ATE399163T1 - Tricyclische modulatoren von nuklearen steroidhormonrezeptoren - Google Patents

Tricyclische modulatoren von nuklearen steroidhormonrezeptoren

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Publication number
ATE399163T1
ATE399163T1 AT04811084T AT04811084T ATE399163T1 AT E399163 T1 ATE399163 T1 AT E399163T1 AT 04811084 T AT04811084 T AT 04811084T AT 04811084 T AT04811084 T AT 04811084T AT E399163 T1 ATE399163 T1 AT E399163T1
Authority
AT
Austria
Prior art keywords
tricyclic
modulators
steroid hormone
hormone receptors
nuclear steroid
Prior art date
Application number
AT04811084T
Other languages
English (en)
Inventor
Konstantinos Gavardinas
Jonathan Green
Prabhakar Jadhav
Donald Matthews
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Application granted granted Critical
Publication of ATE399163T1 publication Critical patent/ATE399163T1/de

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/26—Oxygen atoms
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AT04811084T 2003-12-19 2004-12-08 Tricyclische modulatoren von nuklearen steroidhormonrezeptoren ATE399163T1 (de)

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US53128303P 2003-12-19 2003-12-19

Publications (1)

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ATE399163T1 true ATE399163T1 (de) 2008-07-15

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US (1) US7803814B2 (de)
EP (1) EP1697350B1 (de)
JP (1) JP4846596B2 (de)
CN (1) CN1918151A (de)
AR (1) AR046951A1 (de)
AT (1) ATE399163T1 (de)
AU (1) AU2004312293A1 (de)
BR (1) BRPI0416882A (de)
CA (1) CA2549053C (de)
CY (1) CY1108309T1 (de)
DE (1) DE602004014640D1 (de)
DK (1) DK1697350T3 (de)
ES (1) ES2308296T3 (de)
IL (1) IL175996A0 (de)
MX (1) MXPA06007055A (de)
NO (1) NO20063329L (de)
PL (1) PL1697350T3 (de)
PT (1) PT1697350E (de)
SI (1) SI1697350T1 (de)
WO (1) WO2005066161A1 (de)
ZA (1) ZA200604889B (de)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
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TW200400816A (en) * 2002-06-26 2004-01-16 Lilly Co Eli Tricyclic steroid hormone nuclear receptor modulators
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US20070037788A1 (en) 2007-02-15
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SI1697350T1 (sl) 2008-12-31
JP4846596B2 (ja) 2011-12-28
JP2007515431A (ja) 2007-06-14
MXPA06007055A (es) 2007-01-30
IL175996A0 (en) 2006-10-05
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PT1697350E (pt) 2008-09-18
WO2005066161A1 (en) 2005-07-21
CA2549053A1 (en) 2005-07-21
ZA200604889B (en) 2007-11-28
CN1918151A (zh) 2007-02-21
AU2004312293A1 (en) 2005-07-21
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AR046951A1 (es) 2006-01-04
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