NO140931C - Analogifremgangsmaate til fremstilling av terapeutisk virksomme estere av alfa-aminobenzylpenicilliner - Google Patents

Analogifremgangsmaate til fremstilling av terapeutisk virksomme estere av alfa-aminobenzylpenicilliner

Info

Publication number
NO140931C
NO140931C NO3449/71A NO344971A NO140931C NO 140931 C NO140931 C NO 140931C NO 3449/71 A NO3449/71 A NO 3449/71A NO 344971 A NO344971 A NO 344971A NO 140931 C NO140931 C NO 140931C
Authority
NO
Norway
Prior art keywords
aminobenzylpenicillines
alfa
preparation
therapeutically effective
effective esters
Prior art date
Application number
NO3449/71A
Other languages
English (en)
Norwegian (no)
Other versions
NO140931B (no
Inventor
Bertil Aake Ekstroem
Berndt Olof Harald Sjoeberg
Original Assignee
Astra Laekemedel Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from SE7012688A external-priority patent/SE374747B/xx
Priority claimed from SE7015720A external-priority patent/SE380806B/xx
Application filed by Astra Laekemedel Ab filed Critical Astra Laekemedel Ab
Priority to NO74744606A priority Critical patent/NO142670C/no
Publication of NO140931B publication Critical patent/NO140931B/no
Publication of NO140931C publication Critical patent/NO140931C/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
NO3449/71A 1970-09-17 1971-09-16 Analogifremgangsmaate til fremstilling av terapeutisk virksomme estere av alfa-aminobenzylpenicilliner NO140931C (no)

Priority Applications (1)

Application Number Priority Date Filing Date Title
NO74744606A NO142670C (no) 1970-09-17 1974-12-19 Benzylpenicillinester for anvendelse som utgangsmateriale ved fremstilling av en terapeutisk virksom ester av alfa-aminobenzylpenicilliner

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
SE7012688A SE374747B (cs) 1970-09-17 1970-09-17
SE7015720A SE380806B (sv) 1970-11-20 1970-11-20 Forfarande for framstellning av nya estrar av alfa-aminopenicilliner

Publications (2)

Publication Number Publication Date
NO140931B NO140931B (no) 1979-09-03
NO140931C true NO140931C (no) 1979-12-12

Family

ID=26655897

Family Applications (4)

Application Number Title Priority Date Filing Date
NO3449/71A NO140931C (no) 1970-09-17 1971-09-16 Analogifremgangsmaate til fremstilling av terapeutisk virksomme estere av alfa-aminobenzylpenicilliner
NO236/72A NO140930C (no) 1970-09-17 1972-01-31 6-aminopenicillansyrestere for anvendelse som utgangsmateriale ved fremstilling av terapeutisk virksomme estere av alfa-aminobenzylpenicilliner
NO74744606A NO142670C (no) 1970-09-17 1974-12-19 Benzylpenicillinester for anvendelse som utgangsmateriale ved fremstilling av en terapeutisk virksom ester av alfa-aminobenzylpenicilliner
NO784144A NO142671C (no) 1970-09-17 1978-12-08 Alfa-azidobenzylpenicillinestere for bruk ved fremstilling av terapeutisk virksomme alfa-aminobenzylpenicillinestere

Family Applications After (3)

Application Number Title Priority Date Filing Date
NO236/72A NO140930C (no) 1970-09-17 1972-01-31 6-aminopenicillansyrestere for anvendelse som utgangsmateriale ved fremstilling av terapeutisk virksomme estere av alfa-aminobenzylpenicilliner
NO74744606A NO142670C (no) 1970-09-17 1974-12-19 Benzylpenicillinester for anvendelse som utgangsmateriale ved fremstilling av en terapeutisk virksom ester av alfa-aminobenzylpenicilliner
NO784144A NO142671C (no) 1970-09-17 1978-12-08 Alfa-azidobenzylpenicillinestere for bruk ved fremstilling av terapeutisk virksomme alfa-aminobenzylpenicillinestere

Country Status (21)

