KR101712083B1 - 피라졸 카르복실산 아미드의 제조 방법 - Google Patents

피라졸 카르복실산 아미드의 제조 방법 Download PDF

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KR101712083B1
KR101712083B1 KR1020127005767A KR20127005767A KR101712083B1 KR 101712083 B1 KR101712083 B1 KR 101712083B1 KR 1020127005767 A KR1020127005767 A KR 1020127005767A KR 20127005767 A KR20127005767 A KR 20127005767A KR 101712083 B1 KR101712083 B1 KR 101712083B1
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formula
compound
acid
compounds
viii
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KR20120043059A (ko
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데니스 그리브코프
아드리안 뮐러
마르텡 라게르
파니 조르다노
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신젠타 파티서페이션즈 아게
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C251/00—Compounds containing nitrogen atoms doubly-bound to a carbon skeleton
    • C07C251/32—Oximes
    • C07C251/34—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals
    • C07C251/44—Oximes with oxygen atoms of oxyimino groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with the carbon atom of at least one of the oxyimino groups being part of a ring other than a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/62—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by hydrogenation of carbon-to-carbon double or triple bonds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/65—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by splitting-off hydrogen atoms or functional groups; by hydrogenolysis of functional groups
    • C07C45/66—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by splitting-off hydrogen atoms or functional groups; by hydrogenolysis of functional groups by dehydration
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/61—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups
    • C07C45/67—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton
    • C07C45/68—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
    • C07C45/69—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by reactions not involving the formation of >C = O groups by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms by addition to carbon-to-carbon double or triple bonds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/587—Unsaturated compounds containing a keto groups being part of a ring
    • C07C49/687—Unsaturated compounds containing a keto groups being part of a ring containing halogen
    • C07C49/693—Unsaturated compounds containing a keto groups being part of a ring containing halogen polycyclic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C49/00—Ketones; Ketenes; Dimeric ketenes; Ketonic chelates
    • C07C49/587—Unsaturated compounds containing a keto groups being part of a ring
    • C07C49/703—Unsaturated compounds containing a keto groups being part of a ring containing hydroxy groups
    • C07C49/743—Unsaturated compounds containing a keto groups being part of a ring containing hydroxy groups having unsaturation outside the rings, e.g. humulones, lupulones
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D251/00—Heterocyclic compounds containing 1,3,5-triazine rings
    • C07D251/02—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings
    • C07D251/12—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
    • C07D251/26—Heterocyclic compounds containing 1,3,5-triazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with only hetero atoms directly attached to ring carbon atoms
    • C07D251/40—Nitrogen atoms
    • C07D251/42—One nitrogen atom
    • C07D251/44—One nitrogen atom with halogen atoms attached to the two other ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/56—Ring systems containing bridged rings
    • C07C2603/58—Ring systems containing bridged rings containing three rings
    • C07C2603/60—Ring systems containing bridged rings containing three rings containing at least one ring with less than six members
    • C07C2603/66—Ring systems containing bridged rings containing three rings containing at least one ring with less than six members containing five-membered rings

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
KR1020127005767A 2009-08-06 2010-07-07 피라졸 카르복실산 아미드의 제조 방법 Active KR101712083B1 (ko)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP09167363.2 2009-08-06
EP09167363 2009-08-06
EP09169501.5 2009-09-04
EP09169501 2009-09-04
PCT/EP2010/059703 WO2011015416A1 (en) 2009-08-06 2010-07-07 Process for the preparation of pyrazole carboxylic acid amides

Publications (2)

Publication Number Publication Date
KR20120043059A KR20120043059A (ko) 2012-05-03
KR101712083B1 true KR101712083B1 (ko) 2017-03-03

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KR1020127005767A Active KR101712083B1 (ko) 2009-08-06 2010-07-07 피라졸 카르복실산 아미드의 제조 방법

Country Status (28)

