KE3078A - 3-amino-indazoecarboxylic acid derivatives,process for their preparation and their use as medicaments - Google Patents

3-amino-indazoecarboxylic acid derivatives,process for their preparation and their use as medicaments

Info

Publication number
KE3078A
KE3078A KE3078A KE307880A KE3078A KE 3078 A KE3078 A KE 3078A KE 3078 A KE3078 A KE 3078A KE 307880 A KE307880 A KE 307880A KE 3078 A KE3078 A KE 3078A
Authority
KE
Kenya
Prior art keywords
indazoecarboxylic
medicaments
amino
preparation
acid derivatives
Prior art date
Application number
KE3078A
Other languages
English (en)
Inventor
K H Mayer
W Wuttke
E Klauke
S Petersen
F Hoffmeister
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of KE3078A publication Critical patent/KE3078A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
KE3078A 1974-12-13 1980-08-29 3-amino-indazoecarboxylic acid derivatives,process for their preparation and their use as medicaments KE3078A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE2458965A DE2458965C3 (de) 1974-12-13 1974-12-13 3-Amino-indazol-N-carbonsäure-Derivate, Verfahren zu ihrer Herstellung sowie sie enthaltende Arzneimittel

Publications (1)

Publication Number Publication Date
KE3078A true KE3078A (en) 1980-10-03

Family

ID=5933305

Family Applications (1)

Application Number Title Priority Date Filing Date
KE3078A KE3078A (en) 1974-12-13 1980-08-29 3-amino-indazoecarboxylic acid derivatives,process for their preparation and their use as medicaments

Country Status (27)

Country Link
US (1) US4051252A (enExample)
JP (1) JPS5182266A (enExample)
AT (1) AT343653B (enExample)
BE (1) BE836528A (enExample)
CA (1) CA1059523A (enExample)
CH (1) CH622250A5 (enExample)
CS (1) CS189731B2 (enExample)
DD (1) DD125484A5 (enExample)
DE (1) DE2458965C3 (enExample)
DK (1) DK137082C (enExample)
ES (1) ES443429A1 (enExample)
FI (1) FI753493A7 (enExample)
FR (1) FR2293928A1 (enExample)
GB (1) GB1490306A (enExample)
HK (1) HK52580A (enExample)
HU (1) HU173557B (enExample)
IE (1) IE42208B1 (enExample)
IL (1) IL48642A (enExample)
KE (1) KE3078A (enExample)
LU (1) LU73993A1 (enExample)
NL (1) NL7514521A (enExample)
NO (1) NO145382C (enExample)
PL (1) PL99858B1 (enExample)
SE (1) SE419645B (enExample)
SU (1) SU604487A3 (enExample)
YU (1) YU315275A (enExample)
ZA (1) ZA757777B (enExample)

