NO20025977L - Imidazopyridin - og imidazopyrimidin antivirale forbindelser - Google Patents

Imidazopyridin - og imidazopyrimidin antivirale forbindelser

Info

Publication number
NO20025977L
NO20025977L NO20025977A NO20025977A NO20025977L NO 20025977 L NO20025977 L NO 20025977L NO 20025977 A NO20025977 A NO 20025977A NO 20025977 A NO20025977 A NO 20025977A NO 20025977 L NO20025977 L NO 20025977L
Authority
NO
Norway
Prior art keywords
imidazopyridine
antiviral compounds
imidazopyrimidine
imidazopyrimidine antiviral
compounds
Prior art date
Application number
NO20025977A
Other languages
English (en)
Norwegian (no)
Other versions
NO20025977D0 (no
Inventor
Kuo-Long Yu
Rita L Civiello
Keith Dean Combrink
Hatice Bel Guelgeze
Ny Sin
Xiangdong Wang
Nicholas A Meanwell
Brian Lee Venables
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of NO20025977D0 publication Critical patent/NO20025977D0/no
Publication of NO20025977L publication Critical patent/NO20025977L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
NO20025977A 2000-06-13 2002-12-12 Imidazopyridin - og imidazopyrimidin antivirale forbindelser NO20025977L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US21144700P 2000-06-13 2000-06-13
US26336301P 2001-01-22 2001-01-22
PCT/US2001/014775 WO2001095910A1 (en) 2000-06-13 2001-05-08 Imidazopyridine and imidazopyrimidine antiviral agents

Publications (2)

Publication Number Publication Date
NO20025977D0 NO20025977D0 (no) 2002-12-12
NO20025977L true NO20025977L (no) 2003-01-29

Family

ID=26906145

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20025977A NO20025977L (no) 2000-06-13 2002-12-12 Imidazopyridin - og imidazopyrimidin antivirale forbindelser

Country Status (20)

Country Link
US (1) US6489338B2 (cg-RX-API-DMAC7.html)
EP (1) EP1311268A4 (cg-RX-API-DMAC7.html)
JP (1) JP2004503501A (cg-RX-API-DMAC7.html)
KR (1) KR20030008151A (cg-RX-API-DMAC7.html)
CN (1) CN1436079A (cg-RX-API-DMAC7.html)
AR (1) AR029128A1 (cg-RX-API-DMAC7.html)
AU (2) AU2001272906B2 (cg-RX-API-DMAC7.html)
BR (1) BR0111569A (cg-RX-API-DMAC7.html)
CA (1) CA2412327A1 (cg-RX-API-DMAC7.html)
CZ (1) CZ20024078A3 (cg-RX-API-DMAC7.html)
HU (1) HUP0400766A2 (cg-RX-API-DMAC7.html)
IL (1) IL152889A0 (cg-RX-API-DMAC7.html)
MX (1) MXPA02012204A (cg-RX-API-DMAC7.html)
NO (1) NO20025977L (cg-RX-API-DMAC7.html)
NZ (1) NZ523566A (cg-RX-API-DMAC7.html)
PE (1) PE20011348A1 (cg-RX-API-DMAC7.html)
PL (1) PL360290A1 (cg-RX-API-DMAC7.html)
RU (1) RU2003100828A (cg-RX-API-DMAC7.html)
UY (1) UY26758A1 (cg-RX-API-DMAC7.html)
WO (1) WO2001095910A1 (cg-RX-API-DMAC7.html)

