NO174256C - Analogifremgangsmåte ved fremstilling av terapeutisk aktive kinuklidinderivater - Google Patents

Analogifremgangsmåte ved fremstilling av terapeutisk aktive kinuklidinderivater

Info

Publication number
NO174256C
NO174256C NO904523A NO904523A NO174256C NO 174256 C NO174256 C NO 174256C NO 904523 A NO904523 A NO 904523A NO 904523 A NO904523 A NO 904523A NO 174256 C NO174256 C NO 174256C
Authority
NO
Norway
Prior art keywords
therapeutically active
analogous method
quinuclidine derivatives
preparing therapeutically
halo
Prior art date
Application number
NO904523A
Other languages
English (en)
Norwegian (no)
Other versions
NO174256B (no
NO904523L (no
NO904523D0 (no
Inventor
Peter Edward Cross
Alan Stobie
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of NO904523D0 publication Critical patent/NO904523D0/no
Publication of NO904523L publication Critical patent/NO904523L/no
Publication of NO174256B publication Critical patent/NO174256B/no
Publication of NO174256C publication Critical patent/NO174256C/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/06—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing isoquinuclidine ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D453/00—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02—Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pulmonology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Glass Compositions (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Feeding And Guiding Record Carriers (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NO904523A 1989-10-19 1990-10-18 Analogifremgangsmåte ved fremstilling av terapeutisk aktive kinuklidinderivater NO174256C (no)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB898923590A GB8923590D0 (en) 1989-10-19 1989-10-19 Antimuscarinic bronchodilators

Publications (4)

Publication Number Publication Date
NO904523D0 NO904523D0 (no) 1990-10-18
NO904523L NO904523L (no) 1991-04-22
NO174256B NO174256B (no) 1993-12-27
NO174256C true NO174256C (no) 1994-04-06

Family

ID=10664848

Family Applications (1)

Application Number Title Priority Date Filing Date
NO904523A NO174256C (no) 1989-10-19 1990-10-18 Analogifremgangsmåte ved fremstilling av terapeutisk aktive kinuklidinderivater

Country Status (19)

Country Link
US (1) US5171744A (de)
EP (1) EP0424021B1 (de)
JP (1) JPH06780B2 (de)
KR (1) KR930004845B1 (de)
CN (1) CN1022488C (de)
AT (1) ATE102198T1 (de)
AU (1) AU616362B2 (de)
CA (1) CA2027896A1 (de)
DE (1) DE69007009T2 (de)
FI (1) FI905147A7 (de)
GB (1) GB8923590D0 (de)
HU (1) HU206345B (de)
NO (1) NO174256C (de)
NZ (1) NZ235750A (de)
PL (1) PL287365A1 (de)
PT (1) PT95610A (de)
RU (1) RU2005721C1 (de)
YU (1) YU197290A (de)
ZA (1) ZA908343B (de)

Families Citing this family (78)