Families Citing this family (39)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4431657A (en) * 1982-05-24 1984-02-14 Ayerst, Mckenna & Harrison Inc. Analgesic compositions consisting of 2H-benzothieno[3,2-c]pyrazol-3-amine derivatives
KR20010086657A (ko) * 2000-03-02 2001-09-15 성재갑 아미노인다졸 유도체 및 이를 함유하는 싸이클린 의존키나아제 저해제 조성물
US7473691B2 (en) * 2000-09-15 2009-01-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
US6660731B2 (en) 2000-09-15 2003-12-09 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
CN1926132B (zh) * 2000-09-15 2010-12-29 沃泰克斯药物股份有限公司 可用作蛋白激酶抑制剂的吡唑化合物
EP1698627A1 (en) * 2000-09-15 2006-09-06 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
AU2001290912A1 (en) * 2000-09-15 2002-03-26 Vertex Pharmaceuticals Incorporated Pyrazole compounds useful as protein kinase inhibitors
BR0116493A (pt) * 2000-12-21 2003-09-30 Vertex Pharma Compostos de pirazol úteis como inibidores de proteìna cinase
KR100406634B1 (ko) * 2001-03-12 2003-11-20 주식회사 엘지생명과학 3,5-디아미노인다졸 유도체, 그의 제조방법 및 사이클린의존성 키나아제 저해제로서의 그의 용도
KR20040047869A (ko) 2001-09-26 2004-06-05 파마시아 이탈리아 에스.피.에이. 키나제 억제제로서 활성인 아미노인다졸 유도체, 이의제조방법 및 이를 함유하는 약제학적 조성물
KR20040084896A (ko) * 2002-02-06 2004-10-06 버텍스 파마슈티칼스 인코포레이티드 Ｇｓｋ-3의 억제제로서 유용한 헤테로아릴 화합물
FR2836915B1 (fr) * 2002-03-11 2008-01-11 Aventis Pharma Sa Derives d'aminoindazoles, procede de preparation et intermediaires de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant
US20040009981A1 (en) 2002-03-15 2004-01-15 David Bebbington Compositions useful as inhibitors of protein kinases
WO2003097610A1 (en) 2002-05-17 2003-11-27 Pharmacia Italia S.P.A. Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
MY141867A (en) 2002-06-20 2010-07-16 Vertex Pharma Substituted pyrimidines useful as protein kinase inhibitors
MXPA05001367A (es) 2002-08-02 2005-04-28 Vertex Pharma Composiciones de pirazol utiles como inhibidores de gsk-3.
EP1556053A4 (en) * 2002-10-31 2006-04-19 Amgen Inc ANTI-INFLAMMATORY AGENTS
WO2004072029A2 (en) 2003-02-06 2004-08-26 Vertex Pharmaceuticals Incorporated Pyrazolopyridazines useful as inhibitors of protein kinases
CN1902193B (zh) * 2003-12-04 2011-07-13 沃泰克斯药物股份有限公司 可用作蛋白激酶抑制剂的喹喔啉
DE102004005172A1 (de) * 2004-02-02 2005-08-18 Aventis Pharma Deutschland Gmbh Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase
US7737151B2 (en) 2005-08-18 2010-06-15 Vertex Pharmaceuticals Incorporated Pyrazine kinase inhibitors
JP5249770B2 (ja) 2005-11-03 2013-07-31 バーテックス ファーマシューティカルズ インコーポレイテッド キナーゼインヒビターとして有用なアミノピリジン
UA94100C2 (ru) * 2006-04-14 2011-04-11 Эбботт Леборетриз Способ получения индазолилмочевин, которые угнетают ванилоидные рецепторы подтипа 1 (vr1)
CA2668429A1 (en) 2006-11-02 2008-05-15 Vertex Pharmaceuticals Incorporated Aminopyridines and aminopyrimidines useful as inhibitors of protein kinases
NZ577768A (en) 2006-12-19 2012-01-12 Vertex Pharma Aminopyrimidines useful as inhibitors of protein kinases
JP5393489B2 (ja) 2007-03-09 2014-01-22 バーテックス ファーマシューティカルズ インコーポレイテッド 蛋白キナーゼの阻害剤として有用なアミノピリミジン
CN101663295B (zh) 2007-03-09 2014-11-05 沃泰克斯药物股份有限公司 可用作蛋白激酶抑制剂的氨基嘧啶类化合物
NZ579483A (en) 2007-03-09 2012-07-27 Vertex Pharma Aminopyridines useful as inhibitors of protein kinases
MX2009011059A (es) 2007-04-13 2009-11-26 Vertex Pharma Aminopirimidinas utiles como inhibidores de cinasas.
WO2008137619A2 (en) * 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Thiazoles and pyrazoles useful as kinase inhibitors
CA2688584A1 (en) * 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
AU2008247594A1 (en) 2007-05-02 2008-11-13 Vertex Pharmaceuticals Incorporated Aminopyrimidines useful as kinase inhibitors
AU2008257044A1 (en) * 2007-05-24 2008-12-04 Vertex Pharmaceuticals Incorporated Thiazoles and pyrazoles useful as kinase inhibitors
WO2009018415A1 (en) 2007-07-31 2009-02-05 Vertex Pharmaceuticals Incorporated Process for preparing 5-fluoro-1h-pyrazolo [3, 4-b] pyridin-3-amine and derivatives thereof
AU2009288200A1 (en) * 2008-09-03 2010-03-11 Vertex Pharmaceuticals Incorporated Co-crystals and pharmaceutical formulations comprising the same
DE102009004245A1 (de) 2009-01-09 2010-07-15 Bayer Schering Pharma Aktiengesellschaft Neue anellierte, Heteroatom-verbrückte Pyrazol- und Imidazol-Derivate und ihre Verwendung
CA2879726A1 (en) 2012-07-24 2014-01-30 Bial- Portela & Ca, S.A. Urea compounds and their use as enzyme inhibitors
US20150197503A1 (en) * 2012-07-27 2015-07-16 Bial-Portela & Cª, S.A. Process for the synthesis of substituted urea compounds
WO2015012708A1 (en) 2013-07-24 2015-01-29 BIAL - PORTELA & Cª, S.A. Imidazolecarboxamides and their use as faah inhibitors

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3133081A (en) * 1964-05-12 J-aminoindazole derivatives
CH397698A (de) * 1961-09-08 1965-08-31 Siegfried Ag Verfahren zur Herstellung neuer 1-Carbamyl-indazole
US3274203A (en) * 1963-05-31 1966-09-20 Du Pont 1-carbamyl and thiocarbamyl-3-amino-4-nonsubstituted and substituted pyrazoles
NL6707299A (enExample) * 1966-07-16 1968-01-17
DE1770649A1 (de) * 1968-06-15 1971-11-11 Bayer Ag Substituierte 3-Amino-indazole

