KR20120087875A - Ｇｉｐ 수용체-활성 글루카곤 화합물 - Google Patents

Ｇｉｐ 수용체-활성 글루카곤 화합물 Download PDF

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KR20120087875A
KR20120087875A KR20127000871A KR20127000871A KR20120087875A KR 20120087875 A KR20120087875 A KR 20120087875A KR 20127000871 A KR20127000871 A KR 20127000871A KR 20127000871 A KR20127000871 A KR 20127000871A KR 20120087875 A KR20120087875 A KR 20120087875A
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South Korea
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amino acid
glucagon
seq
analog
peptide
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Korean (ko)
Inventor
리차드 디. 디마르치
데이비드 엘. 스밀레이
마리아 디마르치
조셉 차벤네
조나단 데이
제임스 패터슨
브라이언 피. 와드
마 타오
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인디애나 유니버시티 리서치 앤드 테크놀로지 코퍼레이션
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Publication of KR20120087875A publication Critical patent/KR20120087875A/ko
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/605—Glucagons
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/26—Glucagons

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Diabetes (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Endocrinology (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Genetics & Genomics (AREA)
  • Toxicology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Medicinal Preparation (AREA)
KR20127000871A 2009-06-16 2010-06-16 Ｇｉｐ 수용체-활성 글루카곤 화합물 Ceased KR20120087875A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US18757809P 2009-06-16 2009-06-16
US61/187,578 2009-06-16
PCT/US2010/038825 WO2010148089A1 (en) 2009-06-16 2010-06-16 Gip receptor-active glucagon compounds

Publications (1)

Publication Number Publication Date
KR20120087875A true KR20120087875A (ko) 2012-08-07

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KR20127000871A Ceased KR20120087875A (ko) 2009-06-16 2010-06-16 Ｇｉｐ 수용체-활성 글루카곤 화합물

Country Status (17)

Country Link
US (2) US9150632B2 (en:Method)
EP (1) EP2443146B1 (en:Method)
JP (1) JP5887265B2 (en:Method)
KR (1) KR20120087875A (en:Method)
CN (1) CN102459325B (en:Method)
AU (1) AU2010260058B2 (en:Method)
BR (1) BRPI1014508A2 (en:Method)
CA (1) CA2765026A1 (en:Method)
CL (1) CL2011003173A1 (en:Method)
IL (1) IL216881A (en:Method)
IN (1) IN2012DN00377A (en:Method)
MX (1) MX2011013625A (en:Method)
PE (1) PE20120914A1 (en:Method)
RU (1) RU2012101274A (en:Method)
SG (1) SG176858A1 (en:Method)
TW (1) TWI549687B (en:Method)
WO (1) WO2010148089A1 (en:Method)

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* Cited by examiner, † Cited by third party
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