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US6919331B2 (en) * 2001-12-10 2005-07-19 Bristol-Myers Squibb Company Substituted 2-methyl-benzimidazole respiratory syncytial virus antiviral agents
WO2004043913A2 (en) * 2002-11-08 2004-05-27 Trimeris, Inc. Hetero-substituted benzimidazole compounds and antiviral uses thereof
JP2007501252A (ja) * 2003-08-05 2007-01-25 スリーエム イノベイティブ プロパティズ カンパニー 免疫応答調整剤を含有する製剤
EP1682547B1 (en) 2003-10-30 2012-10-24 Boehringer Ingelheim (Canada) Ltd. Rsv polymerase inhibitors
CN100582109C (zh) 2003-12-24 2010-01-20 生物区科学管理控股有限公司 用于治疗呼吸道合胞体病毒感染的多环试剂
GB0406282D0 (en) * 2004-03-19 2004-04-21 Arrow Therapeutics Ltd Therapeutic compounds
GB0406279D0 (en) * 2004-03-19 2004-04-21 Arrow Therapeutics Ltd Therapeutic compounds
CA2574220C (en) 2004-07-27 2014-09-16 Gilead Sciences, Inc. Imidazo[4,5-d]pyrimidines, their uses and methods of preparation
CA2612263C (en) 2005-06-20 2015-04-14 Tibotec Pharmaceuticals Ltd. 1-(2-amino-3-(substituted alkyl)-3h-benzimidazolylmethyl)-3-subtituted-1,3-dihydro-benzoimidazol-2-ones with activity on respiratory syncytial virus
BRPI0611744B8 (pt) 2005-06-20 2021-05-25 Janssen R & D Ireland benzimidazóis heterociclilaminoalquila substituída, seu processo de preparação e composição farmacêutica
JP5070207B2 (ja) 2005-06-20 2012-11-07 テイボテク・フアーマシユーチカルズ 2−置換ベンズイミダゾール
TWI423972B (zh) 2006-09-28 2014-01-21 Biota Scient Management 治療呼吸系融合細胞病毒感染之多環劑
WO2009084544A1 (ja) * 2007-12-27 2009-07-09 Idemitsu Kosan Co., Ltd. 含窒素複素環誘導体及びそれを用いた有機エレクトロルミネッセンス素子
WO2010103306A1 (en) 2009-03-10 2010-09-16 Astrazeneca Uk Limited Benzimidazole derivatives and their use as antivaral agents
RU2407738C1 (ru) * 2009-07-03 2010-12-27 Общество с ограниченной ответственностью "Интеллектуальный Диалог" Противовирусный активный компонент, фармацевтическая композиция, лекарственное средство, способ лечения вирусных заболеваний
TWI508968B (zh) 2010-02-08 2015-11-21 Biota Scient Management 用於治療呼吸道融合性病毒感染的化合物
WO2011115150A1 (ja) * 2010-03-18 2011-09-22 興和株式会社 ベンゾチアジン化合物の製造方法
US8796303B2 (en) 2010-11-26 2014-08-05 Biota Scientific Management Pty Ltd. Imidazo[2,1-G][1,7]naphthyridines for treating respiratory syncytial virus infections
TWI541241B (zh) * 2010-12-16 2016-07-11 健生科學愛爾蘭無限公司 作為呼吸道融合病毒抗病毒劑之咪唑并吡啶類
TWI515187B (zh) 2010-12-16 2016-01-01 健生科學愛爾蘭無限公司 作為呼吸道融合病毒抗病毒劑之吲哚類
TWI530495B (zh) 2010-12-16 2016-04-21 健生科學愛爾蘭無限公司 苯并咪唑呼吸道融合病毒抑制劑
TWI527814B (zh) 2010-12-16 2016-04-01 健生科學愛爾蘭無限公司 作為呼吸道融合病毒抗病毒劑之氮雜苯并咪唑類
TWI501967B (zh) * 2010-12-16 2015-10-01 Janssen R&D Ireland 作為呼吸道融合病毒抗病毒劑之氮雜吲哚類
CN103860538B (zh) * 2011-03-23 2016-03-02 上海市第一人民医院 靶向人La蛋白的先导化合物及其在制备抗乙型肝炎病毒的药物中的用途
EA028626B1 (ru) * 2012-06-11 2017-12-29 Юсб Байофарма Спрл БЕНЗИМИДАЗОЛЫ, МОДУЛИРУЮЩИЕ TNF-α
CN104470916A (zh) * 2012-06-15 2015-03-25 爱尔兰詹森研发公司 新颖的作为呼吸道合胞病毒抗病毒剂的被苯并咪唑取代的1,3-二氢-2h-苯并咪唑-2-酮衍生物
AU2013276519B2 (en) * 2012-06-15 2017-05-25 Janssen Sciences Ireland Uc 1,3-dihydro-2H-benzimidazol-2-one derivatives substituted with heterocycles as respiratory syncytial virus antiviral agents
