MX9804816A - Suspensiones acuosas de esteres de acido graso de 9-hidroxirrisperidona. - Google Patents

Suspensiones acuosas de esteres de acido graso de 9-hidroxirrisperidona.

Info

Publication number
MX9804816A
MX9804816A MX9804816A MX9804816A MX9804816A MX 9804816 A MX9804816 A MX 9804816A MX 9804816 A MX9804816 A MX 9804816A MX 9804816 A MX9804816 A MX 9804816A MX 9804816 A MX9804816 A MX 9804816A
Authority
MX
Mexico
Prior art keywords
fatty acid
acid esters
pharmaceutically acceptable
active ingredient
aqueous suspensions
Prior art date
Application number
MX9804816A
Other languages
English (en)
Spanish (es)
Inventor
Marc Karel Jozef Francois
Roger Carolus August Embrechts
Herman Karel Borghijs
Johan Monbaliu
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8224016&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX9804816(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of MX9804816A publication Critical patent/MX9804816A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0019Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/517Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with carbocyclic ring systems, e.g. quinazoline, perimidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/02Inorganic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/26Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38Cellulose; Derivatives thereof

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Dermatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
MX9804816A 1996-05-20 1998-06-15 Suspensiones acuosas de esteres de acido graso de 9-hidroxirrisperidona. MX9804816A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP96201429 1996-05-20

Publications (1)

Publication Number Publication Date
MX9804816A true MX9804816A (es) 1998-10-31

Family

ID=8224016

Family Applications (1)

Application Number Title Priority Date Filing Date
MX9804816A MX9804816A (es) 1996-05-20 1998-06-15 Suspensiones acuosas de esteres de acido graso de 9-hidroxirrisperidona.

Country Status (37)

Country Link
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BR (1) BR9706824B8 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
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SI (1) SI0904081T1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
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TR (1) TR199800923T2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
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UA (1) UA61898C2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
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ZA (1) ZA974331B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

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Also Published As

Publication number Publication date
SK62098A3 (en) 2000-04-10
DK0904081T3 (da) 2002-02-25
NO981984D0 (no) 1998-04-30
FR11C0035I2 (fr) 2013-08-16
BG62684B1 (bg) 2000-05-31
HUP9901319A2 (hu) 1999-08-30
PL327995A1 (en) 1999-01-04
LU91842I2 (fr) 2011-09-20
PL188309B1 (pl) 2005-01-31
EE03594B1 (et) 2002-02-15
HRP970276A2 (en) 1998-04-30
EA199800531A1 (ru) 1998-12-24
AR007194A1 (es) 1999-10-13
HUP9901319A3 (en) 1999-11-29
PT904081E (pt) 2002-04-29
KR19990067603A (ko) 1999-08-25
AU715572B2 (en) 2000-02-03
KR100358373B1 (ko) 2003-02-11
WO1997044039A1 (en) 1997-11-27
ID16927A (id) 1997-11-20
MY126302A (en) 2006-09-29
TW487572B (en) 2002-05-21
DE69708284T2 (de) 2002-07-25
CA2236691A1 (en) 1997-11-27
ATE208619T1 (de) 2001-11-15
AU2955997A (en) 1997-12-09
EP0904081A1 (en) 1999-03-31
CN1206347A (zh) 1999-01-27
EE9800136A (et) 1998-10-15
DE69708284D1 (de) 2001-12-20
JP3274687B2 (ja) 2002-04-15
EA000536B1 (ru) 1999-10-28
US6077843A (en) 2000-06-20
NO2011015I2 (no) 2013-03-11
ES2167745T3 (es) 2002-05-16
EP0904081B1 (en) 2001-11-14
IL124551A0 (en) 1998-12-06
FR11C0035I1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 2011-07-10
DE122011100027I1 (de) 2011-11-17
SK284013B6 (sk) 2004-08-03
JP2000513718A (ja) 2000-10-17
NO981984L (no) 1998-11-19
HK1017852A1 (en) 1999-12-03
BR9706824B8 (pt) 2015-02-18
HUS1100013I1 (hu) 2017-03-28
IL124551A (en) 2001-08-26
HU224025B1 (hu) 2005-05-30
CY2011011I2 (el) 2016-12-14
CZ291284B6 (cs) 2003-01-15
SI0904081T1 (en) 2002-04-30
BR9706824A (pt) 1999-03-23
CY2270B1 (en) 2003-07-04
NZ330369A (en) 2000-04-28
UA61898C2 (en) 2003-12-15
NO315931B1 (no) 2003-11-17
NO2011015I1 (no) 2011-09-19
CN1093762C (zh) 2002-11-06
HRP970276B1 (en) 2002-04-30
CY2011011I1 (el) 2016-12-14
CA2236691C (en) 2007-01-02
CZ140198A3 (cs) 1999-04-14
BG102443A (en) 1999-06-30
TR199800923T2 (xx) 1999-09-21
ZA974331B (en) 1998-11-19

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