LU80922A1 - 9-amino-et imino-dibenzopyrannes et leur utilisation therapeutique - Google Patents

9-amino-et imino-dibenzopyrannes et leur utilisation therapeutique

Info

Publication number
LU80922A1
LU80922A1 LU80922A LU80922A LU80922A1 LU 80922 A1 LU80922 A1 LU 80922A1 LU 80922 A LU80922 A LU 80922A LU 80922 A LU80922 A LU 80922A LU 80922 A1 LU80922 A1 LU 80922A1
Authority
LU
Luxembourg
Prior art keywords
dibenzopyrans
imino
amino
therapeutic use
therapeutic
Prior art date
Application number
LU80922A
Other languages
English (en)
French (fr)
Inventor
Allen Day William
Ralph Lavagnino Edward
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of LU80922A1 publication Critical patent/LU80922A1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D311/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings
    • C07D311/02Heterocyclic compounds containing six-membered rings having one oxygen atom as the only hetero atom, condensed with other rings ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D311/78Ring systems having three or more relevant rings
    • C07D311/80Dibenzopyrans; Hydrogenated dibenzopyrans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/02Non-specific cardiovascular stimulants, e.g. drugs for syncope, antihypotensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrane Compounds (AREA)
LU80922A 1978-02-17 1979-02-15 9-amino-et imino-dibenzopyrannes et leur utilisation therapeutique LU80922A1 (fr)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US05/878,844 US4152450A (en) 1978-02-17 1978-02-17 9-Amino-dibenzopyrans

Publications (1)

Publication Number Publication Date
LU80922A1 true LU80922A1 (fr) 1979-06-18

Family

ID=25372961

Family Applications (1)

Application Number Title Priority Date Filing Date
LU80922A LU80922A1 (fr) 1978-02-17 1979-02-15 9-amino-et imino-dibenzopyrannes et leur utilisation therapeutique

Country Status (29)

Country Link
US (1) US4152450A (pl)
EP (1) EP0003883B1 (pl)
JP (1) JPS54122278A (pl)
AR (2) AR224359A1 (pl)
AT (1) AT366039B (pl)
AU (1) AU518718B2 (pl)
BE (1) BE873981A (pl)
CA (1) CA1111425A (pl)
CH (1) CH638800A5 (pl)
CS (1) CS207769B2 (pl)
DD (1) DD142190A5 (pl)
DE (1) DE2963797D1 (pl)
DK (1) DK68179A (pl)
ES (4) ES477832A1 (pl)
FI (1) FI790503A (pl)
FR (1) FR2417510A1 (pl)
GB (1) GB2014571B (pl)
GR (1) GR71465B (pl)
HU (1) HU180729B (pl)
IE (1) IE47999B1 (pl)
IL (1) IL56582A0 (pl)
LU (1) LU80922A1 (pl)
NZ (1) NZ189591A (pl)
PH (1) PH14622A (pl)
PL (5) PL120661B1 (pl)
PT (1) PT69202A (pl)
RO (5) RO82370A (pl)
SU (1) SU812177A3 (pl)
ZA (1) ZA79726B (pl)

