NO20043068L - Kondenserte heterocykliske succinimidforbindelser og analoger derav, modulatorer for nukleaer hormonreseptorfunksjon - Google Patents
Kondenserte heterocykliske succinimidforbindelser og analoger derav, modulatorer for nukleaer hormonreseptorfunksjonInfo
- Publication number
- NO20043068L NO20043068L NO20043068A NO20043068A NO20043068L NO 20043068 L NO20043068 L NO 20043068L NO 20043068 A NO20043068 A NO 20043068A NO 20043068 A NO20043068 A NO 20043068A NO 20043068 L NO20043068 L NO 20043068L
- Authority
- NO
- Norway
- Prior art keywords
- modulators
- analogs
- hormone receptor
- receptor function
- condensed heterocyclic
- Prior art date
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
- C07D491/18—Bridged systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D495/18—Bridged systems
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/22—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains four or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/08—Bridged systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Endocrinology (AREA)
- Diabetes (AREA)
- Reproductive Health (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Physical Education & Sports Medicine (AREA)
- Gynecology & Obstetrics (AREA)
- Neurosurgery (AREA)
- Immunology (AREA)
- Psychiatry (AREA)
- Dermatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Rheumatology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Pain & Pain Management (AREA)
- Pregnancy & Childbirth (AREA)
- Hospice & Palliative Care (AREA)
- Cardiology (AREA)
- Urology & Nephrology (AREA)
- Addiction (AREA)
- Nutrition Science (AREA)
- Heart & Thoracic Surgery (AREA)
- Emergency Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US2511601A | 2001-12-19 | 2001-12-19 | |
PCT/US2002/040598 WO2003062241A1 (en) | 2001-12-19 | 2002-12-18 | Fused heterocyclic succinimidecompounds and analogs thereof, modulators of nuclear hormone receptor function |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20043068L true NO20043068L (no) | 2004-09-08 |
Family
ID=27609007
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20043068A NO20043068L (no) | 2001-12-19 | 2004-07-16 | Kondenserte heterocykliske succinimidforbindelser og analoger derav, modulatorer for nukleaer hormonreseptorfunksjon |
Country Status (31)
Country | Link |
---|---|
EP (1) | EP1458723B1 (de) |
JP (1) | JP2005523257A (de) |
KR (1) | KR20040086248A (de) |
CN (1) | CN1589271A (de) |
AR (1) | AR037950A1 (de) |
AT (1) | ATE411319T1 (de) |
AU (1) | AU2002361785B2 (de) |
BR (1) | BR0215281A (de) |
CA (1) | CA2471342A1 (de) |
CO (1) | CO5640082A2 (de) |
DE (1) | DE60229435D1 (de) |
DK (1) | DK1458723T3 (de) |
ES (1) | ES2314127T3 (de) |
GE (1) | GEP20063817B (de) |
HR (1) | HRP20040567A2 (de) |
HU (1) | HUP0402554A3 (de) |
IL (1) | IL162547A0 (de) |
IS (1) | IS7324A (de) |
MX (1) | MXPA04005876A (de) |
NO (1) | NO20043068L (de) |
NZ (1) | NZ533471A (de) |
PL (1) | PL370904A1 (de) |
PT (1) | PT1458723E (de) |
RU (1) | RU2330038C2 (de) |
SI (1) | SI1458723T1 (de) |
TW (1) | TWI263640B (de) |
UA (1) | UA78265C2 (de) |
UY (1) | UY27595A1 (de) |
WO (1) | WO2003062241A1 (de) |
YU (1) | YU53604A (de) |
ZA (1) | ZA200404812B (de) |
Families Citing this family (39)
Publication number | Priority date | Publication date | Assignee | Title |