KR20150032283A (ko) * 2012-06-15 2015-03-25 얀센 알 앤드 디 아일랜드 호흡기 합포체 바이러스의 항바이러스제로서의 헤테로사이클로 치환된 1,3-디하이드로-2h-벤즈이미다졸-2-온 유도체
JP2015519385A (ja) * 2012-06-15 2015-07-09 ヤンセン・アールアンドデイ・アイルランド Rsウイルス抗ウイルス薬としての、ベンゾイミダゾールによって置換された新規4−置換1,3−ジヒドロ−2h−ベンゾイミダゾル−2−オン誘導体
DK2909195T3 (en) * 2012-10-16 2017-09-25 Janssen Sciences Ireland Uc ANTIVIRAL RELATIONS TO RSV
JP2016145155A (ja) * 2013-04-30 2016-08-12 日本農薬株式会社 フタルアミド誘導体及び該誘導体を含有する農園芸用殺虫剤並びにその使用方法
KR20160075766A (ko) * 2013-10-29 2016-06-29 메디비르 아베 퀴나졸린계 호흡기 세포융합 바이러스 억제제
WO2015065336A1 (en) * 2013-10-29 2015-05-07 Medivir Ab Respiratory syncytial virus inhibitors
WO2017066014A1 (en) * 2015-10-14 2017-04-20 Sunnylife Pharma Inc. Bruton's tyrosine kinase inhibitors
WO2019046364A1 (en) * 2017-08-29 2019-03-07 Emory University INHIBITORS OF SYNCYTIAL RESPIRATORY VIRUS (RSV) REPLICATION AND USES THEREOF
PH12022551042A1 (en) * 2019-10-30 2023-05-29 Janssen Sciences Ireland Unlimited Co Synthesis of 3-({5-chloro-1-[3-(methylsulfonyl)propyl]-1h-indol-2 yl} methyl)-1-(2,2,2-trifluoroethyl)-1,3-dihydro-2h-imidazo[4,5-c]pyridin-2-one
KR20220097385A (ko) * 2019-10-30 2022-07-07 얀센 사이언시즈 아일랜드 언리미티드 컴퍼니 3-니트로-n-(2,2,2-트리플루오로에틸)-4-피리딘아민의 합성
WO2021250180A1 (en) 2020-06-11 2021-12-16 Janssen Sciences Ireland Unlimited Company Hemi (l)-tartrate forms of 3-({5-chloro-1-[3-(methylsulfonyl)propyl]-1h-indol-2 yl} methyl)-1-(2,2,2-trifluoroethyl)-1,3-dihydro-2h-imidazo[4,5-c]pyridin-2-one and pharmaceutical compositions comprising the same
WO2022184606A1 (en) * 2021-03-01 2022-09-09 Janssen Sciences Ireland Unlimited Company Synthesis of rilematovir
MX2024009216A (es) * 2022-01-28 2024-08-06 Insilico Medicine Ip Ltd Inhibidores de ectonucleotido pirofosfatasa-fosfodiesterasa 1 (enpp1) y usos de los mismos.
WO2025026383A1 (en) * 2023-08-02 2025-02-06 Insilico Medicine Ip Limited Crytsalline forms of ectonucleotide pyrophosphatase-phosphodiesterase 1 (enpp1) inhibitors and uses thereof

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Also Published As

Publication number Publication date
AU2001272906B2 (en) 2004-08-26
US6489338B2 (en) 2002-12-03
NO20025977D0 (no) 2002-12-12
KR20030008151A (ko) 2003-01-24
EP1311268A4 (en) 2004-06-30
WO2001095910A1 (en) 2001-12-20
UY26758A1 (es) 2002-01-31
NZ523566A (en) 2004-08-27
PL360290A1 (en) 2004-09-06
BR0111569A (pt) 2003-04-29
IL152889A0 (en) 2003-06-24
MXPA02012204A (es) 2003-10-15
US20020016309A1 (en) 2002-02-07
CN1436079A (zh) 2003-08-13
HUP0400766A2 (hu) 2004-07-28
AR029128A1 (es) 2003-06-04
RU2003100828A (ru) 2004-06-27
CZ20024078A3 (cs) 2003-08-13
AU7290601A (en) 2001-12-24
EP1311268A1 (en) 2003-05-21
PE20011348A1 (es) 2002-02-07
JP2004503501A (ja) 2004-02-05
CA2412327A1 (en) 2001-12-20

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Legal Events

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FC2A Withdrawal, rejection or dismissal of laid open patent application