NO20042792L - Nye peptider som NS3-serinproteaseinhibitorer for hepatitt C-virus - Google Patents

Nye peptider som NS3-serinproteaseinhibitorer for hepatitt C-virus

Info

Publication number
NO20042792L
NO20042792L NO20042792A NO20042792A NO20042792L NO 20042792 L NO20042792 L NO 20042792L NO 20042792 A NO20042792 A NO 20042792A NO 20042792 A NO20042792 A NO 20042792A NO 20042792 L NO20042792 L NO 20042792L
Authority
NO
Norway
Prior art keywords
hepatitis
virus
protease inhibitors
serine protease
new peptides
Prior art date
Application number
NO20042792A
Other languages
English (en)
Norwegian (no)
Inventor
Jesse K Wong
Viyyoor Moopil Girijavallabhan
Anil K Saksena
Raymond G Lovey
Russell E Pike
Yi-Tsung Liu
Marguerita S L Lim-Wilby
Ashit K Ganguly
Jinping L Mccormick
Ashok Arasappan
Srikanth Venkatraman
F George Njoroge
Tin-Yau Chan
Stephane L Bogen
Haiyan Wang
Tejal N Parekh
Patrick A Pinto
Bama Santhanam
Henry A Vaccaro
Scott Jeffrey Kemp
Original Assignee
Ustamura Susan Y
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ustamura Susan Y filed Critical Ustamura Susan Y
Publication of NO20042792L publication Critical patent/NO20042792L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0802—Tripeptides with the first amino acid being neutral
    • C07K5/0804—Tripeptides with the first amino acid being neutral and aliphatic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/0202—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-X-X-C(=0)-, X being an optionally substituted carbon atom or a heteroatom, e.g. beta-amino acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0802—Tripeptides with the first amino acid being neutral
    • C07K5/0812—Tripeptides with the first amino acid being neutral and aromatic or cycloaliphatic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0827—Tripeptides containing heteroatoms different from O, S, or N
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/02—Linear peptides containing at least one abnormal peptide link
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Virology (AREA)
  • Engineering & Computer Science (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Crystallography & Structural Chemistry (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
NO20042792A 2002-01-18 2004-07-02 Nye peptider som NS3-serinproteaseinhibitorer for hepatitt C-virus NO20042792L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10/052,386 US7244721B2 (en) 2000-07-21 2002-01-18 Peptides as NS3-serine protease inhibitors of hepatitis C virus
PCT/US2003/001430 WO2003062265A2 (en) 2002-01-18 2003-01-16 Novel peptides as ns3-serine protease inhibitors of hepatitis c virus

Publications (1)

Publication Number Publication Date
NO20042792L true NO20042792L (no) 2004-10-15

Family

ID=27609106

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20042792A NO20042792L (no) 2002-01-18 2004-07-02 Nye peptider som NS3-serinproteaseinhibitorer for hepatitt C-virus

Country Status (28)

Country Link
US (2) US7244721B2 (https=)
EP (1) EP1481000B1 (https=)
JP (1) JP4563033B2 (https=)
KR (1) KR101020355B1 (https=)
CN (2) CN1633446A (https=)
AR (1) AR038183A1 (https=)
AT (1) ATE469914T1 (https=)
AU (1) AU2009210423B2 (https=)
BR (1) BR0306931A (https=)
CA (1) CA2473032A1 (https=)
CO (1) CO5650168A2 (https=)
CY (1) CY1111225T1 (https=)
DE (1) DE60332814D1 (https=)
DK (1) DK1481000T3 (https=)
EC (1) ECSP045191A (https=)
IL (1) IL162815A0 (https=)
MX (1) MXPA04006934A (https=)
MY (1) MY140710A (https=)
NO (1) NO20042792L (https=)
NZ (1) NZ571073A (https=)
PE (1) PE20030852A1 (https=)
PL (1) PL372747A1 (https=)
PT (1) PT1481000E (https=)
RU (1) RU2404189C9 (https=)
SI (1) SI1481000T1 (https=)
TW (1) TWI334872B (https=)
WO (1) WO2003062265A2 (https=)
ZA (1) ZA200405304B (https=)

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* Cited by examiner, † Cited by third party
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