanley Chupak
Takushi Kaneko
Mark Carl Noe
Usa Reilly
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35809765&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20073367(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of NO20073367L publication Critical patent/NO20073367L/no

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Molecular Biology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Tires In General (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NO20073367A 2004-12-21 2007-06-29 Makrolider NO20073367L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US63809704P 2004-12-21 2004-12-21
US71753005P 2005-09-14 2005-09-14
PCT/IB2005/003829 WO2006067589A1 (fr) 2004-12-21 2005-12-12 Macrolides

Publications (1)

Publication Number Publication Date
NO20073367L true NO20073367L (no) 2007-09-05

Family

ID=35809765

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20073367A NO20073367L (no) 2004-12-21 2007-06-29 Makrolider

Country Status (35)

Country Link
US (1) US7462600B2 (fr)
EP (2) EP2233493A1 (fr)
JP (1) JP4111994B1 (fr)
KR (1) KR100897678B1 (fr)
CN (1) CN101120011A (fr)
AP (1) AP2007004026A0 (fr)
AR (1) AR052824A1 (fr)
AT (1) ATE459633T1 (fr)
AU (1) AU2005317735B2 (fr)
BR (1) BRPI0519135A2 (fr)
CA (1) CA2591746A1 (fr)
CR (1) CR9202A (fr)
DE (1) DE602005019786D1 (fr)
DK (1) DK1836211T3 (fr)
EA (1) EA011281B1 (fr)
ES (1) ES2339871T3 (fr)
GE (1) GEP20094834B (fr)
GT (1) GT200500378A (fr)
HN (1) HN2005036113A (fr)
HR (1) HRP20100253T1 (fr)
IL (1) IL183661A0 (fr)
MA (1) MA29108B1 (fr)
MX (1) MX2007007598A (fr)
NL (1) NL1030713C2 (fr)
NO (1) NO20073367L (fr)
PE (1) PE20060948A1 (fr)
PL (1) PL1836211T3 (fr)
PT (1) PT1836211E (fr)
SI (1) SI1836211T1 (fr)
TN (1) TNSN07233A1 (fr)
TW (1) TW200626608A (fr)
UA (1) UA85937C2 (fr)
UY (1) UY29285A1 (fr)
WO (1) WO2006067589A1 (fr)
ZA (1) ZA200705108B (fr)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8367669B2 (en) * 2005-06-15 2013-02-05 Vanderbilt University Inhibitors of hemeprotein-catalyzed lipid peroxidation
US9133212B1 (en) 2005-06-15 2015-09-15 Vanderbilt University Inhibitors of hemeprotein-catalyzed lipid peroxidation
DK1934238T3 (en) 2005-08-24 2017-09-18 Melinta Therapeutics Inc TRIAZOL COMPOUNDS AND METHODS FOR THE PREPARATION AND USE OF THESE
