CS189731B2 - Method of producing new derivatives of 3-aminoindazolcarboxylic acid - Google Patents
Method of producing new derivatives of 3-aminoindazolcarboxylic acidInfo
- Publication number
- CS189731B2 CS189731B2 CS758165A CS816575A CS189731B2 CS 189731 B2 CS189731 B2 CS 189731B2 CS 758165 A CS758165 A CS 758165A CS 816575 A CS816575 A CS 816575A CS 189731 B2 CS189731 B2 CS 189731B2
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- aminoindazolcarboxylic
- acid
- producing new
- new derivatives
- derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
- C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE2458965A DE2458965C3 (de) | 1974-12-13 | 1974-12-13 | 3-Amino-indazol-N-carbonsäure-Derivate, Verfahren zu ihrer Herstellung sowie sie enthaltende Arzneimittel |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CS189731B2 true CS189731B2 (en) | 1979-04-30 |
Family
ID=5933305
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CS758165A CS189731B2 (en) | 1974-12-13 | 1975-12-02 | Method of producing new derivatives of 3-aminoindazolcarboxylic acid |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US4051252A (enExample) |
| JP (1) | JPS5182266A (enExample) |
| AT (1) | AT343653B (enExample) |
| BE (1) | BE836528A (enExample) |
| CA (1) | CA1059523A (enExample) |
| CH (1) | CH622250A5 (enExample) |
| CS (1) | CS189731B2 (enExample) |
| DD (1) | DD125484A5 (enExample) |
| DE (1) | DE2458965C3 (enExample) |
| DK (1) | DK137082C (enExample) |
| ES (1) | ES443429A1 (enExample) |
| FI (1) | FI753493A7 (enExample) |
| FR (1) | FR2293928A1 (enExample) |
| GB (1) | GB1490306A (enExample) |
| HK (1) | HK52580A (enExample) |
| HU (1) | HU173557B (enExample) |
| IE (1) | IE42208B1 (enExample) |
| IL (1) | IL48642A (enExample) |
| KE (1) | KE3078A (enExample) |
| LU (1) | LU73993A1 (enExample) |
| NL (1) | NL7514521A (enExample) |
| NO (1) | NO145382C (enExample) |
| PL (1) | PL99858B1 (enExample) |
| SE (1) | SE419645B (enExample) |
| SU (1) | SU604487A3 (enExample) |
| YU (1) | YU315275A (enExample) |
| ZA (1) | ZA757777B (enExample) |
Families Citing this family (39)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4431657A (en) * | 1982-05-24 | 1984-02-14 | Ayerst, Mckenna & Harrison Inc. | Analgesic compositions consisting of 2H-benzothieno[3,2-c]pyrazol-3-amine derivatives |
| KR20010086657A (ko) * | 2000-03-02 | 2001-09-15 | 성재갑 | 아미노인다졸 유도체 및 이를 함유하는 싸이클린 의존키나아제 저해제 조성물 |
| CN1926132B (zh) * | 2000-09-15 | 2010-12-29 | 沃泰克斯药物股份有限公司 | 可用作蛋白激酶抑制剂的吡唑化合物 |
| US6660731B2 (en) | 2000-09-15 | 2003-12-09 | Vertex Pharmaceuticals Incorporated | Pyrazole compounds useful as protein kinase inhibitors |
| US7473691B2 (en) * | 2000-09-15 | 2009-01-06 | Vertex Pharmaceuticals Incorporated | Pyrazole compounds useful as protein kinase inhibitors |
| EP1698627A1 (en) * | 2000-09-15 | 2006-09-06 | Vertex Pharmaceuticals Incorporated | Pyrazole compounds useful as protein kinase inhibitors |
