KR19990063676A - 신규한 환상 데프시펩티드 pf1022 유도체 - Google Patents

신규한 환상 데프시펩티드 pf1022 유도체 Download PDF

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Publication number
KR19990063676A
KR19990063676A KR1019980702138A KR19980702138A KR19990063676A KR 19990063676 A KR19990063676 A KR 19990063676A KR 1019980702138 A KR1019980702138 A KR 1019980702138A KR 19980702138 A KR19980702138 A KR 19980702138A KR 19990063676 A KR19990063676 A KR 19990063676A
Authority
KR
South Korea
Prior art keywords
group
meleu
phlac
lac
alkoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
KR1019980702138A
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English (en)
Korean (ko)
Inventor
오사무 사카나카
유미코 오카다
마코토 오오야마
마키 마츄모토
마사아키 타카하시
야수시 무라이
카튜하루 이이누마
아킴 하아더
놀베르 멘케
겔하아드 본스
피터 제쉬케
Original Assignee
빌프리더 하이더
바이엘 악티엔게젤샤프트
이치로 키타사토
메이지 세이카 카이샤 리미티드
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 빌프리더 하이더, 바이엘 악티엔게젤샤프트, 이치로 키타사토, 메이지 세이카 카이샤 리미티드 filed Critical 빌프리더 하이더
Publication of KR19990063676A publication Critical patent/KR19990063676A/ko
Ceased legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D273/00—Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
KR1019980702138A 1995-09-22 1996-09-20 신규한 환상 데프시펩티드 pf1022 유도체 Ceased KR19990063676A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP24405195 1995-09-22
JP7-244051 1995-09-22
PCT/JP1996/002730 WO1997011064A1 (en) 1995-09-22 1996-09-20 Novel cyclic depsipeptide pf1022 derivatives

Publications (1)

Publication Number Publication Date
KR19990063676A true KR19990063676A (ko) 1999-07-26

Family

ID=17113003

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019980702138A Ceased KR19990063676A (ko) 1995-09-22 1996-09-20 신규한 환상 데프시펩티드 pf1022 유도체

Country Status (18)

Country Link
US (1) US6329338B1 (enExample)
EP (1) EP0903347B1 (enExample)
KR (1) KR19990063676A (enExample)
CN (1) CN1082051C (enExample)
AT (1) ATE299871T1 (enExample)
AU (1) AU727532B2 (enExample)
BR (1) BR9610527A (enExample)
CA (1) CA2232668C (enExample)
CZ (1) CZ295705B6 (enExample)
DE (1) DE69634961T2 (enExample)
DK (1) DK0903347T3 (enExample)
ES (1) ES2246496T3 (enExample)
HU (1) HU228004B1 (enExample)
IL (1) IL123776A (enExample)
NO (1) NO310622B1 (enExample)
NZ (1) NZ318515A (enExample)
PL (1) PL186168B1 (enExample)
WO (1) WO1997011064A1 (enExample)