EP2125851B1 (fr) * 2007-03-13 2010-06-23 Pfizer Products Inc. Macrolides à base d'erythromycine
EP2136806A4 (fr) * 2007-03-21 2011-11-23 Creative Antibiotics Sweden Ab Procédé et moyens pour prévenir et inhiber une sécrétion de type iii dans des infections provoquées par une bactérie à gram-négatif
JP5698979B2 (ja) 2007-10-25 2015-04-08 センプラ ファーマシューティカルズ,インコーポレイテッド マクロライド系抗菌剤の調製プロセス
EP2220104A1 (fr) * 2007-10-25 2010-08-25 Sandoz AG Procédé de fabrication de télithromycine
KR101610607B1 (ko) 2007-12-21 2016-04-07 에프. 호프만-라 로슈 아게 헤테로사이클릭 항바이러스 화합물
CA2769551A1 (fr) 2009-08-13 2011-02-17 Basilea Pharmaceutica Ag Nouveaux macrolides et leur utilisation
EP3009442B1 (fr) * 2010-03-22 2019-06-19 Cempra Pharmaceuticals, Inc. Formes cristallines d'un macrolide et leurs utilisations
EP2696873B1 (fr) 2011-04-12 2022-08-03 The United States of America, as represented by The Secretary, Department of Health and Human Services Inhibiteurs du canal anionique de surface de plasmodium pour le traitement ou la prévention de la malaria
CN102558047B (zh) * 2011-12-14 2013-10-30 天津药物研究院药业有限责任公司 3-甲基喹啉的制备方法
RU2658050C2 (ru) 2012-03-27 2018-06-19 Семпра Фармасьютикалз, Инк. Парентеральные составы для введения макролидных антибиотиков
CN104507913B (zh) 2012-07-13 2017-07-28 霍夫曼-拉罗奇有限公司 抗增殖的苯并[b]氮杂*‑2‑酮
KR101612179B1 (ko) * 2013-04-19 2016-04-12 영남대학교 산학협력단 아미도피리딘올 유도체 또는 이의 약제학적 허용가능한 염을 유효성분으로 함유하는 암질환 예방 또는 치료용 약학조성물
TW201534586A (zh) 2013-06-11 2015-09-16 Orion Corp 新穎cyp17抑制劑/抗雄激素劑
CN103739643A (zh) * 2013-12-30 2014-04-23 华东理工大学 利用分子印迹技术对红霉素进行回收分离纯化的方法
CN104230891B (zh) * 2014-08-27 2016-03-30 于宗光 一种托匹司他的制备方法
EP3522896A4 (fr) * 2016-10-04 2020-06-17 Biopharmati SA Cétolides à activité antibactrienne
JP2022534709A (ja) * 2019-06-04 2022-08-03 ヘイガー バイオサイエンシズ,エルエルシー オレキシンアンタゴニストとしてのピラゾール及びイミダゾール誘導体、組成物、並びに方法
CN111793022A (zh) * 2020-04-27 2020-10-20 滁州拜奥生物科技有限公司 一种3-甲基喹啉的制备方法
WO2024050061A2 (fr) * 2022-09-01 2024-03-07 Hager Biosciences, Llc Dérivés de pyrazole et d'imidazole utilisés en tant que modulateurs des récepteurs double d'orexine et d'opioïdes kappa, composition, procédés de traitement de troubles neurologiques et psychiatriques

