DK1697350T3 - Tricykliske modulatorer af cellekernereceptor for steroidhormon - Google Patents
Tricykliske modulatorer af cellekernereceptor for steroidhormonInfo
- Publication number
- DK1697350T3 DK1697350T3 DK04811084T DK04811084T DK1697350T3 DK 1697350 T3 DK1697350 T3 DK 1697350T3 DK 04811084 T DK04811084 T DK 04811084T DK 04811084 T DK04811084 T DK 04811084T DK 1697350 T3 DK1697350 T3 DK 1697350T3
- Authority
- DK
- Denmark
- Prior art keywords
- tricyclic
- modulators
- nuclear receptor
- steroid hormone
- cell nuclear
- Prior art date
Links
Classifications
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/26—Oxygen atoms
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- Health & Medical Sciences (AREA)
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- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Hematology (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Immunology (AREA)
- Physical Education & Sports Medicine (AREA)
- Dermatology (AREA)
- Neurosurgery (AREA)
- Rheumatology (AREA)
- Obesity (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Pulmonology (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Emergency Medicine (AREA)
- Vascular Medicine (AREA)
- Hospice & Palliative Care (AREA)
- Urology & Nephrology (AREA)
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Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US53128303P | 2003-12-19 | 2003-12-19 | |
PCT/US2004/038233 WO2005066161A1 (en) | 2003-12-19 | 2004-12-08 | Tricyclic steroid hormone nuclear receptor modulators |
Publications (1)
Publication Number | Publication Date |
---|---|
DK1697350T3 true DK1697350T3 (da) | 2008-10-13 |
Family
ID=34748755
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK04811084T DK1697350T3 (da) | 2003-12-19 | 2004-12-08 | Tricykliske modulatorer af cellekernereceptor for steroidhormon |
Country Status (21)
Country | Link |
---|---|
US (1) | US7803814B2 (da) |
EP (1) | EP1697350B1 (da) |
JP (1) | JP4846596B2 (da) |
CN (1) | CN1918151A (da) |
AR (1) | AR046951A1 (da) |
AT (1) | ATE399163T1 (da) |
AU (1) | AU2004312293A1 (da) |
BR (1) | BRPI0416882A (da) |
CA (1) | CA2549053C (da) |
CY (1) | CY1108309T1 (da) |
DE (1) | DE602004014640D1 (da) |
DK (1) | DK1697350T3 (da) |
ES (1) | ES2308296T3 (da) |
IL (1) | IL175996A0 (da) |
MX (1) | MXPA06007055A (da) |
NO (1) | NO20063329L (da) |
PL (1) | PL1697350T3 (da) |
PT (1) | PT1697350E (da) |
SI (1) | SI1697350T1 (da) |
WO (1) | WO2005066161A1 (da) |
ZA (1) | ZA200604889B (da) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW200400816A (en) * | 2002-06-26 | 2004-01-16 | Lilly Co Eli | Tricyclic steroid hormone nuclear receptor modulators |
CA2594264C (en) * | 2004-12-23 | 2013-05-21 | Athersys, Inc. | 4-piperidinol tertiary amines as histamine 3 receptor inhibitors for the treatment of obesity and other cns disorders |
DE102005022020A1 (de) * | 2005-05-12 | 2006-11-23 | Merckle Gmbh | Dibenzocycloheptanverbindungen und pharmazeutische Mittel, welche diese Verbindungen enthalten |
TWI385161B (zh) | 2006-02-02 | 2013-02-11 | Mitsubishi Tanabe Pharma Corp | 含氮雜雙環化合物 |
US8034940B2 (en) | 2006-08-09 | 2011-10-11 | Bristol-Myers Squibb Company | Modulators of glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof |
AP2527A (en) | 2006-10-31 | 2012-12-06 | Pfizer Prod Inc | Pyrazoline compounds as mineralocorticoid receptorantagonists |
TWI431010B (zh) | 2007-12-19 | 2014-03-21 | Lilly Co Eli | 礦皮質素受體拮抗劑及使用方法 |
AU2009204155A1 (en) * | 2008-01-11 | 2009-07-16 | Eli Lilly And Company | (E)-N-{3- [1-(8-Fluoro-11H-10-oxa-1-aza-dibenzo [a,d] cyclohepten-5ylidene)-propyl]-phenyl }-methynsulfon amide as glucocorticoid receptor modulator for the treatment of rheumatoid |
EP2308880A4 (en) * | 2008-07-03 | 2012-06-06 | Kyowa Hakko Kirin Co Ltd | TETRACYCLIC CONNECTION |
MX2011009506A (es) * | 2009-03-12 | 2011-09-28 | Lilly Co Eli | Antagonista del receptor mineralcorticoide y metodos de uso. |
WO2011081173A1 (ja) * | 2009-12-29 | 2011-07-07 | 協和発酵キリン株式会社 | 四環系化合物 |
US8957052B2 (en) | 2010-05-10 | 2015-02-17 | Universite Paris Descartes | Methods and compositions for the treatment of fluid accumulation in and/or under the retina |