| DK1318997T3 (da) * | 2000-09-15 | 2006-09-25 | Vertex Pharma | Pyrazolforbindelser der er nyttige som proteinkinase-inhibitorer |
| HUP0400639A3 (en) | 2000-12-21 | 2010-03-29 | Vertex Pharma | Pyrazole compounds useful as protein kinase inhibitors and pharmaceutical compositions containing them |
| KR100406634B1 (ko) * | 2001-03-12 | 2003-11-20 | 주식회사 엘지생명과학 | 3,5-디아미노인다졸 유도체, 그의 제조방법 및 사이클린의존성 키나아제 저해제로서의 그의 용도 |
| ES2357502T3 (es) | 2001-09-26 | 2011-04-27 | Pfizer Italia S.R.L. | Derivados de aminoindazol activos como inhibidores de quinasa, procedimiento para su preparación y composiciones farmaceuticas que los contienen. |
| KR20040084896A (ko) * | 2002-02-06 | 2004-10-06 | 버텍스 파마슈티칼스 인코포레이티드 | Gsk-3의 억제제로서 유용한 헤테로아릴 화합물 |
| FR2836915B1 (fr) * | 2002-03-11 | 2008-01-11 | Aventis Pharma Sa | Derives d'aminoindazoles, procede de preparation et intermediaires de ce procede a titre de medicaments et compositions pharmaceutiques les renfermant |
| ATE468336T1 (de) | 2002-03-15 | 2010-06-15 | Vertex Pharma | Azolylaminoazine als proteinkinasehemmer |
| EP1506176B1 (en) | 2002-05-17 | 2013-04-24 | Pfizer Italia S.r.l. | Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them |
| MY141867A (en) | 2002-06-20 | 2010-07-16 | Vertex Pharma | Substituted pyrimidines useful as protein kinase inhibitors |
| DE60308387T2 (de) | 2002-08-02 | 2007-09-20 | Vertex Pharmaceuticals Inc., Cambridge | Pyrazolenthaltende zusammensetzungen und ihre verwendung als gsk-3 inhibitoren |
| JP2006512313A (ja) * | 2002-10-31 | 2006-04-13 | アムジェン インコーポレイテッド | 抗炎症剤 |
| WO2004072029A2 (en) | 2003-02-06 | 2004-08-26 | Vertex Pharmaceuticals Incorporated | Pyrazolopyridazines useful as inhibitors of protein kinases |
| JP2007513184A (ja) * | 2003-12-04 | 2007-05-24 | バーテックス ファーマシューティカルズ インコーポレイテッド | プロテインキナーゼのインヒビターとして有用なキノキサリン |
| DE102004005172A1 (de) | 2004-02-02 | 2005-08-18 | Aventis Pharma Deutschland Gmbh | Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase |
| AU2006279376B2 (en) | 2005-08-18 | 2011-04-14 | Vertex Pharmaceuticals Incoporated | Pyrazine kinase inhibitors |
| TW200734327A (en) | 2005-11-03 | 2007-09-16 | Vertex Pharma | Aminopyrimidines useful as kinase inhibitors |
| JP2009533474A (ja) * | 2006-04-14 | 2009-09-17 | アボット・ラボラトリーズ | バニロイドサブタイプ1(vr1)受容体を阻害するインダゾリルウレアの製造方法 |
| WO2008057940A1 (en) | 2006-11-02 | 2008-05-15 | Vertex Pharmaceuticals Incorporated | Aminopyridines and aminopyrimidines useful as inhibitors of protein kinases |
| WO2008077086A1 (en) | 2006-12-19 | 2008-06-26 | Vertex Pharmaceuticals Incorporated | Aminopyrimidines useful as inhibitors of protein kinases |
| EP2137183B1 (en) | 2007-03-09 | 2011-09-28 | Vertex Pharmaceuticals Incorporated | Aminopyrimidines useful as inhibitors of protein kinases |
| WO2008112642A1 (en) | 2007-03-09 | 2008-09-18 | Vertex Pharmaceuticals Incorporated | Aminopyrimidines useful as inhibitors of protein kinases |