Family Cites Families (74)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2653899A (en) 1952-04-14 1953-09-29 Lilly Co Eli Erythromycin, its salts, and method of preparation
US2823203A (en) 1954-06-24 1958-02-11 Abbott Lab Method of producing substantially pure erythromycin a
US4331803A (en) 1980-06-04 1982-05-25 Taisho Pharmaceutical Co., Ltd. Novel erythromycin compounds
YU43006B (en) 1981-03-06 1989-02-28 Pliva Pharm & Chem Works Process for preparing n-methyl-11-aza-10-deoxo-10-dihydro erythromycin and derivatives thereof
US4474768A (en) 1982-07-19 1984-10-02 Pfizer Inc. N-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates therefor
US4742049A (en) * 1986-06-04 1988-05-03 Abbott Laboratories Semisynthetic erythromycin antibiotics
US5075289A (en) 1988-06-07 1991-12-24 Abbott Laboratories 9-r-azacyclic erythromycin antibiotics
IE70593B1 (en) 1989-09-29 1996-12-11 Eisai Co Ltd Biphenylmethane derivative the use of it and pharmacological compositions containing same
US5523399A (en) 1991-12-27 1996-06-04 Taisho Pharmaceutical Co., Ltd. 5-O-desosaminylerythronolide derivatives
US5527780A (en) 1992-11-05 1996-06-18 Roussel Uclaf Erythromycin derivatives
FR2697524B1 (fr) * 1992-11-05 1994-12-23 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
FR2719587B1 (fr) 1994-05-03 1996-07-12 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
US5629322A (en) 1994-11-15 1997-05-13 Merck & Co., Inc. Cyclic amidine analogs as inhibitors of nitric oxide synthase
FR2727969B1 (fr) * 1994-12-09 1997-01-17 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
US5747466A (en) * 1995-11-08 1998-05-05 Abbott Laboratories 3-deoxy-3-descladinose derivatives of erythromycins A and B
FR2742757B1 (fr) 1995-12-22 1998-01-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
EP0918783A1 (fr) * 1996-05-07 1999-06-02 Abbott Laboratories Erythromycines 6-o substituees et leur procede de preparation
US5750510A (en) * 1997-04-04 1998-05-12 Abbott Laboratories 3-descladinose-2,3-anhydroerythromycin derivatives
FR2748746B1 (fr) * 1996-05-14 1998-08-14 Hoechst Marion Roussel Inc Nouveau procede d'isomerisation du radical methyle en 10 de derives de l'erythromycine
US6271255B1 (en) 1996-07-05 2001-08-07 Biotica Technology Limited Erythromycins and process for their preparation
FR2751656B1 (fr) * 1996-07-24 1998-10-16 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
CN100441591C (zh) 1996-09-04 2008-12-10 艾博特公司 酮基内酯类化合物,其用途和制备方法以及药用组合物
US5804565A (en) 1996-09-24 1998-09-08 Taisho Pharmaceutical Co., Ltd. Erythromycin A derivatives
CZ180799A3 (cs) 1996-11-27 1999-09-15 Taisho Pharmaceutical Co., Ltd. Deriváty erythromycinu A
AU6421398A (en) 1997-03-24 1998-10-20 Taisho Pharmaceutical Co., Ltd. Erythromycin a derivatives
US6162794A (en) 1997-05-09 2000-12-19 Pfizer Inc. Erythromycin derivatives
US20020025937A1 (en) 2000-03-20 2002-02-28 Yong-Jin Wu 9-oxime erythromycin derivatives
EP0895999A1 (fr) * 1997-08-06 1999-02-10 Pfizer Products Inc. Macrolides antibiotiques substitués C"-4
ZA987689B (en) 1997-09-02 1999-02-24 Abbott Lab 3-descladinose 6-O substituted erythromycin derivatives
US6034069A (en) * 1997-09-30 2000-03-07 Abbott Laboratories 3-'N-modified 6-O-substituted erythromycin ketolide derivatives having antibacterial activity
ZA989835B (en) 1997-10-29 1999-05-05 Taisho Pharmaceutical Co Ltd Erythromycin a derivatives
PA8461401A1 (es) 1997-10-29 2000-05-24 Pfizer Prod Inc Derivados de eritromicina triciclicos
HN1998000159A (es) 1997-10-29 1999-02-09 Monsanto Co Derivados de 9- amino - 3 ceto eritromicina
AP1060A (en) 1998-01-02 2002-04-23 Pfizer Prod Inc Novel erythromycin derivatives.
AP9801420A0 (en) 1998-01-02 1998-12-31 Pfizer Prod Inc Novel macrolides.
DE69919769T2 (de) 1998-03-03 2005-01-27 Pfizer Products Inc., Groton 3,6-Ketal-Makrolidantibiotika
