NO20063329L - Tricykliske steroidhormone nukleaer reseptormodulatorer - Google Patents
Tricykliske steroidhormone nukleaer reseptormodulatorerInfo
- Publication number
- NO20063329L NO20063329L NO20063329A NO20063329A NO20063329L NO 20063329 L NO20063329 L NO 20063329L NO 20063329 A NO20063329 A NO 20063329A NO 20063329 A NO20063329 A NO 20063329A NO 20063329 L NO20063329 L NO 20063329L
- Authority
- NO
- Norway
- Prior art keywords
- receptor modulators
- nuclear receptor
- steroid hormone
- compound
- formula
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/26—Oxygen atoms
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- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
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Abstract
Foreliggende oppfinnelse tilveiebringer en forbindelse med Formel (I): eller et farmasøytisk akseptabelt salt derav; farmasøytiske sammensetninger som innbefatter en effektiv mengde av en forbindelse med Formel (I) i kombinasjon med en egnet bærer, fortynningsmiddel eller eksipient; fremgangsmåter for behandling av fysiologiske forstyrrelser, særlig kongestiv hjertesvikt, hypertensjon, reumatoid artritt eller inflammasjon, som innbefatter administrering til en pasient som trenger det av en effektiv mengde av en forbindelse med Formel (I).
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US53128303P | 2003-12-19 | 2003-12-19 | |
PCT/US2004/038233 WO2005066161A1 (en) | 2003-12-19 | 2004-12-08 | Tricyclic steroid hormone nuclear receptor modulators |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20063329L true NO20063329L (no) | 2006-09-14 |
Family
ID=34748755
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20063329A NO20063329L (no) | 2003-12-19 | 2006-07-18 | Tricykliske steroidhormone nukleaer reseptormodulatorer |
Country Status (21)
Country | Link |
---|---|
US (1) | US7803814B2 (no) |
EP (1) | EP1697350B1 (no) |
JP (1) | JP4846596B2 (no) |
CN (1) | CN1918151A (no) |
AR (1) | AR046951A1 (no) |
AT (1) | ATE399163T1 (no) |
AU (1) | AU2004312293A1 (no) |
BR (1) | BRPI0416882A (no) |
CA (1) | CA2549053C (no) |
CY (1) | CY1108309T1 (no) |
DE (1) | DE602004014640D1 (no) |
DK (1) | DK1697350T3 (no) |
ES (1) | ES2308296T3 (no) |
IL (1) | IL175996A0 (no) |
MX (1) | MXPA06007055A (no) |
NO (1) | NO20063329L (no) |
PL (1) | PL1697350T3 (no) |
PT (1) | PT1697350E (no) |
SI (1) | SI1697350T1 (no) |
WO (1) | WO2005066161A1 (no) |
ZA (1) | ZA200604889B (no) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW200400816A (en) * | 2002-06-26 | 2004-01-16 | Lilly Co Eli | Tricyclic steroid hormone nuclear receptor modulators |
JP2008525484A (ja) * | 2004-12-23 | 2008-07-17 | アサーシス, インク. | 肥満症およびその他のcns障害の治療のためのヒスタミン3受容体阻害剤としての4−ピペリジノール第三級アミン |
DE102005022020A1 (de) * | 2005-05-12 | 2006-11-23 | Merckle Gmbh | Dibenzocycloheptanverbindungen und pharmazeutische Mittel, welche diese Verbindungen enthalten |
TWI385161B (zh) | 2006-02-02 | 2013-02-11 | Mitsubishi Tanabe Pharma Corp | 含氮雜雙環化合物 |
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PE20091057A1 (es) | 2007-12-19 | 2009-07-20 | Lilly Co Eli | Antagonistas del receptor mineralcorticoide y metodos de uso |
WO2009089312A1 (en) * | 2008-01-11 | 2009-07-16 | Eli Lilly And Company | (e)-n-{3- [1-(8-fluoro-11h-10-oxa-1-aza-dibenzo [a,d] cycl0hepten-5ylidene)-propyl]-phenyl }-methynsulfon amide as glucocorticoid receptor modulator for the treatment of rheumatoid |
JPWO2010001990A1 (ja) | 2008-07-03 | 2011-12-22 | 協和発酵キリン株式会社 | 四環系化合物 |