Families Citing this family (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0930304A4 (en) * 1996-08-07 2000-03-01 Meiji Seika Co METHOD FOR PRODUCING CYCLODEPSIPEPTID COMPOUNDS AND CYCLODEPSIPEPTID
WO1998037088A1 (en) * 1997-02-19 1998-08-27 Meiji Seika Kaisha Ltd. Derivatives of cyclodepsipeptide, pf1022 substance
DE19811559A1 (de) * 1998-03-17 1999-09-23 Bayer Ag Cyclooctadepsipeptide
CN100489095C (zh) 1999-09-29 2009-05-20 明治制果株式会社 生产被官能团修饰的次级代谢产物的转化体和新的生物合成基因
DE10031044A1 (de) * 2000-06-26 2002-01-03 Bayer Ag Endoparasitizide Mittel zur freiwilligen oralen Aufnahme durch Tiere
DE10104362A1 (de) * 2001-02-01 2002-08-08 Bayer Ag Kristallmodifikation eines cyclischen Depsipeptids mit besserer Wirksamkeit
DE102004055316A1 (de) * 2004-11-16 2006-05-18 Bayer Healthcare Ag Verhinderung vertikaler Endoparasiten-Infektionen
DE102008022520A1 (de) 2008-05-07 2009-11-12 Bayer Animal Health Gmbh Feste Arzneimittelformulierung mit verzögerter Freisetzung
DE102008030764A1 (de) 2008-06-28 2009-12-31 Bayer Animal Health Gmbh Kombination von Amidin-Derivaten mit cyclischen Depsipeptiden
DE102008031283A1 (de) * 2008-07-02 2010-01-07 Bayer Schering Pharma Aktiengesellschaft Neue Bekämpfungsmöglichkeit von durch Trichomonadida hervorgerufenen Krankheiten
DE102008031284A1 (de) * 2008-07-02 2010-01-07 Bayer Schering Pharma Aktiengesellschaft Neue Bekämpfungsmöglichkeit der Giardiose
DE102009012423A1 (de) 2009-03-10 2010-09-16 Bayer Animal Health Gmbh Zubereitung auf Ölbasis
DE102010064245A1 (de) 2010-12-28 2012-06-28 Bayer Animal Health Gmbh Makrocylischen Lactone und deren Verwendung und deren Kombinationen mit anderen Wirkstoffen
WO2012028556A1 (en) 2010-08-31 2012-03-08 Bayer Animal Health Gmbh Macrocyclic lactones and their use and their combinations with other active substances
US10081656B2 (en) 2015-05-20 2018-09-25 Merial, Inc. Anthelmintic depsipeptide compounds
HUE065907T2 (hu) 2015-12-28 2024-06-28 Boehringer Ingelheim Vetmedica Gmbh Anthelmintikus hatású depszipeptid vegyületek
EP3541789A1 (en) 2016-11-16 2019-09-25 Boehringer Ingelheim Animal Health USA Inc. Anthelmintic depsipeptide compounds
MY203299A (en) 2017-11-07 2024-06-21 The Kitasato Inst Method for the synthesis of cyclic depsipeptides
RU2747149C9 (ru) 2017-11-29 2021-06-29 ЗОЕТИС СЕРВИСИЗ ЭлЭлСи Анти-эндопаразитарные депсипептиды
SG11202010187RA (en) 2018-05-10 2020-11-27 Zoetis Services Llc Endoparasitic depsipeptides

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH477172A (de) * 1965-05-18 1969-08-31 Agripat Sa Beifuttermittel
AU1933583A (en) * 1982-09-22 1984-03-29 Meiji Seika K.K. Hydroxylamine derivatives
NO176766C (no) * 1989-02-07 1995-05-24 Meiji Seika Kaisha Fremgangsmåte for fremstilling av en forbindelse med anthelmintaktivitet
ES2166359T3 (es) * 1992-03-17 2002-04-16 Fujisawa Pharmaceutical Co Derivado de depsipeptido, su produccion y uso.
JP2873894B2 (ja) * 1992-10-19 1999-03-24 明治製菓株式会社 環状デプシペプチドおよびその製造法
EP0685469A4 (en) * 1993-02-19 1996-04-03 Meiji Seika Kaisha DERIVATIVE OF PF 1022 USED AS A CYCLIC DEPSIPEPTIDE.
DE4317432A1 (de) * 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung
DE4317457A1 (de) 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung
JPH07233068A (ja) * 1993-12-27 1995-09-05 Meiji Seika Kaisha Ltd 高コレステロール血症、高脂血症又は動脈硬化症の治療薬

Also Published As

Publication number Publication date
DK0903347T3 (da) 2005-11-21
ATE299871T1 (de) 2005-08-15
DE69634961T2 (de) 2006-04-20
HUP0001164A2 (hu) 2000-11-28
WO1997011064A1 (en) 1997-03-27
CA2232668C (en) 2011-10-18
PL326024A1 (en) 1998-08-17
NO981250D0 (no) 1998-03-19
CA2232668A1 (en) 1997-03-27
BR9610527A (pt) 1999-12-21
EP0903347A1 (en) 1999-03-24
AU7001996A (en) 1997-04-09
DE69634961D1 (de) 2005-08-25
HUP0001164A3 (en) 2001-04-28
NO981250L (no) 1998-05-22
IL123776A0 (en) 1998-10-30
US6329338B1 (en) 2001-12-11
NZ318515A (en) 2000-05-26
ES2246496T3 (es) 2006-02-16
CZ85598A3 (cs) 1998-08-12
MX9802268A (es) 1998-08-30
PL186168B1 (pl) 2003-11-28
AU727532B2 (en) 2000-12-14
HU228004B1 (en) 2012-08-28
JP4001381B1 (enExample) 2007-10-31
EP0903347A4 (enExample) 1999-03-24
NO310622B1 (no) 2001-07-30
CN1201456A (zh) 1998-12-09
IL123776A (en) 2002-09-12
CN1082051C (zh) 2002-04-03
EP0903347B1 (en) 2005-07-20
CZ295705B6 (cs) 2005-10-12

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