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US7202264B2 (en) | 2003-01-31 | 2007-04-10 | Isis Pharmaceuticals, Inc. | Supports for oligomer synthesis |
FR2860793A1 (fr) * | 2003-10-14 | 2005-04-15 | Entomed | Composes derives de norcantharidine, leurs procedes de preparation, les compositions les contenant et leurs utilisations |
DK1692139T3 (da) * | 2003-11-13 | 2013-03-11 | Isis Pharmaceuticals Inc | 5,6-dihydroxy-isoindol-derivater som linkere til fastfasesyntese af oligomerer |
US7625921B2 (en) | 2004-01-16 | 2009-12-01 | Bristol-Myers Squibb Company | Modulators of the glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof |
US7273881B2 (en) | 2004-01-16 | 2007-09-25 | Bristol-Myers Squibb Company | Modulators of glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof |
US7605264B2 (en) | 2004-01-16 | 2009-10-20 | Bristol-Myers Squibb Company | Heterocyclic modulators of the glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof |
US7326728B2 (en) | 2004-01-16 | 2008-02-05 | Bristol-Myers Squibb Company | Modulators of glucocorticoid receptor, AP-1, and/or NF-κβ activity and use thereof |
US7253283B2 (en) | 2004-01-16 | 2007-08-07 | Bristol-Myers Squibb Company | Tricyclic modulators of the glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof |
US7569689B2 (en) | 2004-01-16 | 2009-08-04 | Bristol-Myers Squibb Company | Modulators of the glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof |
EA200601461A1 (ru) * | 2004-03-17 | 2007-02-27 | Пфайзер Продактс, Инк. | Новые производные бензил(иден)лактама |
US7642273B2 (en) | 2005-01-13 | 2010-01-05 | Bristol-Myers Squibb Company | Modulators of the glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof |
US7317024B2 (en) | 2005-01-13 | 2008-01-08 | Bristol-Myers Squibb Co. | Heterocyclic modulators of the glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof |
US7361654B2 (en) | 2005-01-13 | 2008-04-22 | Bristol-Myers Squibb Co. | Substituted heteroaryl amide modulators of glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof |
US7411071B2 (en) | 2005-01-13 | 2008-08-12 | Bristol-Myers Squibb Company | Modulators of the glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof |
ATE478852T1 (de) * | 2005-09-09 | 2010-09-15 | Schering Corp | Neue 4-cyano-, 4-amino-, und 4- aminomethylderivative von pyrazoloä1,5- aüpyridinen, pyrazoloä1,5-cüpyrimidinen und 2h- indazolverbindungen und 5-cyano-, 5-amino- und 5- aminomethylderivative von imidazoä1,2-aüpyridinen,und imidazoä1,5-aüpyrazinverbindungen als inhibitoren der cyclinabhänggen kinase |
WO2008042571A2 (en) | 2006-09-29 | 2008-04-10 | Smithkline Beecham Corporation | Substituted indole compounds |
WO2008157291A2 (en) * | 2007-06-15 | 2008-12-24 | Bristol-Myers Squibb Company | CRYSTALLINE FORMS OF (3Aα, 4β, 5α, 7β, 7Aα)-4-(OCTAHYDRO-5-ETHYLSULFONAMIDO-4,7-DIMETHYL-1,3-DIOXO-4,7-EPOXY-2H-ISOINDOL-2-YL)-2-(TRIFLUOROMETHYL)BENZONITRILE AND METHOD OF PREPARATION |
EP2426117A4 (de) * | 2009-04-30 | 2012-09-19 | Sumitomo Chemical Co | Thiophenderivat |
EP2455370A1 (de) | 2009-07-17 | 2012-05-23 | Shionogi&Co., Ltd. | Pharmazeutisches produkt mit lactam- oder benzen-sulfonamid-verbindung |
EP2475366A1 (de) | 2009-09-11 | 2012-07-18 | Bayer Pharma Aktiengesellschaft | Substituierte (heteroarylmethyl)-thiohydantoine als tumormittel |