US9241944B2 (en) | 2010-06-16 | 2016-01-26 | Institut National De La Santé Et De La Recherche Médicale (Inserm) | Methods and compositions for stimulating reepithelialisation during wound healing |
JP2013542255A (ja) * | 2010-11-10 | 2013-11-21 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | ミネラルコルチコイド受容体アンタゴニストとしてのピリジル尿素 |
TW201311678A (zh) * | 2011-08-03 | 2013-03-16 | Kyowa Hakko Kirin Co Ltd | 二苯并氧呯衍生物 |
JP2024513538A (ja) * | 2021-04-12 | 2024-03-25 | インパクト セラピューティクス (シャンハイ), インコーポレイテッド | Parp阻害剤としての置換融合二環式化合物及びその使用 |
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DE3730258A1 (de) * | 1986-09-10 | 1988-04-07 | Canon Kk | Elektrophotographisches lichtempfindliches aufzeichnungsmaterial, 5h-dibenzo(a,d)cycloheptanylidenderivat, 5h-dibenzo(a,d)cycloheptenylidenderivat und verfahren zu ihrer herstellung |
JPH01161245A (ja) | 1987-12-18 | 1989-06-23 | Canon Inc | 電子写真感光体 |
CA1338625C (en) * | 1988-06-09 | 1996-10-01 | Kyowa Hakko Kogyo Co., Ltd. | Tricyclic compounds |
US5093210A (en) * | 1989-06-30 | 1992-03-03 | Ricoh Company, Ltd. | Electroluminescent device |
JPH0446352A (ja) | 1990-06-14 | 1992-02-17 | Minolta Camera Co Ltd | 感光体 |
CO4980885A1 (es) | 1997-12-29 | 2000-11-27 | Ortho Mcneil Pharm Inc | Compuestos de trifenilpropanamida utiles en el tratamiento de inflamaciones y metodos para preparar dicho compuesto |
EP1154997A4 (en) | 1999-01-26 | 2002-11-04 | Dana Farber Cancer Inst Inc | PHARMACEUTICALLY ACTIVE COMPOUNDS AND METHODS OF USE |
JP4434740B2 (ja) * | 2001-12-19 | 2010-03-17 | ブリストル−マイヤーズ スクイブ カンパニー | 核ホルモン受容体機能の調節剤である、縮合ヘテロ環化合物およびその類似体 |
CA2478172A1 (en) | 2002-03-15 | 2003-09-25 | Eli Lilly And Company | Dihydroindol-2-one derivatives as steroid hormone nuclear receptor modulators |
TW200400816A (en) | 2002-06-26 | 2004-01-16 | Lilly Co Eli | Tricyclic steroid hormone nuclear receptor modulators |
-
2004
- 2004-12-08 CN CNA2004800418534A patent/CN1918151A/zh active Pending
- 2004-12-08 PL PL04811084T patent/PL1697350T3/pl unknown
- 2004-12-08 AT AT04811084T patent/ATE399163T1/de not_active IP Right Cessation
- 2004-12-08 JP JP2006545655A patent/JP4846596B2/ja not_active Expired - Fee Related
- 2004-12-08 AU AU2004312293A patent/AU2004312293A1/en not_active Abandoned
- 2004-12-08 WO PCT/US2004/038233 patent/WO2005066161A1/en active Application Filing
- 2004-12-08 MX MXPA06007055A patent/MXPA06007055A/es unknown
- 2004-12-08 ES ES04811084T patent/ES2308296T3/es active Active
- 2004-12-08 DE DE602004014640T patent/DE602004014640D1/de active Active
- 2004-12-08 SI SI200430840T patent/SI1697350T1/sl unknown
- 2004-12-08 CA CA2549053A patent/CA2549053C/en not_active Expired - Fee Related
- 2004-12-08 PT PT04811084T patent/PT1697350E/pt unknown
- 2004-12-08 EP EP04811084A patent/EP1697350B1/en not_active Not-in-force
- 2004-12-08 DK DK04811084T patent/DK1697350T3/da active
- 2004-12-08 US US10/576,761 patent/US7803814B2/en not_active Expired - Fee Related
- 2004-12-08 BR BRPI0416882-8A patent/BRPI0416882A/pt not_active Application Discontinuation
- 2004-12-17 AR ARP040104730A patent/AR046951A1/es unknown
-
2006
- 2006-05-29 IL IL175996A patent/IL175996A0/en unknown
- 2006-06-13 ZA ZA200604889A patent/ZA200604889B/en unknown
- 2006-07-18 NO NO20063329A patent/NO20063329L/no not_active Application Discontinuation
-
2008
- 2008-09-03 CY CY20081100936T patent/CY1108309T1/el unknown
Also Published As
Publication number | Publication date |
---|---|
PT1697350E (pt) | 2008-09-18 |
AU2004312293A1 (en) | 2005-07-21 |
CA2549053A1 (en) | 2005-07-21 |
US20070037788A1 (en) | 2007-02-15 |
SI1697350T1 (sl) | 2008-12-31 |
ES2308296T3 (es) | 2008-12-01 |
DE602004014640D1 (de) | 2008-08-07 |
CA2549053C (en) | 2012-08-28 |
AR046951A1 (es) | 2006-01-04 |
ATE399163T1 (de) | 2008-07-15 |
MXPA06007055A (es) | 2007-01-30 |
JP4846596B2 (ja) | 2011-12-28 |
EP1697350A1 (en) | 2006-09-06 |
EP1697350B1 (en) | 2008-06-25 |
CY1108309T1 (el) | 2014-02-12 |
NO20063329L (no) | 2006-09-14 |
ZA200604889B (en) | 2007-11-28 |
PL1697350T3 (pl) | 2008-11-28 |
WO2005066161A1 (en) | 2005-07-21 |
JP2007515431A (ja) | 2007-06-14 |
US7803814B2 (en) | 2010-09-28 |
IL175996A0 (en) | 2006-10-05 |
CN1918151A (zh) | 2007-02-21 |
BRPI0416882A (pt) | 2007-02-27 |
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