NO20063371L - Aminosubstituerte diaryl[a,d]cykloheptenanaloger som muscarinagonister og fremgangsmater for behandling av neuropsykiatriske lidelser - Google Patents

Aminosubstituerte diaryl[a,d]cykloheptenanaloger som muscarinagonister og fremgangsmater for behandling av neuropsykiatriske lidelser

Info

Publication number
NO20063371L
NO20063371L NO20063371A NO20063371A NO20063371L NO 20063371 L NO20063371 L NO 20063371L NO 20063371 A NO20063371 A NO 20063371A NO 20063371 A NO20063371 A NO 20063371A NO 20063371 L NO20063371 L NO 20063371L
Authority
NO
Norway
Prior art keywords
methods
amino
cycloheptene
analogues
substituted diaryl
Prior art date
Application number
NO20063371A
Other languages
English (en)
Norwegian (no)
Inventor
Fredrik Ek
Roger Olsson
Jorgen Ohlsson
Original Assignee
Acadia Pharm Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Acadia Pharm Inc filed Critical Acadia Pharm Inc
Publication of NO20063371L publication Critical patent/NO20063371L/no

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/38[b, e]- or [b, f]-condensed with six-membered rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Anesthesiology (AREA)
  • Psychology (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
NO20063371A 2003-12-22 2006-07-20 Aminosubstituerte diaryl[a,d]cykloheptenanaloger som muscarinagonister og fremgangsmater for behandling av neuropsykiatriske lidelser NO20063371L (no)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US53192703P 2003-12-22 2003-12-22
US54809004P 2004-02-24 2004-02-24
US54860404P 2004-02-27 2004-02-27
PCT/US2004/043224 WO2005063254A2 (fr) 2003-12-22 2004-12-21 Analogues de diaryl[a,d]cycloheptene amino substitues utilises comme agonistes muscariniques, et procedes de traitement de troubles neuropsychiatriques

Publications (1)

Publication Number Publication Date
NO20063371L true NO20063371L (no) 2006-09-22

Family

ID=34743692

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20063371A NO20063371L (no) 2003-12-22 2006-07-20 Aminosubstituerte diaryl[a,d]cykloheptenanaloger som muscarinagonister og fremgangsmater for behandling av neuropsykiatriske lidelser

Country Status (23)

Country Link
US (5) US7550454B2 (fr)
EP (2) EP1696931B1 (fr)
JP (1) JP2007534656A (fr)
KR (1) KR101157881B1 (fr)
CN (1) CN101962369A (fr)
AT (1) ATE426405T1 (fr)
AU (1) AU2004308955B2 (fr)
BR (1) BRPI0417749A (fr)
CA (1) CA2550735A1 (fr)
CY (1) CY1109171T1 (fr)
DE (1) DE602004020263D1 (fr)
DK (1) DK1696931T3 (fr)
ES (1) ES2324713T3 (fr)
HK (1) HK1095092A1 (fr)
IL (1) IL176447A0 (fr)
MX (1) MXPA06007244A (fr)
NO (1) NO20063371L (fr)
NZ (1) NZ547911A (fr)
PL (1) PL1696931T3 (fr)
PT (1) PT1696931E (fr)
SG (1) SG133606A1 (fr)
SI (1) SI1696931T1 (fr)
WO (1) WO2005063254A2 (fr)

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US7622461B2 (en) 2009-11-24
NZ547911A (en) 2010-06-25
US7517871B2 (en) 2009-04-14
AU2004308955A1 (en) 2005-07-14
EP1696931A2 (fr) 2006-09-06
PT1696931E (pt) 2009-06-12
CY1109171T1 (el) 2014-07-02
ES2324713T3 (es) 2009-08-13
EP2088147A1 (fr) 2009-08-12
ATE426405T1 (de) 2009-04-15
KR101157881B1 (ko) 2012-07-06
PL1696931T3 (pl) 2009-10-30
HK1095092A1 (en) 2007-04-27
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US20060199798A1 (en) 2006-09-07
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US20100129473A1 (en) 2010-05-27
US7550454B2 (en) 2009-06-23
WO2005063254A3 (fr) 2005-09-15
BRPI0417749A (pt) 2007-04-10
CA2550735A1 (fr) 2005-07-14
WO2005063254A2 (fr) 2005-07-14
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US7491715B2 (en) 2009-02-17
US20060194784A1 (en) 2006-08-31
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