KR101834024B1 - 치환된 베타―시클로덱스트린에 의해 안정화된 포사코나졸 정맥내 용액 제제 - Google Patents

치환된 베타―시클로덱스트린에 의해 안정화된 포사코나졸 정맥내 용액 제제 Download PDF

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KR101834024B1
KR101834024B1 KR1020127034087A KR20127034087A KR101834024B1 KR 101834024 B1 KR101834024 B1 KR 101834024B1 KR 1020127034087 A KR1020127034087 A KR 1020127034087A KR 20127034087 A KR20127034087 A KR 20127034087A KR 101834024 B1 KR101834024 B1 KR 101834024B1
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posaconazole
pharmaceutical composition
cyclodextrin
solution
composition according
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KR20130114603A (ko
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수잔 케이. 헤임베처
데이비드 몬테이스
제임스 디. 핍킨
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머크 샤프 앤드 돔 코포레이션
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  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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KR1020127034087A 2010-06-29 2011-06-24 치환된 베타―시클로덱스트린에 의해 안정화된 포사코나졸 정맥내 용액 제제 Active KR101834024B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US35970110P 2010-06-29 2010-06-29
US61/359,701 2010-06-29
PCT/US2011/041715 WO2012005973A1 (en) 2010-06-29 2011-06-24 Posaconazole intravenous solution formulations stabilized by substituted beta-cyclodextrin

Publications (2)

Publication Number Publication Date
KR20130114603A KR20130114603A (ko) 2013-10-17
KR101834024B1 true KR101834024B1 (ko) 2018-03-02

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US (2) US9023790B2 (https=)
EP (3) EP3391890B1 (https=)
JP (1) JP6008849B2 (https=)
KR (1) KR101834024B1 (https=)
CN (2) CN102958528A (https=)
AU (1) AU2011276680B2 (https=)
BR (1) BR112012033077B8 (https=)
CA (1) CA2802929C (https=)
CY (1) CY1124690T1 (https=)
DK (1) DK3391890T3 (https=)
ES (1) ES2893444T3 (https=)
HR (1) HRP20211686T1 (https=)
HU (1) HUE056581T2 (https=)
LT (1) LT3391890T (https=)
MX (2) MX338685B (https=)
PL (1) PL3391890T3 (https=)
PT (1) PT3391890T (https=)
RS (1) RS62583B1 (https=)
SI (1) SI3391890T1 (https=)
WO (1) WO2012005973A1 (https=)

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HUE056581T2 (hu) 2010-06-29 2022-02-28 Merck Sharp & Dohme Szubsztituált béta-ciklodextrinnel stabilizált pozakonazol intravénás oldat formulációk
US8039494B1 (en) 2010-07-08 2011-10-18 Dow Pharmaceutical Sciences, Inc. Compositions and methods for treating diseases of the nail
DK3702374T3 (da) 2012-02-15 2022-06-27 Cydex Pharmaceuticals Inc Fremsgangsmåde til fremstilling for cyclodextrin-derivater
SG11201602596UA (en) 2013-10-03 2016-04-28 Dow Pharmaceutical Sciences Stabilized efinaconazole compositions
CN104546724A (zh) * 2013-10-12 2015-04-29 博瑞生物医药技术(苏州)有限公司 一种抗真菌药的固体分散体
KR102612453B1 (ko) 2013-11-22 2023-12-08 다우 파마슈티컬 사이언시즈, 인코포레이티드 항­감염 방법，조성물，및 장치
CN105879041A (zh) * 2014-11-14 2016-08-24 北京赛林泰医药技术有限公司 一种泊沙康唑口服液及其制备方法
WO2016079749A2 (en) * 2014-11-19 2016-05-26 Gufic Biosciences Limited Process for preparation of parenteral formulation of anidulafungin
CN104473871B (zh) * 2014-11-28 2017-03-08 济南康和医药科技有限公司 一种泊沙康唑脂肪乳注射液及其制备方法
CN106265534A (zh) * 2015-05-25 2017-01-04 江苏正大丰海制药有限公司 一种泊沙康唑冻干粉针剂的制备方法
CN106511262A (zh) * 2015-09-11 2017-03-22 上海美悦生物科技发展有限公司 一种泊沙康唑口服溶液剂及其制备方法
US10517867B2 (en) 2016-02-04 2019-12-31 Wuhan Ll Science And Technology Development Co., Ltd. Posaconazole derivative, pharmaceutical composition and use thereof
TW201828938A (zh) 2016-11-18 2018-08-16 德商艾庫里斯抗感染治療有限公司 以改質的環糊精及酸化劑為基底之經脒取代之β-內醯胺化合物的新穎調配物，其製備方法及作為抗微生物醫藥組合物之用途
AU2019254483B2 (en) 2018-04-16 2025-02-27 Merck Patent Gmbh Viscosity reduction of highly concentrated protein formulations
CN110711174A (zh) * 2018-07-11 2020-01-21 郑州泰丰制药有限公司 一种泊沙康唑注射液中间体溶液配制方法
TR201820816A2 (tr) * 2018-12-28 2020-07-21 Polifarma Ilac Sanayi Ve Ticaret Anonim Sirketi Si̇klodekstri̇n ve şeker i̇çeren stabi̇l enjekte edi̇lebi̇li̇r posakonazol formülasyonlari
WO2021245703A2 (en) * 2020-06-06 2021-12-09 Inventia Healthcare Limited Stable liquid compositions of posaconazole
CN115429748A (zh) * 2021-06-02 2022-12-06 江苏奥赛康药业有限公司 一种泊沙康唑注射液的制备方法
WO2023148763A1 (en) * 2022-02-01 2023-08-10 Cipla Limited Injectable pharmaceutical compositions of azole antifungal agents

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