SI2523731T1 (sl) * | 2010-01-14 | 2019-02-28 | Novartis Ag | Uporaba sredstva, ki modificira adrenalni hormon |
WO2014111871A1 (en) | 2013-01-17 | 2014-07-24 | Aurigene Discovery Technologies Limited | 4,5-dihydroisoxazole derivatives as nampt inhibitors |
EP2991994B1 (de) * | 2013-05-01 | 2018-08-15 | Vitae Pharmaceuticals, Inc. | Thiazolopyrrolidininhibitoren von ror-gamma |
JP6156074B2 (ja) * | 2013-11-08 | 2017-07-05 | 住友化学株式会社 | スクシンイミド化合物及びその用途 |
EA031804B1 (ru) | 2014-02-03 | 2019-02-28 | Вайтаи Фармасьютиклз, Инк. | Дигидропирролопиридиновые ингибиторы ror-гамма |
US9663515B2 (en) | 2014-11-05 | 2017-05-30 | Vitae Pharmaceuticals, Inc. | Dihydropyrrolopyridine inhibitors of ROR-gamma |
PL3372584T3 (pl) * | 2014-12-19 | 2021-07-05 | Aragon Pharmaceuticals, Inc. | Sposób wytwarzania związku diarylotiohydantoiny |
KR102564925B1 (ko) * | 2015-01-20 | 2023-08-07 | 아비나스 오퍼레이션스, 인코포레이티드 | 안드로겐 수용체의 표적화된 분해를 위한 화합물 및 방법 |
US20170327469A1 (en) | 2015-01-20 | 2017-11-16 | Arvinas, Inc. | Compounds and methods for the targeted degradation of androgen receptor |
ES2856931T3 (es) | 2015-08-05 | 2021-09-28 | Vitae Pharmaceuticals Llc | Moduladores de ROR-gamma |
EP3377482B1 (de) | 2015-11-20 | 2021-05-12 | Vitae Pharmaceuticals, LLC | Modulatoren von ror-gamma |
TW202220968A (zh) | 2016-01-29 | 2022-06-01 | 美商維它藥物有限責任公司 | ROR-γ調節劑 |
EP3562818B1 (de) | 2016-12-29 | 2022-05-18 | ENYO Pharma | Thiophenederivate als antivirale agenzien |
WO2019018975A1 (en) | 2017-07-24 | 2019-01-31 | Vitae Pharmaceuticals, Inc. | INHIBITORS OF ROR GAMMA |
AR112461A1 (es) | 2017-07-24 | 2019-10-30 | Vitae Pharmaceuticals Inc | PROCESOS PARA LA PRODUCCIÓN DE SALES Y FORMAS CRISTALINAS DE INHIBIDORES DE RORg |
EP4121044A4 (de) * | 2020-03-20 | 2024-03-13 | University Of Southern California | Androgenrezeptorregulierung durch kleinmolekülige enantiomere |
CN114848795B (zh) * | 2021-02-03 | 2023-04-14 | 四川大学 | RORa蛋白及其激动剂在制备抗衰老药物中的应用 |
WO2023154939A2 (en) * | 2022-02-14 | 2023-08-17 | The Johns Hopkins University | Gcpii inhibition for the treatment of sarcopenia and aging |
WO2024059200A1 (en) | 2022-09-14 | 2024-03-21 | Halia Therapeutics, Inc. | Nek7 inhibitors |
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US4892943A (en) * | 1985-10-16 | 1990-01-09 | American Home Products Corporation | Fused bicyclic imides with psychotropic activity |
JPS63170383A (ja) * | 1987-02-26 | 1988-07-14 | Nippon Zeon Co Ltd | 脂環式ジカルボン酸イミド化合物 |
WO1991006297A1 (en) * | 1989-10-27 | 1991-05-16 | The Du Pont Merck Pharmaceutical Company | (n-phthalimidoalkyl) piperidines |
ES2221040T3 (es) * | 1996-10-25 | 2004-12-16 | Daiichi Pharmaceutical Co., Ltd. | Derivados de amina triciclicos. |
FR2764890B1 (fr) * | 1997-06-24 | 1999-08-27 | Adir | Nouveaux derives chromeniques, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
JP2002533345A (ja) * | 1998-12-22 | 2002-10-08 | イーライ・リリー・アンド・カンパニー | 置換三環式化合物 |
CA2413417A1 (en) * | 2000-06-28 | 2002-01-03 | Bristol-Myers Squibb Company | Selective androgen receptor modulators and methods for their identification, design and use |
CN1307181C (zh) * | 2000-09-19 | 2007-03-28 | 布里斯托尔-迈尔斯斯奎布公司 | 核激素受体功能的调节剂稠合杂环琥珀酰亚胺化合物及其类似物 |
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