US5955440A (en) * 1998-03-27 1999-09-21 Abbott Laboratories Macrolide LHRH antagonists
WO1999062920A1 (fr) 1998-06-03 1999-12-09 Pfizer Products Inc. Derives 3-keto tricycliques de 6-o-methylerythromycine
JP4573925B2 (ja) * 1998-07-09 2010-11-04 アベンティス・ファーマ・ソシエテ・アノニム 新規のエリスロマイシン誘導体、その製造方法及びその薬剤としての使用
US6020521A (en) 1998-08-26 2000-02-01 Abbott Laboratories Macrolide LHRH antagonists
US6387885B1 (en) * 1998-08-26 2002-05-14 Abbott Laboratories 3′,3′-N-bis-desmethyl-3′-N-cycloalkyl erythromycin derivatives as LHRH antagonists
US6262030B1 (en) 1998-11-03 2001-07-17 Pfizer Inc. Erythromycin derivatives
KR20010083944A (ko) 1998-11-03 2001-09-03 실버스타인 아써 에이. 신규 마크롤라이드 항생물질
EP1137654A1 (fr) * 1998-12-10 2001-10-04 Pfizer Products Inc. Antibiotiques a base de cetolides de carbamate et de carbazate
SI1147121T1 (en) 1999-01-27 2004-04-30 Pfizer Products Inc. Ketolide antibiotics
US6054435A (en) * 1999-03-19 2000-04-25 Abbott Laboratories 6-O-substituted macrolides having antibacterial activity
US6399582B1 (en) * 1999-04-16 2002-06-04 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
MXPA01010524A (es) * 1999-04-16 2002-03-14 Kosan Biosciences Inc Agentes macrolidos anti-infecciosos.
US6939861B2 (en) 1999-04-16 2005-09-06 Kosan Biosciences, Inc. Amido macrolides
US20020061857A1 (en) 1999-04-23 2002-05-23 Yong-Jin Wu 9-amino-3-oxo erythromycin derivatives
US20020077302A1 (en) 1999-04-23 2002-06-20 Yong-Jin Wu Tricyclic erythromycin derivatives
US6355620B1 (en) * 1999-05-14 2002-03-12 Abbott Laboratories C-2 modified erythromycin derivatives
EE200100613A (et) 1999-05-24 2003-02-17 Pfizer Products Inc. 13-metüülerütromütsiini derivaadid
JP2001072669A (ja) 1999-09-07 2001-03-21 Showa Kako Kk 7−クロロ−2,4(1h,3h)−キナゾリンジオンの製造方法
US6569836B2 (en) * 1999-12-02 2003-05-27 Abbott Laboratories 6-O-alkyl-2-nor-2-substituted ketolide derivatives
EP1114826A3 (fr) 1999-12-29 2001-10-31 Pfizer Products Inc. Macrolides antibactériennes et prokinétiques
EP1122261A3 (fr) 2000-01-31 2001-09-26 Pfizer Products Inc. Macrolides antibactériennes à 13 ou 14 chainons
JP2001261694A (ja) 2000-03-06 2001-09-26 Pfizer Prod Inc ケトライド抗生物質
EP1146051A3 (fr) 2000-04-10 2001-10-31 Pfizer Products Inc. Dérivées de l' érythromycine A
US20020061856A1 (en) 2000-04-24 2002-05-23 Yong-Jin Wu Novel tricyclic erythromycin derivatives
TR200401847T4 (tr) 2000-06-30 2004-09-21 Pfizer Products Inc. Makrolit antibiyotikler.
US20020115621A1 (en) 2000-08-07 2002-08-22 Wei-Gu Su Macrolide antibiotics
HUP0302526A2 (hu) 2000-12-21 2003-11-28 Glaxo Group Limited Makrolid vegyületek, eljárás az előállításukra, alkalmazásuk és ezeket tartalmazó gyógyszerkészítmények
US20020132782A1 (en) * 2001-01-18 2002-09-19 Zhenkun Ma 9-amino erythromycin derivatives with antibacterial activity
CA2451391A1 (fr) * 2001-07-03 2003-01-16 Chiron Corporation Macrolides et cetolides d'erythromycine modifiee c12 a activite antibacterienne
US7064110B2 (en) 2002-05-13 2006-06-20 Enanta Pharmaceuticals, Inc. 6-11 bicycle ketolide derivatives
WO2005070918A1 (fr) 2002-05-13 2005-08-04 Enanta Pharmaceuticals, Inc. Procede de preparation de derives bicycliques 6-11 d'erythromycine
PL378841A1 (pl) 2003-04-21 2006-05-29 Daiichi Pharmaceutical Co., Ltd. Pochodna pięcioczłonowego układu heterocyklicznego
US20080287376A1 (en) 2004-07-28 2008-11-20 Mohammad Salman Ketolide Derivatives as Antibacterial Agents
US20090170790A1 (en) 2004-10-25 2009-07-02 Biswajit Das Ketolide derivatives as antibacterial agents
GB0424951D0 (en) 2004-11-11 2004-12-15 Glaxo Group Ltd Novel compounds
JP2008522978A (ja) 2004-12-07 2008-07-03 エナンタ ファーマシューティカルズ インコーポレイテッド 3,6−ビシクロライド
US7312201B2 (en) 2004-12-13 2007-12-25 Enanta Pharmaceuticals, Inc. Tetracyclic bicyclolides
WO2006065721A2 (fr) 2004-12-13 2006-06-22 Enanta Pharmaceuticals, Inc. Bicyclolides de 11, 12-lactone