Country Link
US (1) US8507694B2 (enExample)
EP (1) EP2462108B1 (enExample)
JP (1) JP5667186B2 (enExample)
KR (1) KR101712083B1 (enExample)
CN (1) CN102574779B (enExample)
AR (1) AR077707A1 (enExample)
AU (1) AU2010280923B2 (enExample)
BR (1) BR112012002641B1 (enExample)
CA (1) CA2770144C (enExample)
CL (1) CL2012000272A1 (enExample)
CO (1) CO6430457A2 (enExample)
CR (1) CR20120056A (enExample)
DK (1) DK2462108T3 (enExample)
EA (1) EA019475B1 (enExample)
EC (1) ECSP12011647A (enExample)
EG (1) EG26957A (enExample)
ES (1) ES2417315T3 (enExample)
GE (1) GEP20146010B (enExample)
IL (1) IL217692A (enExample)
IN (1) IN2012DN00289A (enExample)
MX (1) MX2012001480A (enExample)
MY (1) MY161666A (enExample)
NZ (1) NZ597576A (enExample)
PL (1) PL2462108T3 (enExample)
TW (1) TWI441812B (enExample)
UY (1) UY32835A (enExample)
WO (1) WO2011015416A1 (enExample)
ZA (1) ZA201200413B (enExample)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI534126B (zh) 2011-01-25 2016-05-21 先正達合夥公司 用於製備吡唑羧酸醯胺之方法
TWI510472B (zh) * 2012-02-15 2015-12-01 Syngenta Participations Ag 立體選擇性製備吡唑羧醯胺之方法
GB201403438D0 (en) * 2014-02-27 2014-04-16 Syngenta Participations Ag Polymorphs
EP3119200A4 (en) 2014-03-20 2017-08-23 Mitsui Chemicals Agro, Inc. Plant disease control composition and method for controlling plant disease by application of same
IL318101A (en) 2022-07-22 2025-02-01 Syngenta Crop Protection Ag Solid form of a heterocyclic amide derivative
CN120835879A (zh) * 2022-10-11 2025-10-24 先正达农作物保护股份公司 用于制备吡唑羧酸酰胺的方法
CN117362179B (zh) * 2023-09-22 2025-07-08 浙江工业大学 一种苯并烯氟菌唑中间体9-二氯亚甲基-1,4-二氢-5-硝基-1,4-甲桥萘的制备方法
TW202545915A (zh) 2024-01-26 2025-12-01 瑞士商先正達農作物保護股份公司 化學方法

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4370341A (en) * 1980-12-11 1983-01-25 Ayerst, Mckenna & Harrison, Ltd. 6,7,8,9-Tetrahydro-3H-benz[E]indol-8-amine derivatives
JPS58194853A (ja) * 1982-05-11 1983-11-12 Showa Denko Kk シクロヘキセン−アセチルオキシム誘導体
US5093347A (en) 1991-01-28 1992-03-03 Monsanto Company 3-difluoromethylpyrazolecarboxamide fungicides, compositions and use
US5932752A (en) * 1995-12-29 1999-08-03 Council Of Scientific And Industrial Research Process for the C-C bond forming reaction using solid acid catalysts
GB0224316D0 (en) * 2002-10-18 2002-11-27 Syngenta Participations Ag Chemical compounds
CN1618783A (zh) * 2004-04-22 2005-05-25 复旦大学 一种多取代苯醌的制备方法
EA014297B1 (ru) * 2005-10-25 2010-10-29 Зингента Партисипейшнс Аг Гетероциклические амиды, применимые в качестве микробиоцидов

Also Published As

Publication number Publication date
CN102574779B (zh) 2014-10-15
MY161666A (en) 2017-04-28
MX2012001480A (es) 2012-02-22
DK2462108T3 (da) 2013-07-08
ECSP12011647A (es) 2012-03-30
CA2770144C (en) 2017-03-21
CA2770144A1 (en) 2011-02-10
AR077707A1 (es) 2011-09-14
KR20120043059A (ko) 2012-05-03
EA201200246A1 (ru) 2012-08-30
EP2462108B1 (en) 2013-04-17
EP2462108A1 (en) 2012-06-13
NZ597576A (en) 2013-01-25
WO2011015416A1 (en) 2011-02-10
UY32835A (es) 2011-03-31
EG26957A (en) 2015-02-01
IL217692A (en) 2015-07-30
ES2417315T3 (es) 2013-08-07
IN2012DN00289A (enExample) 2015-05-08
CL2012000272A1 (es) 2012-09-28
TW201107297A (en) 2011-03-01
JP2013501016A (ja) 2013-01-10
US20120136162A1 (en) 2012-05-31
BR112012002641A2 (pt) 2016-03-22
PL2462108T3 (pl) 2013-09-30
CN102574779A (zh) 2012-07-11
GEP20146010B (en) 2014-01-10
CR20120056A (es) 2012-03-06
TWI441812B (zh) 2014-06-21
CO6430457A2 (es) 2012-04-30
AU2010280923B2 (en) 2014-08-07
JP5667186B2 (ja) 2015-02-12
EA019475B1 (ru) 2014-03-31
BR112012002641B1 (pt) 2018-05-22
ZA201200413B (en) 2012-10-31
AU2010280923A1 (en) 2012-02-09
US8507694B2 (en) 2013-08-13

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