Families Citing this family (28)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4309545A (en) * 1980-07-28 1982-01-05 Pfizer Inc. Oximino-1-hydroxyoctahydrobenzo[c]quinolines and derivatives thereof
US4351833A (en) * 1980-07-28 1982-09-28 Pfizer Inc. 9-Amino-1-hydroxyoctahydrobenzo[c]quinolines and derivatives thereof as analgesics and anti-emetics
US4863934A (en) * 1982-03-16 1989-09-05 Pfizer Inc. Bicyclic benzo fused pyran compounds used for producing analgesia
US4473704A (en) * 1982-03-16 1984-09-25 Pfizer Inc. Substituted dodecahydrotriphenylenes, decahydro-1H-cyclopenta[1]phenanthrenes, decahydro-1H-pyrido[1,2-f]phenanthridines and decahydropyrrolo[1,2-f]phenanthridines as CNS agents
US4841078A (en) * 1982-03-16 1989-06-20 Pfizer Inc. Benzopyrans
US4870084A (en) * 1982-03-16 1989-09-26 Pfizer Inc. Bicyclic benzo fused pyran compounds used for nausea treatment and prevention
US4642373A (en) * 1982-03-16 1987-02-10 Pfizer Inc. Substituted dodecahydrotripheylenes, and decahydropyrrolo[1,2-f]phenanthridines as CNS agents
US4486428A (en) * 1982-03-16 1984-12-04 Pfizer Inc. Bicyclic benzo fused compounds
US4442089A (en) * 1982-07-06 1984-04-10 E. R. Squibb & Sons, Inc. Method for treating glaucoma with topical or systemic ACE inhibitor compositions
US4680404A (en) * 1983-01-13 1987-07-14 Pfizer Inc. Benzopyrans
US5180736A (en) * 1989-03-23 1993-01-19 Warner-Lambert Company Polycyclic amines useful as cerebrovascular agents
WO1999057106A1 (en) * 1998-05-04 1999-11-11 The University Of Connecticut Novel analgesic and immunomodulatory cannabinoids
US7897598B2 (en) * 1998-06-09 2011-03-01 Alexandros Makriyannis Inhibitors of the anandamide transporter
US7589220B2 (en) * 1998-06-09 2009-09-15 University Of Connecticut Inhibitors of the anandamide transporter
US7161016B1 (en) 1998-11-24 2007-01-09 University Of Connecticut Cannabimimetic lipid amides as useful medications
US7276613B1 (en) 1998-11-24 2007-10-02 University Of Connecticut Retro-anandamides, high affinity and stability cannabinoid receptor ligands
CA2387764A1 (en) 1999-10-18 2001-04-26 University Of Connecticut Peripheral cannabinoid receptor (cb2) selective ligands
US7119108B1 (en) * 1999-10-18 2006-10-10 University Of Connecticut Pyrazole derivatives as cannabinoid receptor antagonists
US7741365B2 (en) * 1999-10-18 2010-06-22 University Of Connecticut Peripheral cannabinoid receptor (CB2) selective ligands
US7393842B2 (en) * 2001-08-31 2008-07-01 University Of Connecticut Pyrazole analogs acting on cannabinoid receptors
US6900236B1 (en) 1999-10-18 2005-05-31 University Of Connecticut Cannabimimetic indole derivatives
US8084467B2 (en) * 1999-10-18 2011-12-27 University Of Connecticut Pyrazole derivatives as cannabinoid receptor antagonists
US6943266B1 (en) 1999-10-18 2005-09-13 University Of Connecticut Bicyclic cannabinoid agonists for the cannabinoid receptor
JP2004532185A (ja) * 2001-01-26 2004-10-21 ユニバーシティ オブ コネチカット 新規なカンナビミメティックリガンド
CA2436133A1 (en) 2001-01-29 2002-08-08 University Of Connecticut Receptor selective cannabimimetic aminoalkylindoles
US7057076B2 (en) 2001-07-13 2006-06-06 University Of Connecticut Bicyclic and tricyclic cannabinoids
EP1448557A4 (en) * 2001-10-26 2005-02-02 Univ Connecticut HETEROINDANE: A NEW CLASS OF HIGH-ACTIVITY CANNABIMIMETIC LIGANDS
CA2496097A1 (en) 2002-08-23 2004-03-04 University Of Connecticut Keto cannabinoids with therapeutic indications

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3676462A (en) * 1970-01-08 1972-07-11 Little Inc A 7,8,9,10-TETRAHYDRO (AND 7,8,9,10,11,12-HEXAHYDRO) 6H-DIBENZO {8 b,d{9 {0 PYRANS
US3649650A (en) * 1970-02-13 1972-03-14 Little Inc A Novel derivatives of tetrahydro-cannabinol
AU7612874A (en) * 1973-12-27 1976-06-10 Erba Carlo Spa Benzopyran derivatives

Also Published As

Publication number Publication date
ATA123979A (de) 1981-07-15
AT366039B (de) 1982-03-10
CH638800A5 (fr) 1983-10-14
RO82370A (ro) 1983-08-03
AU4398379A (en) 1979-08-23
RO82370B (ro) 1983-07-30
PL213479A1 (pl) 1980-03-10
AR225939A1 (es) 1982-05-14
RO82376A (ro) 1983-08-03
ES8502106A1 (es) 1980-07-16
US4152450A (en) 1979-05-01
PL121009B1 (en) 1982-04-30
ES485619A0 (es) 1980-07-16
RO82369A (ro) 1983-08-03
GR71465B (pl) 1983-05-30
AU518718B2 (en) 1981-10-15
RO82375A (ro) 1983-08-03
ES485620A0 (es) 1980-07-16
JPS54122278A (en) 1979-09-21
PL120658B1 (en) 1982-03-31
IE47999B1 (en) 1984-08-22
ES8502105A1 (es) 1980-07-16
FI790503A (fi) 1979-08-18
BE873981A (fr) 1979-08-07
DK68179A (da) 1979-09-17
IL56582A0 (en) 1979-05-31
PT69202A (en) 1979-03-01
DD142190A5 (de) 1980-06-11
DE2963797D1 (en) 1982-11-11
RO82376B (ro) 1983-07-30
GB2014571B (en) 1982-11-17
RO76886A (ro) 1982-02-01
GB2014571A (en) 1979-08-30
AR224359A1 (es) 1981-11-30
IE790304L (en) 1979-08-17
ZA79726B (en) 1980-10-29
ES485621A1 (es) 1980-07-01
SU812177A3 (ru) 1981-03-07
RO82369B (ro) 1983-07-30
CS207769B2 (en) 1981-08-31
EP0003883B1 (en) 1982-10-06
PL120661B1 (en) 1982-03-31
CA1111425A (en) 1981-10-27
PL118576B1 (en) 1981-10-31
PH14622A (en) 1981-10-12
ES477832A1 (es) 1980-04-01
FR2417510B1 (pl) 1980-08-14
FR2417510A1 (fr) 1979-09-14
NZ189591A (en) 1980-10-08
PL120645B1 (en) 1982-03-31
EP0003883A1 (en) 1979-09-05
HU180729B (en) 1983-04-29

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