HK1187253A1 - 取代的 -雜芳酰基氨基-丙酸衍生物及其作為藥物的用途 - Google Patents

取代的 -雜芳酰基氨基-丙酸衍生物及其作為藥物的用途

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Publication number
HK1187253A1
HK1187253A1 HK14100230.4A HK14100230A HK1187253A1 HK 1187253 A1 HK1187253 A1 HK 1187253A1 HK 14100230 A HK14100230 A HK 14100230A HK 1187253 A1 HK1187253 A1 HK 1187253A1
Authority
HK
Hong Kong
Prior art keywords
heteroaroylamino
pharmaceuticals
substituted
propionic acid
acid derivatives
Prior art date
Application number
HK14100230.4A
Other languages
English (en)
Inventor
Sven Ruf
Thorsten Sadowski
Klaus Wirth
Herman Schreuder
Christian Buning
Original Assignee
Sanofi Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=44041622&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1187253(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Sanofi Sa filed Critical Sanofi Sa
Publication of HK1187253A1 publication Critical patent/HK1187253A1/zh

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    • C07D413/06Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/44Radicals substituted by doubly-bound oxygen, sulfur, or nitrogen atoms, or by two such atoms singly-bound to the same carbon atom
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    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • C07D213/04Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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HK14100230.4A 2011-01-26 2014-01-09 取代的 -雜芳酰基氨基-丙酸衍生物及其作為藥物的用途 HK1187253A1 (zh)

Applications Claiming Priority (2)

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EP11305078 2011-01-26
PCT/EP2012/051189 WO2012101197A1 (en) 2011-01-26 2012-01-26 Substituted 3-heteroaroylamino-propionic acid derivatives and their use as pharmaceuticals

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HK1187253A1 true HK1187253A1 (zh) 2014-04-04

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US (3) US8669370B2 (zh)
EP (1) EP2667870B1 (zh)
JP (1) JP5957467B2 (zh)
KR (1) KR20140007399A (zh)
CN (1) CN103442712B (zh)
AR (1) AR085013A1 (zh)
AU (1) AU2012210513B2 (zh)
BR (1) BR112013016508A2 (zh)
CA (1) CA2822120C (zh)
CL (1) CL2013002129A1 (zh)
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