| EP2134709A1 (en) | 2007-03-09 | 2009-12-23 | Vertex Pharmaceuticals, Inc. | Aminopyridines useful as inhibitors of protein kinases |
| JP2010523700A (ja) | 2007-04-13 | 2010-07-15 | バーテックス ファーマシューティカルズ インコーポレイテッド | キナーゼインヒビターとして有用なアミノピリミジン |
| CN101679378A (zh) | 2007-05-02 | 2010-03-24 | 沃泰克斯药物股份有限公司 | 用作激酶抑制剂的噻唑和吡唑 |
| CN101801959A (zh) | 2007-05-02 | 2010-08-11 | 沃泰克斯药物股份有限公司 | 可用作激酶抑制剂的氨基嘧啶类化合物 |
| AU2008247595A1 (en) * | 2007-05-02 | 2008-11-13 | Vertex Pharmaceuticals Incorporated | Aminopyrimidines useful as kinase inhibitors |
| AU2008257044A1 (en) * | 2007-05-24 | 2008-12-04 | Vertex Pharmaceuticals Incorporated | Thiazoles and pyrazoles useful as kinase inhibitors |
| AR067762A1 (es) | 2007-07-31 | 2009-10-21 | Vertex Pharma | Proceso para preparar 5-fluoro-1h-pirazolo (3,4-b) piridin-3-amina y derivados de la misma |
| AU2009288200A1 (en) * | 2008-09-03 | 2010-03-11 | Vertex Pharmaceuticals Incorporated | Co-crystals and pharmaceutical formulations comprising the same |
| DE102009004245A1 (de) | 2009-01-09 | 2010-07-15 | Bayer Schering Pharma Aktiengesellschaft | Neue anellierte, Heteroatom-verbrückte Pyrazol- und Imidazol-Derivate und ihre Verwendung |
| KR102137714B1 (ko) | 2012-07-24 | 2020-07-27 | 바이알 - 포르텔라 앤드 씨에이 에스에이 | 요소 화합물 및 효소 억제제로서 이들의 용도 |
| EP2882712A2 (en) * | 2012-07-27 | 2015-06-17 | BIAL - Portela & Cª S.A. | Process for the synthesis of substituted urea compounds |
| AU2014293731B2 (en) | 2013-07-24 | 2018-03-08 | Bial - Portela & Ca, S.A. | Imidazolecarboxamides and their use as FAAH inhibitors |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3133081A (en) * | 1964-05-12 | J-aminoindazole derivatives | ||
| CH397698A (de) * | 1961-09-08 | 1965-08-31 | Siegfried Ag | Verfahren zur Herstellung neuer 1-Carbamyl-indazole |
| US3277100A (en) * | 1963-05-31 | 1966-10-04 | Du Pont | Novel substituted pyrazoles |
| NL6707299A (enExample) * | 1966-07-16 | 1968-01-17 | ||
| DE1770649A1 (de) * | 1968-06-15 | 1971-11-11 | Bayer Ag | Substituierte 3-Amino-indazole |
-
1974
- 1974-12-13 DE DE2458965A patent/DE2458965C3/de not_active Expired
-
1975
- 1975-10-28 GB GB44299/75A patent/GB1490306A/en not_active Expired
- 1975-11-24 US US05/634,914 patent/US4051252A/en not_active Expired - Lifetime
- 1975-11-27 CA CA240,662A patent/CA1059523A/en not_active Expired
- 1975-11-28 NO NO754024A patent/NO145382C/no unknown
- 1975-12-02 CS CS758165A patent/CS189731B2/cs unknown
- 1975-12-08 SU SU752195302A patent/SU604487A3/ru active
- 1975-12-09 CH CH1599575A patent/CH622250A5/de not_active IP Right Cessation
- 1975-12-10 IL IL48642A patent/IL48642A/xx unknown
- 1975-12-11 LU LU73993A patent/LU73993A1/xx unknown
- 1975-12-11 DD DD190061A patent/DD125484A5/xx unknown
- 1975-12-11 PL PL1975185475A patent/PL99858B1/pl unknown
- 1975-12-11 HU HU75BA3349A patent/HU173557B/hu unknown
- 1975-12-11 BE BE162651A patent/BE836528A/xx unknown
- 1975-12-11 SE SE7513990A patent/SE419645B/xx unknown
- 1975-12-11 AT AT939775A patent/AT343653B/de not_active IP Right Cessation