Also Published As

Publication number Publication date
ATA939775A (de) 1977-10-15
HK52580A (en) 1980-09-26
CA1059523A (en) 1979-07-31
LU73993A1 (enExample) 1976-11-11
FR2293928A1 (fr) 1976-07-09
YU315275A (en) 1982-02-28
DK137082B (da) 1978-01-16
IL48642A0 (en) 1976-02-29
DE2458965A1 (de) 1976-06-16
PL99858B1 (pl) 1978-08-31
ES443429A1 (es) 1977-04-16
FI753493A7 (enExample) 1976-06-14
CH622250A5 (enExample) 1981-03-31
ZA757777B (en) 1976-11-24
NO145382B (no) 1981-11-30
IL48642A (en) 1979-12-30
CS189731B2 (en) 1979-04-30
BE836528A (fr) 1976-06-11
FR2293928B1 (enExample) 1979-09-21
HU173557B (hu) 1979-06-28
DE2458965C3 (de) 1979-10-11
GB1490306A (en) 1977-11-02
SE419645B (sv) 1981-08-17
JPS5182266A (en) 1976-07-19
DK567275A (da) 1976-06-14
NL7514521A (nl) 1976-06-15
IE42208B1 (en) 1980-06-18
SU604487A3 (ru) 1978-04-25
AU8717075A (en) 1977-06-09
US4051252A (en) 1977-09-27
AT343653B (de) 1978-06-12
SE7513990L (sv) 1976-06-14
DD125484A5 (enExample) 1977-04-20
NO754024L (enExample) 1976-06-15
IE42208L (en) 1976-06-13
NO145382C (no) 1982-03-10
DK137082C (da) 1978-06-19
DE2458965B2 (de) 1979-02-22

Similar Documents

Publication Publication Date Title
ZA757777B (en) 3-amino-indazolecarboxylic acid derivatives,process for their preparation and their use as medicaments
EG11718A (en) Triazolyl-alkanones and triazolyl-alkanols,process for their preparation and their use as fungicides
KE3022A (en) Azolyl-(1)-methanes and their salts,process for their preparation and their use as medicaments
IE41091B1 (en) Benzamides, processes for their preparation and their use as medicaments
EG11983A (en) Substituted phenylguanides,a process for their preparation and their use as medicaments
IL47360A (en) -amino- and -formyl- -(p-acycloxyphenyl) acetamido-3-cephem-4-carboxylic acid derivatives,their preparation and pharmaceutical compositions containing them
ZA753124B (en) 3-amino-phenylacetic acid derivatives process for their preparation and their use as herbicides
HK7977A (en) Pyrazole derivatives, process for their preparation and their use as medicaments
IL48707A0 (en) Novel phenylacetic acid derivatives,their preparation and pharmaceutical compositions containing them
IL48396A0 (en) New furanhydroxamic acid derivatives,their manufacture and their use as fungicides
EG11586A (en) Cephalosporins,processes for preparation and their use as medicaments
IL48394A0 (en) New benzophenone derivatives,process for preparing them and pharmaceutical compositions
IL47593A (en) 15,15-ethylenedioxy-prostanoic acid derivatives and process for their manufacture
IL46543A0 (en) New phenoxyalkyl-carboxylic acid derivatives,process for the preparation thereof and pharmaceutical compositions containing the same
ZA754558B (en) Substituted phenylisothioureas, a process for their preparation and their use as medicaments
IL47299A (en) 3-thiomethyl-3-cephem-4-carboxylic acid derivatives,their preparation and pharmaceutical compositions containing them
IL47519A (en) 7-sulphinimidoyl(sulphimidoyl)-xanthone-2-carboxylic acid derivatives, their preparation and pharmaceutical compositions containing them
ZA755688B (en) Basically substituted 3-sulfamoylbenzoic acid derivatives and process for their preparation
GR60560B (en) Penicillines,preparation process and use thereof as medicines
IL44027A (en) 7-acylamido-3-alkyl-ceph-3-eme-4-carboxylic acid derivatives,process for preparing them and pharmaceutical compositions containing them
IL46707A0 (en) Phenylbutanol derivatives,process for their preparation and compositions containing them
AU493473B2 (en) 3-amino-indazolecarboxylic acid derivatives, process for their preparation and their use as medicaments
ZA755310B (en) Process for the preparation of 9,11,15-trihydroxy-13, 14-dehydro-prostaglandins and new prost-5-en-13-ynoic acid derivatives
AU489917B2 (en) Cephalosporins, process for their preparation and their use as medicaments
ZA751969B (en) Pyridylalkylamidines process for their preparation and their use as medicaments