SI1697350T1 - Modulatorji jedrnega receptorja tricikličnih steroidnih hormonov - Google Patents

Modulatorji jedrnega receptorja tricikličnih steroidnih hormonov

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Publication number
SI1697350T1
SI1697350T1 SI200430840T SI200430840T SI1697350T1 SI 1697350 T1 SI1697350 T1 SI 1697350T1 SI 200430840 T SI200430840 T SI 200430840T SI 200430840 T SI200430840 T SI 200430840T SI 1697350 T1 SI1697350 T1 SI 1697350T1
Authority
SI
Slovenia
Prior art keywords
receptor modulators
nuclear receptor
steroid hormone
hormone nuclear
tricyclic steroid
Prior art date
Application number
SI200430840T
Other languages
English (en)
Inventor
Konstantinos Gavardinas
Jonathan Edward Green
Prabhakar Kondaji Jadhav
Donald P Matthews
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of SI1697350T1 publication Critical patent/SI1697350T1/sl

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    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/26Oxygen atoms
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  • Bioinformatics & Cheminformatics (AREA)
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SI200430840T 2003-12-19 2004-12-08 Modulatorji jedrnega receptorja tricikličnih steroidnih hormonov SI1697350T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US53128303P 2003-12-19 2003-12-19
EP04811084A EP1697350B1 (en) 2003-12-19 2004-12-08 Tricyclic steroid hormone nuclear receptor modulators
PCT/US2004/038233 WO2005066161A1 (en) 2003-12-19 2004-12-08 Tricyclic steroid hormone nuclear receptor modulators

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SI1697350T1 true SI1697350T1 (sl) 2008-12-31

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US (1) US7803814B2 (sl)
EP (1) EP1697350B1 (sl)
JP (1) JP4846596B2 (sl)
CN (1) CN1918151A (sl)
AR (1) AR046951A1 (sl)
AT (1) ATE399163T1 (sl)
AU (1) AU2004312293A1 (sl)
BR (1) BRPI0416882A (sl)
CA (1) CA2549053C (sl)
CY (1) CY1108309T1 (sl)
DE (1) DE602004014640D1 (sl)
DK (1) DK1697350T3 (sl)
ES (1) ES2308296T3 (sl)
IL (1) IL175996A0 (sl)
MX (1) MXPA06007055A (sl)
NO (1) NO20063329L (sl)
PL (1) PL1697350T3 (sl)
PT (1) PT1697350E (sl)
SI (1) SI1697350T1 (sl)
WO (1) WO2005066161A1 (sl)
ZA (1) ZA200604889B (sl)

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TW200400816A (en) * 2002-06-26 2004-01-16 Lilly Co Eli Tricyclic steroid hormone nuclear receptor modulators
CA2594264C (en) * 2004-12-23 2013-05-21 Athersys, Inc. 4-piperidinol tertiary amines as histamine 3 receptor inhibitors for the treatment of obesity and other cns disorders
DE102005022020A1 (de) * 2005-05-12 2006-11-23 Merckle Gmbh Dibenzocycloheptanverbindungen und pharmazeutische Mittel, welche diese Verbindungen enthalten
TWI385161B (zh) 2006-02-02 2013-02-11 Mitsubishi Tanabe Pharma Corp 含氮雜雙環化合物
US8034940B2 (en) 2006-08-09 2011-10-11 Bristol-Myers Squibb Company Modulators of glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof
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