NO20076675L - Aminopiperidinquinoliner og deres azaisosteriske analoger med antibakteriell aktivitet - Google Patents
Aminopiperidinquinoliner og deres azaisosteriske analoger med antibakteriell aktivitetInfo
- Publication number
- NO20076675L NO20076675L NO20076675A NO20076675A NO20076675L NO 20076675 L NO20076675 L NO 20076675L NO 20076675 A NO20076675 A NO 20076675A NO 20076675 A NO20076675 A NO 20076675A NO 20076675 L NO20076675 L NO 20076675L
- Authority
- NO
- Norway
- Prior art keywords
- antibacterial activity
- medicaments
- humans
- warm
- bacterial infections
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
- C07D491/056—Ortho-condensed systems with two or more oxygen atoms as ring hetero atoms in the oxygen-containing ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/4738—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
- A61K31/4745—Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Communicable Diseases (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Abstract
Foreliggende oppfinnelse angår forbindelser som demonstrerer antibakteriell aktivitet, fremgangsmåter for deres fremstilling, farmasøytiske sammensetninger som inneholder dem som aktiv ingrediens, deres anvendelse som medikamenter og deres anvendelse ved fremstilling av medikamenter for anvendelse ved behandling av bakterielle infeksjoner hos varmblodige dyr slik som mennesker. Spesielt angår foreliggende oppfinnelse forbindelser anvendelige for behandling av bakterielle infeksjoner hos varmblodige dyr slik som mennesker, mer spesielt anvendelse av disse forbindelsene ved fremstilling av medikamenter for anvendelse ved behandling av bakterielle infeksjoner hos varmblodige dyr slik som mennesker.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US68403005P | 2005-05-24 | 2005-05-24 | |
PCT/GB2006/001889 WO2006125974A1 (en) | 2005-05-24 | 2006-05-23 | Aminopiperidine quinolines and their azaisosteric analogues with antibacterial activity |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20076675L true NO20076675L (no) | 2007-12-27 |
Family
ID=36685663
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20076675A NO20076675L (no) | 2005-05-24 | 2007-12-27 | Aminopiperidinquinoliner og deres azaisosteriske analoger med antibakteriell aktivitet |
Country Status (14)
Country | Link |
---|---|
US (1) | US20090131444A1 (no) |
EP (1) | EP1891078A1 (no) |
JP (1) | JP2008542249A (no) |
KR (1) | KR20080016577A (no) |
CN (1) | CN101258157A (no) |
AU (1) | AU2006250987A1 (no) |
BR (1) | BRPI0609887A2 (no) |
CA (1) | CA2608072A1 (no) |
IL (1) | IL187134A0 (no) |
MX (1) | MX2007014507A (no) |
NO (1) | NO20076675L (no) |
RU (1) | RU2007147413A (no) |
WO (1) | WO2006125974A1 (no) |
ZA (1) | ZA200709870B (no) |
Families Citing this family (31)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
MY150958A (en) | 2005-06-16 | 2014-03-31 | Astrazeneca Ab | Compounds for the treatment of multi-drug resistant bacterial infections |
CA2643962A1 (en) * | 2006-03-10 | 2007-09-20 | Actelion Pharmaceuticals Ltd | Antibiotic compounds |
WO2007115947A1 (en) | 2006-04-06 | 2007-10-18 | Glaxo Group Limited | Pyrrolo-quinoxalinone derivatives as antibacterials |
JP5171618B2 (ja) | 2006-05-26 | 2013-03-27 | 富山化学工業株式会社 | 新規な複素環化合物またはその塩ならびにその中間体 |
BRPI0712430A2 (pt) * | 2006-06-08 | 2012-07-03 | Speedel Experimenta Ag | piperidinas 2,5-di-substitìdas. |
AU2008240764C1 (en) * | 2007-04-20 | 2011-10-20 | Glaxo Group Limited | Tricyclic nitrogen containing compounds as antibacterial agents |
ATE520687T1 (de) | 2007-06-15 | 2011-09-15 | Actelion Pharmaceuticals Ltd | 3-amino-6-(1-amino-ethyl)-tetrahydropyranderiva e |
MX2010008922A (es) | 2008-02-20 | 2010-09-07 | Actelion Pharmaceuticals Ltd | Compuestos antibioticos azatriciclicos. |
BRPI0920895A8 (pt) | 2008-10-07 | 2017-12-26 | Actelion Pharmaceuticals Ltd | Compostos antibióticos de oxazolidinona tricíclica |
WO2010043714A1 (en) | 2008-10-17 | 2010-04-22 | Glaxo Group Limited | Tricyclic nitrogen compounds used as antibacterials |
ES2435596T3 (es) | 2008-12-12 | 2013-12-20 | Actelion Pharmaceuticals Ltd. | Derivados de 5-amino-2-(1-hidroxi-etil)-tetrahidropirano |
US20120053350A1 (en) * | 2009-04-30 | 2012-03-01 | Ian Mangion | Preparation of alkyl esters of n-protected oxo-azacycloalkylcarboxylic acids |
SG10201507846YA (en) * | 2010-04-02 | 2015-10-29 | Senomyx Inc | Sweet flavor modifier |