Country Link
US (2) US3873521A (cs)
JP (2) JPS5317597B1 (cs)
AR (2) AR201730A1 (cs)
AT (2) AT309681B (cs)
BE (1) BE772723A (cs)
BR (1) BR7106116D0 (cs)
CA (2) CA960211A (cs)
CH (5) CH577513A5 (cs)
CS (2) CS187312B2 (cs)
DD (1) DD94815A5 (cs)
DK (6) DK132759C (cs)
ES (3) ES395145A1 (cs)
FI (4) FI55203C (cs)
FR (1) FR2106578B1 (cs)
GB (1) GB1363506A (cs)
HU (1) HU165868B (cs)
IE (1) IE35642B1 (cs)
IT (1) IT1049876B (cs)
NL (3) NL164860C (cs)
NO (4) NO140931C (cs)
SU (2) SU553936A3 (cs)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1426869A (en) * 1972-03-13 1976-03-03 Astra Laekemedel Ab Penicillins
US4089963A (en) * 1972-03-13 1978-05-16 Astra Pharmaceutical Products, Inc. Esters of amidinopenicillanic acids, pharmaceutical preparations and method for treating infectious diseases
GB1425933A (en) * 1972-03-13 1976-02-25 Astra Laekemedel Ab Cephalosporins
GB1437088A (en) * 1972-05-25 1976-05-26 Beecham Group Ltd Esters of penicillins and cephalosporins
NL7401782A (cs) * 1973-02-14 1974-08-16
GB1550359A (en) * 1975-08-07 1979-08-15 Beecham Group Ltd Antibiotic compositions for oral administration
US4247461A (en) * 1979-11-16 1981-01-27 Bristol-Myers Company Esterification process using methoxymethyl-P-toluenesulfonate
US4340539A (en) * 1980-01-21 1982-07-20 Bristol-Myers Company Derivatives of 6-bromo penicillanic acid
CA1212105A (en) 1980-04-30 1986-09-30 Shoji Ikeda Ampicillin esters and production thereof
FR2482587A1 (fr) * 1980-05-14 1981-11-20 Poudres & Explosifs Ste Nale Procede de synthese de chloroformiates a-chlores et nouveaux chloroformiates a-chlores
US4321253A (en) * 1980-08-22 1982-03-23 Beatty Morgan L Suspension of microencapsulated bacampicillin acid addition salt for oral, especially pediatric, administration
US4479947A (en) * 1981-07-13 1984-10-30 Merck & Co., Inc. Oral absorption enhancement of carboxylic acid pharmaceuticals using (5-alkyl-2-oxo-1,3-dioxolen-4-yl)methyl ester group
CA1202617A (en) * 1982-03-19 1986-04-01 Norman B. Jones Bacampicillin napsylate
FR2532933B1 (fr) * 1982-06-29 1987-11-13 Astra Laekemedel Ab Perfectionnements apportes a la preparation d'antibiotiques
SE454879B (sv) * 1982-06-29 1988-06-06 Astra Laekemedel Ab Alfa-bromodietylkarbonat samt dess anvendning som mellanprodukt vid framstellning av penicillin g
GB2123821B (en) * 1982-06-29 1987-04-23 Astra Laekemedel Ab At-halogeno diethyl carbonates and their use in the preparation of antibiotics
IT1190897B (it) * 1982-06-29 1988-02-24 Opos Biochimica Srl Procedimento per la preparazione dell'estere 1-etossicarbonilossietilico dell'acido 6-(d(-)-alfa aminoalfa fenilacetamido)-penicillanico
JPS5927900A (ja) * 1982-08-09 1984-02-14 Wakunaga Seiyaku Kk 固定化オリゴヌクレオチド
US4606865A (en) * 1982-09-20 1986-08-19 Astra Lakemedel Aktiebolag Methods for the preparation of α-bromodiethylcarbonate
DK149079C (da) * 1982-10-06 1986-06-23 Novo Industri As Fremgangsmaade til fremstilling af et immobiliseret enzympraeparat
IL67177A (en) * 1982-11-04 1985-08-30 Orvet Bv 1-bromoethyl ethyl carbonate,methods for its preparation and 1-bromoethylchloroformate and 1-bromoethylbromoformate obtained as intermediates
IL67637A0 (en) * 1983-01-07 1983-05-15 Orvet Bv Preparation of 1'-ethoxycarbonyl-oxyethyl esters of penicillins and novel intermediates
IL67445A (en) * 1982-12-09 1985-11-29 Teva Pharma Ethoxycarbonyloxy ethyl esters of non-steroidal anti-inflammatory carboxylic acids
FR2551058B1 (fr) * 1983-08-26 1986-09-26 Poudres & Explosifs Ste Nale Procede de preparation de chloroformiates a-chlores
SE8405611D0 (sv) * 1984-11-09 1984-11-09 Astra Laekemedel Ab Process for stabilization of bacampicillin hydrochloride
US4855455A (en) * 1988-01-22 1989-08-08 W. R. Grace & Co.-Conn. Preparation of amino acid derivatives

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1021654A (fr) * 1949-07-07 1953-02-23 Lphivens Kemiske Fabrik Ved A Procédé de production d'éthers-sels aminés de pénicilline et de composés qui s'y rattachent
GB1241844A (en) * 1968-08-23 1971-08-04 Beecham Group Ltd Penicillins
US3697507A (en) * 1968-09-26 1972-10-10 Leo Pharm Prod Ltd Esters of {60 -aminobenzylpenicillin
US3660575A (en) * 1968-09-26 1972-05-02 Leo Pharm Prod Ltd Esters of alpha-aminobenzylpenicillin in dosage unit form

