PT1697350E - Moduladores do receptor nuclear da hormona esteróide tricíclica - Google Patents

Moduladores do receptor nuclear da hormona esteróide tricíclica Download PDF

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Publication number
PT1697350E
PT1697350E PT04811084T PT04811084T PT1697350E PT 1697350 E PT1697350 E PT 1697350E PT 04811084 T PT04811084 T PT 04811084T PT 04811084 T PT04811084 T PT 04811084T PT 1697350 E PT1697350 E PT 1697350E
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PT
Portugal
Prior art keywords
receptor modulators
nuclear receptor
steroid hormone
hormone nuclear
tricyclic steroid
Prior art date
Application number
PT04811084T
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English (en)
Inventor
Donald P Matthews
Konstantinos Gavardinas
Jonathan Edward Green
Prabhakar Kondaji Jadhav
Original Assignee
Lilly Co Eli
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Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of PT1697350E publication Critical patent/PT1697350E/pt

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    • C07D235/02Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/26Oxygen atoms
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PT04811084T 2003-12-19 2004-12-08 Moduladores do receptor nuclear da hormona esteróide tricíclica PT1697350E (pt)

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PT1697350E true PT1697350E (pt) 2008-09-18

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US (1) US7803814B2 (pt)
EP (1) EP1697350B1 (pt)
JP (1) JP4846596B2 (pt)
CN (1) CN1918151A (pt)
AR (1) AR046951A1 (pt)
AT (1) ATE399163T1 (pt)
AU (1) AU2004312293A1 (pt)
BR (1) BRPI0416882A (pt)
CA (1) CA2549053C (pt)
CY (1) CY1108309T1 (pt)
DE (1) DE602004014640D1 (pt)
DK (1) DK1697350T3 (pt)
ES (1) ES2308296T3 (pt)
IL (1) IL175996A0 (pt)
MX (1) MXPA06007055A (pt)
NO (1) NO20063329L (pt)
PL (1) PL1697350T3 (pt)
PT (1) PT1697350E (pt)
SI (1) SI1697350T1 (pt)
WO (1) WO2005066161A1 (pt)
ZA (1) ZA200604889B (pt)

Families Citing this family (16)

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TW200400816A (en) * 2002-06-26 2004-01-16 Lilly Co Eli Tricyclic steroid hormone nuclear receptor modulators
JP2008525484A (ja) * 2004-12-23 2008-07-17 アサーシス, インク. 肥満症およびその他のcns障害の治療のためのヒスタミン3受容体阻害剤としての4−ピペリジノール第三級アミン
DE102005022020A1 (de) * 2005-05-12 2006-11-23 Merckle Gmbh Dibenzocycloheptanverbindungen und pharmazeutische Mittel, welche diese Verbindungen enthalten
TWI385161B (zh) 2006-02-02 2013-02-11 Mitsubishi Tanabe Pharma Corp 含氮雜雙環化合物
US8034940B2 (en) 2006-08-09 2011-10-11 Bristol-Myers Squibb Company Modulators of glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof
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