NO20064000L - Heteroarylkoblede pyrazoloderivater - Google Patents
Heteroarylkoblede pyrazoloderivaterInfo
- Publication number
- NO20064000L NO20064000L NO20064000A NO20064000A NO20064000L NO 20064000 L NO20064000 L NO 20064000L NO 20064000 A NO20064000 A NO 20064000A NO 20064000 A NO20064000 A NO 20064000A NO 20064000 L NO20064000 L NO 20064000L
- Authority
- NO
- Norway
- Prior art keywords
- heteroeryl
- linked
- pyrazolo derivatives
- pyrazolo
- derivatives
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/04—Drugs for disorders of the respiratory system for throat disorders
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/16—Central respiratory analeptics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/02—Drugs for genital or sexual disorders; Contraceptives for disorders of the vagina
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
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- A—HUMAN NECESSITIES
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- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
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- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Abstract
Forbindelser med formel I hvor A, B, X, Y, Z, k, R1, R2 og R3 er de definert her og preparater omfattende disse. Foreliggende oppfinnelse tilveiebringer også metoder for fremstilling av forbindelser med formel I og anvendelse av dem ved behandling av p38 medierte lidelser hos en pasient.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US54864204P | 2004-02-27 | 2004-02-27 | |
PCT/EP2005/001815 WO2005085248A1 (en) | 2004-02-27 | 2005-02-22 | Heteroaryl-fused pyrazolo derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20064000L true NO20064000L (no) | 2006-09-22 |
Family
ID=34919387
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20064000A NO20064000L (no) | 2004-02-27 | 2006-09-06 | Heteroarylkoblede pyrazoloderivater |
Country Status (16)
Country | Link |
---|---|
US (1) | US7452880B2 (no) |
EP (1) | EP1720878A1 (no) |
JP (1) | JP2007523936A (no) |
KR (1) | KR100844864B1 (no) |
CN (1) | CN1934111A (no) |
AR (1) | AR048069A1 (no) |
AU (1) | AU2005219517A1 (no) |
BR (1) | BRPI0508220A (no) |
CA (1) | CA2558109A1 (no) |
IL (1) | IL177259A0 (no) |
MX (1) | MXPA06009462A (no) |
NO (1) | NO20064000L (no) |
RU (1) | RU2006134021A (no) |
TW (1) | TW200533671A (no) |
WO (1) | WO2005085248A1 (no) |
ZA (1) | ZA200606615B (no) |
Families Citing this family (77)
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EP1675858A2 (en) * | 2003-09-03 | 2006-07-05 | Neurogen Corporation | 5-aryl-pyrazolo [4,3-d] pyrimidines, pyridines, and pyrazines and related compounds |
WO2005085249A1 (en) * | 2004-02-27 | 2005-09-15 | F. Hoffmann-La Roche Ag | Fused derivatives of pyrazole |
AU2005219517A1 (en) | 2004-02-27 | 2005-09-15 | F.Hoffmann-La Roche Ag | Heteroaryl-fused pyrazolo derivatives |
US7405220B2 (en) * | 2004-06-09 | 2008-07-29 | Hoffmann-La Roche Inc. | Pyrazolopyrimidines |
CN101098872B (zh) | 2004-11-22 | 2012-09-05 | 沃泰克斯药物股份有限公司 | 可用作蛋白激酶抑制剂的吡咯并吡嗪和吡唑并吡嗪 |
GB0427604D0 (en) * | 2004-12-16 | 2005-01-19 | Novartis Ag | Organic compounds |
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JP2009506007A (ja) * | 2005-08-25 | 2009-02-12 | エフ.ホフマン−ラ ロシュ アーゲー | p38MAPキナーゼ阻害剤及びその使用方法 |
KR101011958B1 (ko) | 2005-08-25 | 2011-01-31 | 에프. 호프만-라 로슈 아게 | p38 MAP 키나아제 저해제로서의 융합형 피라졸 |
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2005
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- 2005-02-22 EP EP05715442A patent/EP1720878A1/en not_active Withdrawn
- 2005-02-22 WO PCT/EP2005/001815 patent/WO2005085248A1/en active Application Filing
- 2005-02-22 JP JP2007500126A patent/JP2007523936A/ja active Pending
- 2005-02-22 BR BRPI0508220-0A patent/BRPI0508220A/pt not_active IP Right Cessation
- 2005-02-22 CA CA002558109A patent/CA2558109A1/en not_active Abandoned
- 2005-02-22 CN CNA2005800063457A patent/CN1934111A/zh active Pending
- 2005-02-22 MX MXPA06009462A patent/MXPA06009462A/es not_active Application Discontinuation
- 2005-02-22 KR KR1020067017108A patent/KR100844864B1/ko not_active IP Right Cessation
- 2005-02-22 RU RU2006134021/04A patent/RU2006134021A/ru unknown
- 2005-02-23 TW TW094105458A patent/TW200533671A/zh unknown
- 2005-02-24 AR ARP050100665A patent/AR048069A1/es unknown
- 2005-02-25 US US11/065,890 patent/US7452880B2/en not_active Expired - Fee Related
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2006
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- 2006-08-08 ZA ZA200606615A patent/ZA200606615B/xx unknown
- 2006-09-06 NO NO20064000A patent/NO20064000L/no not_active Application Discontinuation
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AR048069A1 (es) | 2006-03-29 |
MXPA06009462A (es) | 2007-03-15 |
JP2007523936A (ja) | 2007-08-23 |
CN1934111A (zh) | 2007-03-21 |
US20050203091A1 (en) | 2005-09-15 |
EP1720878A1 (en) | 2006-11-15 |
US7452880B2 (en) | 2008-11-18 |
RU2006134021A (ru) | 2008-04-10 |
KR20060117359A (ko) | 2006-11-16 |
IL177259A0 (en) | 2006-12-10 |
BRPI0508220A (pt) | 2007-07-17 |
ZA200606615B (en) | 2008-02-27 |
TW200533671A (en) | 2005-10-16 |
CA2558109A1 (en) | 2005-09-15 |
WO2005085248A1 (en) | 2005-09-15 |
KR100844864B1 (ko) | 2008-07-09 |
AU2005219517A1 (en) | 2005-09-15 |
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