SI3391890T1 - Formulacije intravenske raztopine posakonazola, stabilizirane s substituiranim beta-ciklodekstrinom - Google Patents

Formulacije intravenske raztopine posakonazola, stabilizirane s substituiranim beta-ciklodekstrinom

Info

Publication number
SI3391890T1
SI3391890T1 SI201132006T SI201132006T SI3391890T1 SI 3391890 T1 SI3391890 T1 SI 3391890T1 SI 201132006 T SI201132006 T SI 201132006T SI 201132006 T SI201132006 T SI 201132006T SI 3391890 T1 SI3391890 T1 SI 3391890T1
Authority
SI
Slovenia
Prior art keywords
cyclodextrin
intravenous solution
solution formulations
substituted beta
formulations stabilized
Prior art date
Application number
SI201132006T
Other languages
English (en)
Slovenian (sl)
Inventor
Susan K. Heimbecher
David Monteith
Original Assignee
Merck Sharp & Dohme Corp.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=45441500&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI3391890(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Merck Sharp & Dohme Corp. filed Critical Merck Sharp & Dohme Corp.
Publication of SI3391890T1 publication Critical patent/SI3391890T1/sl

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/40—Cyclodextrins; Derivatives thereof
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965—Non-condensed pyrazines
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
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    • A61K31/715—Polysaccharides, i.e. having more than five saccharide radicals attached to each other by glycosidic linkages; Derivatives thereof, e.g. ethers, esters
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    • A61K47/6957—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the conjugate being characterised by physical or galenical forms, e.g. emulsion, particle, inclusion complex, stent or kit the form being a device or a kit, e.g. stents or microdevices
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    • A61P31/10—Antimycotics
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    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
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  • AIDS & HIV (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medical Preparation Storing Or Oral Administration Devices (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
SI201132006T 2010-06-29 2011-06-24 Formulacije intravenske raztopine posakonazola, stabilizirane s substituiranim beta-ciklodekstrinom SI3391890T1 (sl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US35970110P 2010-06-29 2010-06-29
EP18171672.1A EP3391890B1 (en) 2010-06-29 2011-06-24 Posaconazole intravenous solution formulations stabilized by substituted beta-cyclodextrin

Publications (1)

Publication Number Publication Date
SI3391890T1 true SI3391890T1 (sl) 2021-11-30

Family

ID=45441500

Family Applications (1)

Application Number Title Priority Date Filing Date
SI201132006T SI3391890T1 (sl) 2010-06-29 2011-06-24 Formulacije intravenske raztopine posakonazola, stabilizirane s substituiranim beta-ciklodekstrinom

Country Status (20)

Country Link
US (2) US9023790B2 (https=)
EP (3) EP3960185A1 (https=)
JP (1) JP6008849B2 (https=)
KR (1) KR101834024B1 (https=)
CN (2) CN102958528A (https=)
AU (1) AU2011276680B2 (https=)
BR (1) BR112012033077B8 (https=)
CA (1) CA2802929C (https=)
CY (1) CY1124690T1 (https=)
DK (1) DK3391890T3 (https=)
ES (1) ES2893444T3 (https=)
HR (1) HRP20211686T1 (https=)
HU (1) HUE056581T2 (https=)
LT (1) LT3391890T (https=)
MX (2) MX338685B (https=)
PL (1) PL3391890T3 (https=)
PT (1) PT3391890T (https=)
RS (1) RS62583B1 (https=)
SI (1) SI3391890T1 (https=)
WO (1) WO2012005973A1 (https=)

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