- 1975-12-11 JP JP50146940A patent/JPS5182266A/ja active Pending
- 1975-12-11 FI FI753493A patent/FI753493A7/fi not_active Application Discontinuation
- 1975-12-12 YU YU03152/75A patent/YU315275A/xx unknown
- 1975-12-12 ZA ZA757777A patent/ZA757777B/xx unknown
- 1975-12-12 NL NL7514521A patent/NL7514521A/xx not_active Application Discontinuation
- 1975-12-12 DK DK567275A patent/DK137082C/da active
- 1975-12-12 IE IE2714/75A patent/IE42208B1/en unknown
- 1975-12-12 FR FR7538124A patent/FR2293928A1/fr active Granted
- 1975-12-12 ES ES443429A patent/ES443429A1/es not_active Expired
-
1980
- 1980-08-29 KE KE3078A patent/KE3078A/xx unknown
- 1980-09-18 HK HK525/80A patent/HK52580A/xx unknown
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CS189731B2 (en) | Method of producing new derivatives of 3-aminoindazolcarboxylic acid | |
| JPS53101385A (en) | Method of producing phenyllpyrimidine | |
| CS188985B2 (en) | Method of producing aryl-1-azolylmethanes | |
| CS190478B2 (en) | Method of producing novel biphenylyl derivatives | |
| CS194749B2 (en) | Method of producing novel derivatives of 3-sulphonyl-ox!-crotonic acid | |
| CS189709B2 (en) | Method of producing 6-d-/-/-alpha-amino-alpha-/p-acetoxyphenylacetamido/penicillanic acid | |
| CS188235B2 (en) | Method of producing new derivatives ryfamicine | |
| CS191264B2 (en) | Method of producing new pyridobenzodiazepinones | |
| CS183850B2 (en) | Method of producing 5-fluor-2-methyl-1-/p-methyl-sulphinylbenzyliden/-3-indenylacetic acid | |
| CS188938B2 (en) | Method of producing xanthene-9-spiro-4-piperidines | |
| SU677666A3 (en) | Method of producing 7l-or extradiols | |
| YU118575A (en) | Process for obtaining new derivatives of 13-thiaprostanoic acid | |
| CS190489B2 (en) | Method of producing novel derivatives of prostanoic acid | |
| HU170859B (hu) | Sposob poluchenija novykh proizvodnykh 6-skobka-al'fa-ureido-fenilacetilamido-skobka zakryta-penam-3-karbonovojj kisloty | |
| CS189635B2 (en) | Method of producing bromderivatives of 4-imido-thioazetidin-2-one | |
| CS192518B2 (en) | Method of producing derivatives of 3-cinnolincarboxylic acid | |
| CS182298B2 (en) | Method of producing substituted benzendisulphon-amides | |
| CS187333B2 (en) | Method of producing derivatives of prostanoic acid | |
| HU171053B (hu) | Sposob poluchenija novykh proizvodnykh 7-skobka-2-ureido-acetamido-skobka zakryta-3-geterociklicheskijj-tiometil-cef-3-em-4-karbonovojj kisloty | |
| CS189753B2 (en) | Method of producing derivatives of prostanic acid | |
| HU175345B (hu) | Sposob poluchenija novykh proizvodnykh 15-gidroksi-16s- i -16r-alkil-prost-5-en-13-in-karbonovykh kislot | |
| CS188945B2 (en) | Method of producing 1-aryluracils | |
| CS185675B2 (en) | Method of producing 7-amino-delta up3-cephem derivatives | |
| CS181278B2 (en) | Method of producing cephalosporane acid derivatives | |
| BG25086A3 (en) | A method of obtaining derivatives of thiazolidinon-acetic acid |