MX366793B - Metodos para preparar oxazolidinonas y composiciones que las contienen. - Google Patents

Metodos para preparar oxazolidinonas y composiciones que las contienen.

Info

Publication number
MX366793B
MX366793B MX2014004600A MX2014004600A MX366793B MX 366793 B MX366793 B MX 366793B MX 2014004600 A MX2014004600 A MX 2014004600A MX 2014004600 A MX2014004600 A MX 2014004600A MX 366793 B MX366793 B MX 366793B
Authority
MX
Mexico
Prior art keywords
methods
compositions containing
preparing
oxazolidinones
preparing oxazolidinones
Prior art date
Application number
MX2014004600A
Other languages
English (en)
Inventor
Carrie A Costello
Jaqueline A Simson
Robert J Duguid
Douglas Phillipson
Original Assignee
Merck Sharp & Dohme Corp Star
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Sharp & Dohme Corp Star filed Critical Merck Sharp & Dohme Corp Star
Publication of MX366793B publication Critical patent/MX366793B/es

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
    • C07F5/02—Boron compounds
    • C07F5/025—Boronic and borinic acid compounds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6558—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system
    • C07F9/65583—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Vascular Medicine (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Epidemiology (AREA)
  • Cardiology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

Abstract

Se describen métodos para preparar una clase de oxazolidinonas útiles para impedir el crecimiento bacteriano.
MX2014004600A 2008-10-10 2009-10-09 Metodos para preparar oxazolidinonas y composiciones que las contienen. MX366793B (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10446908P 2008-10-10 2008-10-10
PCT/US2009/060267 WO2010042887A2 (en) 2008-10-10 2009-10-09 Methods for preparing oxazolidinones and compositions containing them

Publications (1)

Publication Number Publication Date
MX366793B true MX366793B (es) 2019-07-24

Family

ID=41382395

Family Applications (2)

Application Number Title Priority Date Filing Date
MX2011003820A MX2011003820A (es) 2008-10-10 2009-10-09 Metodos para preparar oxazolidinonas y composiciones que las contienen.
MX2014004600A MX366793B (es) 2008-10-10 2009-10-09 Metodos para preparar oxazolidinonas y composiciones que las contienen.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
MX2011003820A MX2011003820A (es) 2008-10-10 2009-10-09 Metodos para preparar oxazolidinonas y composiciones que las contienen.

Country Status (13)

Country Link
US (2) US8604209B2 (es)
EP (2) EP2346858B1 (es)
JP (1) JP5773875B2 (es)
KR (1) KR101674146B1 (es)
CN (2) CN106220621B (es)
AU (1) AU2009303301B2 (es)
CA (1) CA2738671C (es)
ES (2) ES2744907T3 (es)
HK (2) HK1200169A1 (es)
MX (2) MX2011003820A (es)
RU (2) RU2659792C1 (es)
SG (2) SG195544A1 (es)
WO (1) WO2010042887A2 (es)

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CN106146485B (zh) * 2015-04-01 2021-04-30 上海迪赛诺化学制药有限公司 一种制备泰地唑胺的方法及其得到的泰地唑胺结晶体
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CN106279282B (zh) * 2015-05-21 2019-08-23 博瑞生物医药（苏州）股份有限公司 一种磷酸特地唑胺的纯化方法
CN106317114B (zh) * 2015-07-02 2018-11-20 南京优科制药有限公司 一种磷酸特地唑胺的制备方法
CN105131037B (zh) * 2015-07-28 2017-05-03 济南爱思医药科技有限公司 一种高纯度泰地唑胺磷酸酯的制备方法
CN106632298B (zh) * 2015-11-03 2021-06-01 上海科胜药物研发有限公司 一种泰地唑胺的制备方法及其中间体
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CN106632240A (zh) * 2016-11-25 2017-05-10 山东轩德医药科技有限公司 一种2‑甲基‑5‑(5‑溴吡啶‑2‑基)四氮唑的制备方法
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CN110938058B (zh) * 2018-09-22 2022-04-12 南京优科生物医药研究有限公司 一种噁唑烷酮类抗生素中间体的制备方法
CN111116652A (zh) * 2019-12-06 2020-05-08 山东中医药大学 一种高纯度磷酸特地唑胺的制备方法
CN113121518B (zh) * 2019-12-31 2022-06-28 北京福元医药股份有限公司 一种特地唑胺杂质的制备方法
CN111285848A (zh) * 2020-04-10 2020-06-16 苏州敬业医药化工有限公司 一种5-溴-2-(2-甲基-2h-四唑-5-基)吡啶的纯化方法
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CN112961186A (zh) * 2021-02-04 2021-06-15 海南通用康力制药有限公司 一种磷酸特地唑胺的纯化方法
CN113488445A (zh) * 2021-07-05 2021-10-08 合肥巨一动力系统有限公司 一种igbt封装散热结构及其应用的电机控制器
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KR101674146B1 (ko) 2016-11-08
CA2738671A1 (en) 2010-05-15
RU2011115109A (ru) 2012-11-20
CN106220621B (zh) 2019-06-11
AU2009303301A1 (en) 2010-04-15
WO2010042887A3 (en) 2010-06-24
US20100093669A1 (en) 2010-04-15
HK1232221A1 (zh) 2018-01-05
RU2659792C1 (ru) 2018-07-04
US9328087B2 (en) 2016-05-03
RU2556234C2 (ru) 2015-07-10
US8604209B2 (en) 2013-12-10
EP2346858A2 (en) 2011-07-27
SG195544A1 (en) 2013-12-30
CN102177156B (zh) 2016-08-24
AU2009303301B2 (en) 2014-09-11
ES2748505T3 (es) 2020-03-17
EP2346858B1 (en) 2019-08-07
US20140206878A1 (en) 2014-07-24
KR20110071107A (ko) 2011-06-28
HK1200169A1 (en) 2015-07-31
JP2012505252A (ja) 2012-03-01
EP2757104A1 (en) 2014-07-23
CN106220621A (zh) 2016-12-14
WO2010042887A2 (en) 2010-04-15
CA2738671C (en) 2018-05-01
CN102177156A (zh) 2011-09-07
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EP2757104B1 (en) 2019-08-14

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