KR101299426B1 - 오렉신 수용체 길항제로서의 치환된 디아제판 화합물 - Google Patents
오렉신 수용체 길항제로서의 치환된 디아제판 화합물 Download PDFInfo
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- KR101299426B1 KR101299426B1 KR1020107002786A KR20107002786A KR101299426B1 KR 101299426 B1 KR101299426 B1 KR 101299426B1 KR 1020107002786 A KR1020107002786 A KR 1020107002786A KR 20107002786 A KR20107002786 A KR 20107002786A KR 101299426 B1 KR101299426 B1 KR 101299426B1
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- triazol
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
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- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
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| PCT/US2007/024690 WO2008069997A1 (en) | 2006-12-01 | 2007-11-30 | Substituted diazepan compounds as orexin receptor antagonists |
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