* Cited by examiner, † Cited by third party
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CA2073005C (en) * 1990-09-06 1998-11-10 Alan Stobie Antimuscarinic bronchodilators
GB9119705D0 (en) * 1991-09-14 1991-10-30 Pfizer Ltd Therapeutic compounds
US5340826A (en) * 1993-02-04 1994-08-23 Pfizer Inc. Pharmaceutical agents for treatment of urinary incontinence
FR2754261B1 (fr) * 1996-10-08 1998-10-30 Synthelabo Derives de quinuclidine, leur preparation et leur application en therapeutique
US5981549A (en) * 1997-02-14 1999-11-09 Synapse Pharmaceutical International Method for controlling or alleviating the symptoms of respiratory disease and allergies
JP2002526482A (ja) * 1998-09-18 2002-08-20 バーテックス ファーマシューティカルズ インコーポレイテッド ｐ３８のインヒビター
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EA017919B1 (ru) 2007-12-10 2013-04-30 Новартис Аг Производные пиразин-2-карбоксамида для лечения заболеваний, которые поддаются лечению путем блокирования эпителиальных натриевых каналов
EP2231642B1 (de) 2008-01-11 2013-10-23 Novartis AG Pyrimidine als kinasehemmer
EP2100598A1 (de) 2008-03-13 2009-09-16 Laboratorios Almirall, S.A. Inhalationszusammensetzung enthaltend Aclidinium zur Behandlung von Asthma sowie chronisch-obstruktiver Lungenerkrankung
EP2100599A1 (de) 2008-03-13 2009-09-16 Laboratorios Almirall, S.A. Inhalationszusammensetzung enthaltend Aclidinium zur Behandlung von Asthma sowie chronisch-obstruktiver Lungenerkrankung
US8268834B2 (en) 2008-03-19 2012-09-18 Novartis Ag Pyrazine derivatives that inhibit phosphatidylinositol 3-kinase enzyme
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US8389526B2 (en) 2009-08-07 2013-03-05 Novartis Ag 3-heteroarylmethyl-imidazo[1,2-b]pyridazin-6-yl derivatives
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EP2813227A1 (de) 2009-10-22 2014-12-17 Vertex Pharmaceuticals Incorporated Zusammensetzungen für die Behandlung von Mukoviszidose und anderen chronischen Erkrankungen
US8247436B2 (en) 2010-03-19 2012-08-21 Novartis Ag Pyridine and pyrazine derivative for the treatment of CF
ES2545812T3 (es) * 2010-06-22 2015-09-16 Chiesi Farmaceutici S.P.A. Derivados aminoéster de alcaloides y composición medicinal de estos
WO2012034095A1 (en) 2010-09-09 2012-03-15 Irm Llc Compounds and compositions as trk inhibitors
US8637516B2 (en) 2010-09-09 2014-01-28 Irm Llc Compounds and compositions as TRK inhibitors
US8372845B2 (en) 2010-09-17 2013-02-12 Novartis Ag Pyrazine derivatives as enac blockers
JP2014505088A (ja) 2011-02-10 2014-02-27 ノバルティス アーゲー Ｃ−ＭＥＴチロシンキナーゼ阻害剤としての［１，２，４］トリアゾロ［４，３−ｂ］ピリダジン化合物
EP2678016B1 (de) 2011-02-23 2016-08-10 Intellikine, LLC Heterocyclische verbindungen und ihre verwendung
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US8883819B2 (en) 2011-09-01 2014-11-11 Irm Llc Bicyclic heterocycle derivatives for the treatment of pulmonary arterial hypertension
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WO2013038381A1 (en) 2011-09-16 2013-03-21 Novartis Ag Pyridine/pyrazine amide derivatives
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CN110507654A (zh) 2012-04-03 2019-11-29 诺华有限公司 有酪氨酸激酶抑制剂的组合产品和其应用
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US10112926B2 (en) 2014-04-24 2018-10-30 Novartis Ag Amino pyridine derivatives as phosphatidylinositol 3-kinase inhibitors
PL3134395T3 (pl) 2014-04-24 2018-07-31 Novartis Ag Pochodne pirazyny jako inhibitory 3-kinazy fosfatydyloinozytolu
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US4644003A (en) * 1985-04-03 1987-02-17 Research Corporation 3-quinuclidinol esters, useful as antagonists of muscarinic acetylcholine receptors
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IT1228288B (it) * 1989-01-09 1991-06-07 Zambon Spa Composti ad attivita' antiserotoninica

Also Published As

Publication number Publication date
YU197290A (sh) 1993-10-20
AU6472690A (en) 1991-07-25
AU616362B2 (en) 1991-10-24
KR910007924A (ko) 1991-05-30
CA2027896A1 (en) 1991-04-20
DE69007009D1 (de) 1994-04-07
FI905147A7 (fi) 1991-04-20
DE69007009T2 (de) 1994-06-09
EP0424021B1 (de) 1994-03-02
ATE102198T1 (de) 1994-03-15
CN1022488C (zh) 1993-10-20
RU2005721C1 (ru) 1994-01-15
NZ235750A (en) 1992-03-26
CN1051041A (zh) 1991-05-01
ZA908343B (en) 1992-06-24
NO174256B (no) 1993-12-27
PL287365A1 (en) 1991-06-03
GB8923590D0 (en) 1989-12-06
JPH06780B2 (ja) 1994-01-05
HU906495D0 (en) 1991-04-29
HUT56365A (en) 1991-08-28
HU206345B (en) 1992-10-28
US5171744A (en) 1992-12-15
KR930004845B1 (ko) 1993-06-09
NO904523L (no) 1991-04-22
FI905147A0 (fi) 1990-10-18
PT95610A (pt) 1991-09-13
EP0424021A1 (de) 1991-04-24
NO904523D0 (no) 1990-10-18
JPH03133980A (ja) 1991-06-07

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