NO20026167L - Kondenserte cykliske forbindelser som modulatorer av nukle¶r hormon reseptor funksjon - Google Patents

Kondenserte cykliske forbindelser som modulatorer av nukle¶r hormon reseptor funksjon

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Publication number
NO20026167L
NO20026167L NO20026167A NO20026167A NO20026167L NO 20026167 L NO20026167 L NO 20026167L NO 20026167 A NO20026167 A NO 20026167A NO 20026167 A NO20026167 A NO 20026167A NO 20026167 L NO20026167 L NO 20026167L
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NO
Norway
Prior art keywords
modulators
hormone receptor
cyclic compounds
receptor function
nuclear hormone
Prior art date
Application number
NO20026167A
Other languages
English (en)
Other versions
NO20026167D0 (no
Inventor
Mark Ernest Salvati
James Aaron Balog
Weifang Shan
Soren Giese
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of NO20026167L publication Critical patent/NO20026167L/no
Publication of NO20026167D0 publication Critical patent/NO20026167D0/no

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    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
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US20030114420A1 (en) * 2000-06-28 2003-06-19 Salvati Mark E. Fused cyclic modulators of nuclear hormone receptor function
CN1395467A (zh) * 2000-09-07 2003-02-05 美国拜尔公司 用作孕酮受体结合剂的环和非环脒以及包含它们的药物组合物
DE10162375A1 (de) * 2001-12-19 2003-07-10 Bayer Ag Bicyclische N-Aryl-amide
WO2003053358A2 (en) * 2001-12-19 2003-07-03 Bristol-Myers Squibb Company Fused heterocyclic compounds and analogs thereof: modulators of nuclear hormone receptor function
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US7199125B2 (en) 2003-10-02 2007-04-03 Bristol-Myers Squibb Company Spiro-cyclic compounds useful as anti-inflammatory agents
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US9409856B2 (en) 2005-11-28 2016-08-09 Gtx, Inc. Estrogen receptor ligands and methods of use thereof
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JP5816087B2 (ja) 2008-08-29 2015-11-18 エンメエッセディ・イタリア・エッセ・エッレ・エッレ Ｓｍｏアンタゴニストとしての飽和二環式複素環誘導体
US9427418B2 (en) 2009-02-23 2016-08-30 Gtx, Inc. Estrogen receptor ligands and methods of use thereof
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EP1299385A2 (en) 2003-04-09
CA2413683A1 (en) 2002-01-03
HUP0303165A2 (hu) 2003-12-29
NZ523802A (en) 2005-11-25
JP2004515462A (ja) 2004-05-27
NO20026167D0 (no) 2002-12-20
MXPA02012563A (es) 2003-05-14
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