Also Published As

Publication number Publication date
TNSN07233A1 (fr) 2008-11-21
SI1836211T1 (sl) 2010-04-30
ES2339871T3 (es) 2010-05-26
ZA200705108B (en) 2009-01-28
KR100897678B1 (ko) 2009-05-14
PE20060948A1 (es) 2006-10-11
NL1030713A1 (nl) 2006-06-22
WO2006067589A1 (fr) 2006-06-29
AP2007004026A0 (en) 2007-06-30
AR052824A1 (es) 2007-04-04
EA200701113A1 (ru) 2007-12-28
JP4111994B1 (ja) 2008-07-02
DE602005019786D1 (de) 2010-04-15
ATE459633T1 (de) 2010-03-15
HN2005036113A (es) 2010-12-06
NL1030713C2 (nl) 2006-12-12
US7462600B2 (en) 2008-12-09
EP1836211A1 (fr) 2007-09-26
US20060135447A1 (en) 2006-06-22
CN101120011A (zh) 2008-02-06
MA29108B1 (fr) 2007-12-03
DK1836211T3 (da) 2010-05-17
KR20070089191A (ko) 2007-08-30
EA011281B1 (ru) 2009-02-27
UY29285A1 (es) 2006-07-31
EP1836211B1 (fr) 2010-03-03
PT1836211E (pt) 2010-04-08
UA85937C2 (uk) 2009-03-10
CA2591746A1 (fr) 2006-06-29
AU2005317735B2 (en) 2009-06-04
HRP20100253T1 (hr) 2010-06-30
CR9202A (es) 2007-07-16
BRPI0519135A2 (pt) 2008-12-23
JP2008524319A (ja) 2008-07-10
IL183661A0 (en) 2007-09-20
EP2233493A1 (fr) 2010-09-29
AU2005317735A1 (en) 2006-06-29
GEP20094834B (en) 2009-11-25
GT200500378A (es) 2006-11-28
MX2007007598A (es) 2007-07-25
PL1836211T3 (pl) 2010-07-30
TW200626608A (en) 2006-08-01

Similar Documents

Publication Publication Date Title
NO20073367L (no) Makrolider
NO20070566L (no) Azin-karboksamider som antikreftmiddel
NO20073719L (no) Kjemiske forbindelser
NO20070199L (no) Substituerte kinazoloner som anti-kreftmidler
NO20056192L (no) Kapaseinhibitorer og anvendelse derav
NO20082124L (no) Bifenyloksyeddiksyrederivater for behandling av respiratorisk sykdom
NO20074703L (no) Antibakterielle piperidinderivater
WO2007044085A3 (fr) Composes heteroaryle et leurs utilisations en tant qu'agents therapeutiques
NO20070224L (no) 2-karbamid-4-fenyltiazolderivater, fremstilling og terapeutisk anvendelse derav
NO20081729L (no) Nye diazaspiroalkaner og deres anvendelse for behandling av CCR8-medierte sykdommer
NO20080338L (no) Forbindelser for behandling av multilegemiddelresistente bakterielle infeksjoner
NO20081844L (no) Terapeutiske forbindelser
NO20082538L (no) Stabiliserte lantankarbonatsammensetninger
NO20091605L (no) Pyridinonforbindelser
WO2007046867A3 (fr) Derives de piperidine et leurs utilisations comme agents therapeutiques
BRPI0517567A (pt) composto ou um sal, solvato, ou derivado fisiologicamente funcional farmaceuticamente aceitável do mesmo, composição farmacêutica, usos de um composto ou um sal, solvato, ou derivado fisiologicamente funcional farmaceuticamente aceitável do mesmo e de uma composição farmacêutica, e, processo para preparar um composto
NO20061743L (no) Kinazolinderivater
NO20076675L (no) Aminopiperidinquinoliner og deres azaisosteriske analoger med antibakteriell aktivitet
NO20076019L (no) Utvortes preparat for hud
NO20091683L (no) Kjemiske forbindelser
NO20070487L (no) 3-aminocyklopentankarboksamider som modulatorer av kjemokinreseptorer.
WO2007009724A3 (fr) Derives de pyrazoline substitues cycloalkane, fabrication et utilisation comme medicaments
MX2007011009A (es) Compuestos de piperidina 3,4,5-substituidos.
WO2006096444A3 (fr) Composes chimiques
DE60206911D1 (de) Imidazol-2-carbonsäureamid derivate als raf-kinase-inhibitoren

Legal Events

Date Code Title Description
FC2A Withdrawal, rejection or dismissal of laid open patent application