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WO2011081173A1 (ja) * | 2009-12-29 | 2011-07-07 | 協和発酵キリン株式会社 | 四環系化合物 |
US8957052B2 (en) | 2010-05-10 | 2015-02-17 | Universite Paris Descartes | Methods and compositions for the treatment of fluid accumulation in and/or under the retina |
EP2582365B1 (en) | 2010-06-16 | 2019-03-20 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Compositions for stimulating reepithelialisation during wound healing |
JP2013542255A (ja) * | 2010-11-10 | 2013-11-21 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | ミネラルコルチコイド受容体アンタゴニストとしてのピリジル尿素 |
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FR2603713B1 (fr) * | 1986-09-10 | 1992-07-24 | Canon Kk | Derive nouveau de 5h-dibenzo(a,d)cycloheptane-(ene)ylidene, son procede de production et support electrophotographique photosensible le contenant |
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JPH0446352A (ja) | 1990-06-14 | 1992-02-17 | Minolta Camera Co Ltd | 感光体 |
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JP2006508893A (ja) * | 2002-03-15 | 2006-03-16 | イーライ・リリー・アンド・カンパニー | ステロイドホルモン核内レセプターモジュレーターとしてのジヒドロインドール−2−オン誘導体 |
TW200400816A (en) * | 2002-06-26 | 2004-01-16 | Lilly Co Eli | Tricyclic steroid hormone nuclear receptor modulators |
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2004
- 2004-12-08 CN CNA2004800418534A patent/CN1918151A/zh active Pending
- 2004-12-08 PL PL04811084T patent/PL1697350T3/pl unknown
- 2004-12-08 MX MXPA06007055A patent/MXPA06007055A/es unknown
- 2004-12-08 US US10/576,761 patent/US7803814B2/en not_active Expired - Fee Related
- 2004-12-08 DE DE602004014640T patent/DE602004014640D1/de active Active
- 2004-12-08 ES ES04811084T patent/ES2308296T3/es active Active
- 2004-12-08 WO PCT/US2004/038233 patent/WO2005066161A1/en active Application Filing
- 2004-12-08 EP EP04811084A patent/EP1697350B1/en not_active Not-in-force
- 2004-12-08 SI SI200430840T patent/SI1697350T1/sl unknown
- 2004-12-08 AU AU2004312293A patent/AU2004312293A1/en not_active Abandoned
- 2004-12-08 DK DK04811084T patent/DK1697350T3/da active
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- 2004-12-08 CA CA2549053A patent/CA2549053C/en not_active Expired - Fee Related
- 2004-12-08 PT PT04811084T patent/PT1697350E/pt unknown
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- 2004-12-08 BR BRPI0416882-8A patent/BRPI0416882A/pt not_active Application Discontinuation
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2006
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Also Published As
Publication number | Publication date |
---|---|
MXPA06007055A (es) | 2007-01-30 |
EP1697350B1 (en) | 2008-06-25 |
CA2549053C (en) | 2012-08-28 |
IL175996A0 (en) | 2006-10-05 |
DE602004014640D1 (de) | 2008-08-07 |
WO2005066161A1 (en) | 2005-07-21 |
US20070037788A1 (en) | 2007-02-15 |
EP1697350A1 (en) | 2006-09-06 |
AR046951A1 (es) | 2006-01-04 |
PT1697350E (pt) | 2008-09-18 |
DK1697350T3 (da) | 2008-10-13 |
CA2549053A1 (en) | 2005-07-21 |
AU2004312293A1 (en) | 2005-07-21 |
US7803814B2 (en) | 2010-09-28 |
ATE399163T1 (de) | 2008-07-15 |
JP4846596B2 (ja) | 2011-12-28 |
ZA200604889B (en) | 2007-11-28 |
CY1108309T1 (el) | 2014-02-12 |
PL1697350T3 (pl) | 2008-11-28 |
JP2007515431A (ja) | 2007-06-14 |
BRPI0416882A (pt) | 2007-02-27 |
CN1918151A (zh) | 2007-02-21 |
ES2308296T3 (es) | 2008-12-01 |
SI1697350T1 (sl) | 2008-12-31 |
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