Also Published As

Publication number Publication date
NL171160B (nl) 1982-09-16
ES395145A1 (es) 1974-11-16
FI55203B (fi) 1979-02-28
DK509674A (cs) 1975-06-02
BE772723A (fr) 1972-03-17
NO744606L (cs) 1972-03-20
NO140930B (no) 1979-09-03
SU553936A3 (ru) 1977-04-05
GB1363506A (en) 1974-08-14
NL171160C (nl) 1983-02-16
CH602745A5 (cs) 1978-07-31
FI773032A (cs) 1977-10-13
DD94815A5 (cs) 1973-01-05
JPS5537996B2 (cs) 1980-10-01
NO142670C (no) 1980-09-24
CH613207A5 (cs) 1979-09-14
FI59103C (fi) 1981-06-10
DK132759C (da) 1976-07-05
NO784144L (no) 1972-03-20
DK163482A (da) 1982-04-07
NO140931B (no) 1979-09-03
FR2106578A1 (cs) 1972-05-05
DK509774A (cs) 1975-05-26
DK150200B (da) 1987-01-05
CS187316B2 (cs) 1979-01-31
DE2144457B2 (de) 1977-05-05
US3873521A (en) 1975-03-25
HU165868B (cs) 1974-12-28
CA960211A (en) 1974-12-31
DK150201C (da) 1987-07-06
NL7801086A (nl) 1978-05-31
FI55203C (fi) 1979-06-11
IT1049876B (it) 1981-02-10
IE35642L (en) 1972-03-17
AR210991A1 (es) 1977-10-14
CH589654A5 (cs) 1977-07-15
DK158519C (da) 1990-11-05
NO140930C (no) 1979-12-12
DE2144457A1 (cs) 1972-03-30
FI57951B (fi) 1980-07-31
FI59600C (fi) 1981-09-10
NO142670B (no) 1980-06-16
NL164860C (nl) 1981-02-16
FI59103B (fi) 1981-02-27
DK158519B (da) 1990-05-28
NL7112789A (cs) 1972-03-21
FI791386A (fi) 1979-04-27
DK375975A (cs) 1975-08-20
JPS5317597B1 (cs) 1978-06-09
CH583239A5 (cs) 1976-12-31
SU1153830A3 (ru) 1985-04-30
FI59600B (fi) 1981-05-29
US3939270A (en) 1976-02-17
ES401745A1 (es) 1976-05-16
AT309681B (de) 1973-08-27
IE35642B1 (en) 1976-04-14
NL8001563A (nl) 1980-06-30
DK133380A (da) 1980-03-27
NO142671C (no) 1980-09-24
ES433637A1 (es) 1976-11-16
CA1008447A (en) 1977-04-12
NO142671B (no) 1980-06-16
FI381474A (cs) 1974-12-31
CH577513A5 (cs) 1976-07-15
DK150201B (da) 1987-01-05
BR7106116D0 (pt) 1973-03-20
CS187312B2 (en) 1979-01-31
AT311557B (de) 1973-11-26
JPS5136491A (cs) 1976-03-27
FI57951C (fi) 1980-11-10
DK132759B (da) 1976-02-02
FR2106578B1 (cs) 1975-06-06
DK150200C (da) 1987-07-06
AR201730A1 (es) 1975-04-15

Similar Documents

Publication Publication Date Title
NO140931C (no) Analogifremgangsmaate til fremstilling av terapeutisk virksomme estere av alfa-aminobenzylpenicilliner
SE393381B (sv) Analogiforfarande for framstellning av 8-azapurin - 6 - onderivat
NO139560C (no) Analogifremgangsmaate til fremstilling av terapeutisk virksomme nonapeptidamid-derivater
NO781312L (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive 3-merkaptotiadiazol- eller merkaptotetrazol-cefalosporiner
NO136837C (no) Analogifremgangsm}te for fremstilling av terapeutisk aktive pleuromutiliner
SE393602B (sv) Forfarande for framstellning av alfa aspartyl-aminosyraestrar
SE390304B (sv) Analogiforfarande for framstellning av 4-hydroxi-5-etyl-6-fonylpyrimidin
SE394678B (sv) Analogiforfarande for framstellning av pyridokinolinderivat
NO137824C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive fenylalkyltetrazoler
NO138999C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive difenylyl-alkanoylaminopyridiner
SE399701B (sv) Forfarande for framstellning av hydroxyalkyldiamin
SE402460B (sv) Analogiforfarande for framstellning av alkaloidestrar av eburnamintyp
NO137858C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive indanoner
SE394436B (sv) Forfarande for framstellning av 7-halogen-linkomyciner
NO137151C (no) Analogifremgangsm}te for fremstilling av terapeutisk aktive ortiotropin-peptider
SE395897B (sv) Forfarande for framstellning av 7beta-acylamido-3-metyl-cef-3-em-4-karbonsyror
SE385011B (sv) Forfarande for framstellning av alfa-linkosaminider
SE392611B (sv) Forfarande for framstellning av antrakinonkarboxylsyra
SE408418B (sv) Forfarande for framstellning av 5-fluor-pyrimidiner
SE395699B (sv) Forfarande for framstellning av kinuklidin-kinolinderivat
NO138375C (no) Analogifremgangsmaate til fremstilling av terapeutisk virksomme cefalosporinderivater
SE380795B (sv) Forfarande for framstellning av tiokarbamider
NO137695C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive n-tienylmetyl-heterocykliske forbindelser
NO139440C (no) Analogifremgangsmaate til fremstilling av terapeutisk aktive 2-amino-4h-pyraner
NO136841C (no) Analogifremgangsm}te for fremstilling av terapeutisk aktive fenylimidazolidinoner