US8829191B2 (en) * | 2011-06-17 | 2014-09-09 | Melanie Simone Ronsheim | Processes for preparing heterocyclic compounds including trans-7-oxo-6-(sulphooxy)-1,6-diazabicyclo[3,2,1]octane-2-carboxamide and salts thereof |
MY179876A (en) | 2011-08-12 | 2020-11-18 | Firmenich Incorporated | Sweet flavor modifier |
US8933232B2 (en) | 2012-03-30 | 2015-01-13 | Cubist Pharmaceuticals, Inc. | 1,3,4-oxadiazole and 1,3,4-thiadiazole beta-lactamase inhibitors |
AR090844A1 (es) | 2012-04-27 | 2014-12-10 | Actelion Pharmaceuticals Ltd | Proceso para elaborar derivados de naftiridina |
WO2014152996A1 (en) | 2013-03-14 | 2014-09-25 | Cubist Pharmaceuticals, Inc. | Crystalline form of a beta-lactamase inhibitor |
US9120796B2 (en) | 2013-10-02 | 2015-09-01 | Cubist Pharmaceuticals, Inc. | B-lactamase inhibitor picoline salt |
CN103613530B (zh) * | 2013-12-02 | 2015-08-19 | 江苏弘和药物研发有限公司 | 一种芴甲氧羰基-3-哌啶醇的合成方法 |
EP3915975A1 (en) * | 2013-12-27 | 2021-12-01 | API Corporation | Method for producing 5-hydroxypiperidine-2-carboxylic acid |
EA031589B1 (ru) | 2014-08-22 | 2019-01-31 | Глэксосмитклайн Интеллекчуал Проперти Дивелопмент Лимитед | Трициклические азотсодержащие соединения для лечения инфекции, вызываемой neisseria gonorrhoeae |
WO2016073251A1 (en) | 2014-11-07 | 2016-05-12 | Senomyx, Inc. | Substituted 4-amino-5-(cyclohexyloxy)quinoline-3-carboxylic acids as sweet flavor modifiers |
UY36851A (es) * | 2015-08-16 | 2017-03-31 | Glaxosmithkline Ip Dev Ltd | Compuestos para uso en aplicaciones antibacterianas |
HUE049547T2 (hu) | 2016-06-08 | 2020-10-28 | Acraf | Új baktériumellenes szerek |
EP4295852A2 (en) | 2016-07-13 | 2023-12-27 | Syros Pharmaceuticals, Inc. | Piperidine derivatives as inhibitors of cyclin dependent kinase 7 (cdk7) |
JP7210483B2 (ja) | 2017-06-30 | 2023-01-23 | バイエル・アニマル・ヘルス・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツング | 新規アザキノリン誘導体 |
MX2020001352A (es) | 2017-08-09 | 2020-03-20 | Denali Therapeutics Inc | Compuestos, composiciones y metodos. |
SI3676297T1 (sl) * | 2017-09-01 | 2023-12-29 | Denali Therapeutics Inc. | Spojine, sestavki in postopki |
TWI802591B (zh) | 2017-09-14 | 2023-05-21 | 日商第一三共股份有限公司 | 具有環狀構造的化合物 |
CR20210426A (es) | 2019-02-13 | 2021-09-30 | Denali Therapeutics Inc | Compuestos, composiciones y métodos |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB9822450D0 (en) * | 1998-10-14 | 1998-12-09 | Smithkline Beecham Plc | Medicaments |
DE60125373T2 (de) * | 2000-07-26 | 2007-10-18 | Smithkline Beecham P.L.C., Brentford | Aminopiperidin chinoline und ihre azaisosteren analoga mit antibakterieller wirkung |
JP2004509885A (ja) * | 2000-09-21 | 2004-04-02 | スミスクライン ビーチャム パブリック リミテッド カンパニー | 抗菌薬としてのキノリン誘導体 |
JP4887297B2 (ja) * | 2004-09-24 | 2012-02-29 | アクテリオン ファーマシューティカルズ リミテッド | 新規二環式抗生物質 |
-
2006
- 2006-05-23 WO PCT/GB2006/001889 patent/WO2006125974A1/en active Application Filing
- 2006-05-23 BR BRPI0609887-8A patent/BRPI0609887A2/pt not_active Application Discontinuation
- 2006-05-23 CA CA002608072A patent/CA2608072A1/en not_active Abandoned
- 2006-05-23 RU RU2007147413/04A patent/RU2007147413A/ru not_active Application Discontinuation
- 2006-05-23 US US11/914,799 patent/US20090131444A1/en not_active Abandoned
- 2006-05-23 MX MX2007014507A patent/MX2007014507A/es not_active Application Discontinuation
- 2006-05-23 AU AU2006250987A patent/AU2006250987A1/en not_active Abandoned
- 2006-05-23 EP EP06743966A patent/EP1891078A1/en not_active Withdrawn
- 2006-05-23 JP JP2008512908A patent/JP2008542249A/ja active Pending
- 2006-05-23 CN CNA2006800266719A patent/CN101258157A/zh active Pending
- 2006-05-23 KR KR1020077027342A patent/KR20080016577A/ko not_active Application Discontinuation
-
2007
- 2007-11-04 IL IL187134A patent/IL187134A0/en unknown
- 2007-11-15 ZA ZA200709870A patent/ZA200709870B/xx unknown
- 2007-12-27 NO NO20076675A patent/NO20076675L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
BRPI0609887A2 (pt) | 2011-10-11 |
RU2007147413A (ru) | 2009-06-27 |
IL187134A0 (en) | 2008-02-09 |
EP1891078A1 (en) | 2008-02-27 |
WO2006125974A1 (en) | 2006-11-30 |
KR20080016577A (ko) | 2008-02-21 |
JP2008542249A (ja) | 2008-11-27 |
AU2006250987A1 (en) | 2006-11-30 |
US20090131444A1 (en) | 2009-05-21 |
MX2007014507A (es) | 2008-02-07 |
CN101258157A (zh) | 2008-09-03 |
ZA200709870B (en) | 2008-11-26 |
CA2608072A1 (en) | 2006-11-30 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC2A | Withdrawal, rejection or dismissal of laid open patent application |