MX351368B - Compuestos heteroarilo y metodos para utilizarlos. - Google Patents

Compuestos heteroarilo y metodos para utilizarlos.

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Publication number
MX351368B
MX351368B MX2012013624A MX2012013624A MX351368B MX 351368 B MX351368 B MX 351368B MX 2012013624 A MX2012013624 A MX 2012013624A MX 2012013624 A MX2012013624 A MX 2012013624A MX 351368 B MX351368 B MX 351368B
Authority
MX
Mexico
Prior art keywords
methods
compounds
disorders
heteroaryl compounds
heteroaryl
Prior art date
Application number
MX2012013624A
Other languages
English (en)
Other versions
MX2012013624A (es
Inventor
Xie Linghong
Charles Hewitt Michael
Emmerson Campbell John
Jones Philip
Original Assignee
Sunovion Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sunovion Pharmaceuticals Inc filed Critical Sunovion Pharmaceuticals Inc
Publication of MX2012013624A publication Critical patent/MX2012013624A/es
Publication of MX351368B publication Critical patent/MX351368B/es

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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/06—Peri-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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    • A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
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  • Diabetes (AREA)
  • Pain & Pain Management (AREA)
  • Psychiatry (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Psychology (AREA)
  • Hospice & Palliative Care (AREA)
  • Addiction (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Otolaryngology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

En la presente se proporcionan los compuestos heteroarilo, los métodos para sintetizarlos, las composiciones farmacéuticas que contienen estos compuestos y los métodos para su uso. En una modalidad, los compuestos que se proporcionan en la presente son útiles para el tratamiento, prevención y/o manejo de diversos trastornos, como pueden ser los trastornos de SNC y trastornos metabólicos, como pueden ser, más no se limitan a, trastornos neurológicos, sicosis, esquizofrenia, obesidad y diabetes.
MX2012013624A 2010-05-26 2011-05-26 Compuestos heteroarilo y metodos para utilizarlos. MX351368B (es)

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CN103038229B (zh) 2016-05-11
AU2011258217A1 (en) 2012-12-20
EP3318561A1 (en) 2018-05-09
IL266168A (en) 2019-06-30
JP2013526615A (ja) 2013-06-24
CA2800618A1 (en) 2011-12-01
IL223240A0 (en) 2013-02-03
JP2016028092A (ja) 2016-02-25
CA2800618C (en) 2018-08-28
IL223240B (en) 2019-05-30
US10562916B2 (en) 2020-02-18
EP2576540A2 (en) 2013-04-10
JP5911476B2 (ja) 2016-04-27
EP2576540B1 (en) 2019-09-04
WO2011150156A2 (en) 2011-12-01
US20130158003A1 (en) 2013-06-20
US8969349B2 (en) 2015-03-03
WO2011150156A3 (en) 2012-04-19
US20150166571A1 (en) 2015-06-18
US9834564B2 (en) 2017-12-05
MX2012013624A (es) 2013-02-11
NZ603789A (en) 2015-03-27
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AU2011258217B2 (en) 2016-12-15
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