MA34917B1 - Dérivés substitués de l'acide 3-hétéroaroylamino-propionique et leur utilisation comme composés pharmaceutiques - Google Patents

Dérivés substitués de l'acide 3-hétéroaroylamino-propionique et leur utilisation comme composés pharmaceutiques

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Publication number
MA34917B1
MA34917B1 MA36196A MA36196A MA34917B1 MA 34917 B1 MA34917 B1 MA 34917B1 MA 36196 A MA36196 A MA 36196A MA 36196 A MA36196 A MA 36196A MA 34917 B1 MA34917 B1 MA 34917B1
Authority
MA
Morocco
Prior art keywords
compounds
heteroaroylamino
substituted
propionic acid
acid derivatives
Prior art date
Application number
MA36196A
Other languages
English (en)
Inventor
Klaus Wirth
Herman Schreuder
Christian Buning
Sven Ruf
Thorsten Sadowski
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44041622&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MA34917(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of MA34917B1 publication Critical patent/MA34917B1/fr

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Abstract

LA PRÉSENTE INVENTION CONCERNE DES COMPOSÉS DE FORMULE (I), DANS LAQUELLE A, D, E, L, G, R10, R30, R40, R50 ET R60 ONT LES SIGNIFICATIONS INDIQUÉES DANS LES REVENDICATIONS, LESDITS COMPOSÉS ÉTANT DES COMPOSÉS PHARMACEUTIQUES ACTIFS DE VALEUR. CE SONT DES INHIBITEURS DE LA PROTÉASE CATHEPSINE A, ET ILS SONT UTILES DANS LE TRAITEMENT DE MALADIES TELLES QUE L'ATHÉROSCLÉROSE, UNE INSUFFISANCE CARDIAQUE, DES MALADIES RÉNALES, DES MALADIES HÉPATIQUES OU DES MALADIES INFLAMMATOIRES, PAR EXEMPLE. L'INVENTION CONCERNE EN OUTRE DES PROCÉDÉS DE PRÉPARATION DES COMPOSÉS DE FORMULE I, LEUR UTILISATION ET DES COMPOSITIONS PHARMACEUTIQUES LES COMPRENANT.
MA36196A 2011-01-26 2012-01-26 Dérivés substitués de l'acide 3-hétéroaroylamino-propionique et leur utilisation comme composés pharmaceutiques MA34917B1 (fr)

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CA2822120A1 (fr) 2012-08-02
AU2012210513A1 (en) 2013-08-15
NZ613672A (en) 2015-04-24
HRP20161545T1 (hr) 2016-12-30
WO2012101197A1 (fr) 2012-08-02
US20120252809A1 (en) 2012-10-04
HK1187253A1 (zh) 2014-04-04
CN103442712B (zh) 2016-01-20
ES2604556T3 (es) 2017-03-07
CA2822120C (fr) 2019-02-26
IL249826A0 (en) 2017-02-28
CL2013002129A1 (es) 2013-12-20
RU2632897C2 (ru) 2017-10-11
UY33874A (es) 2012-08-31
SI2667870T1 (sl) 2016-12-30
RU2013139349A (ru) 2015-03-10
AU2012210513B2 (en) 2016-09-22
JP5957467B2 (ja) 2016-07-27
US8669370B2 (en) 2014-03-11
MX2013007608A (es) 2013-09-06
SG10201600592WA (en) 2016-02-26
IL227025A (en) 2017-05-29
DK2667870T3 (en) 2016-12-12
US20140194445A1 (en) 2014-07-10
AR085013A1 (es) 2013-08-07
US9120783B2 (en) 2015-09-01
CY1118844T1 (el) 2018-01-10
EP2667870A1 (fr) 2013-12-04
HUE029781T2 (en) 2017-04-28
US20140135328A1 (en) 2014-05-15
CN103442712A (zh) 2013-12-11
MX340370B (es) 2016-07-07
PL2667870T3 (pl) 2017-02-28
BR112013016508A2 (pt) 2016-09-27
LT2667870T (lt) 2016-12-12
ZA201304463B (en) 2014-02-26
MX347157B (es) 2017-04-18
SG191826A1 (en) 2013-08-30
PT2667870T (pt) 2016-11-16
IL249825A0 (en) 2017-02-28
KR20140007399A (ko) 2014-01-17
EP2667870B1 (fr) 2016-08-24
CO6761373A2 (es) 2013-09-30
US9029559B2 (en) 2015-05-12
JP2014505063A (ja) 2014-02-27

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