JPH08500110A - ブプロピオン含有持続放出型錠剤 - Google Patents
ブプロピオン含有持続放出型錠剤Info
- Publication number
- JPH08500110A JPH08500110A JP6506019A JP50601994A JPH08500110A JP H08500110 A JPH08500110 A JP H08500110A JP 6506019 A JP6506019 A JP 6506019A JP 50601994 A JP50601994 A JP 50601994A JP H08500110 A JPH08500110 A JP H08500110A
- Authority
- JP
- Japan
- Prior art keywords
- hydrochloride
- bupropion hydrochloride
- release tablet
- bupropion
- tablet according
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/16—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
- A61K47/18—Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
- A61K47/183—Amino acids, e.g. glycine, EDTA or aspartame
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/20—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing sulfur, e.g. dimethyl sulfoxide [DMSO], docusate, sodium lauryl sulfate or aminosulfonic acids
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Neurosurgery (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Psychiatry (AREA)
- Pain & Pain Management (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- General Preparation And Processing Of Foods (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB929217295A GB9217295D0 (en) | 1992-08-14 | 1992-08-14 | Controlled released tablets |
| GB9217295.6 | 1992-08-14 | ||
| PCT/GB1993/001722 WO1994004138A1 (en) | 1992-08-14 | 1993-08-13 | Sustained release tablets containing bupropion |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| JPH08500110A true JPH08500110A (ja) | 1996-01-09 |
Family
ID=10720358
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP6506019A Pending JPH08500110A (ja) | 1992-08-14 | 1993-08-13 | ブプロピオン含有持続放出型錠剤 |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US5427798A (enExample) |
| EP (1) | EP0656775B1 (enExample) |
| JP (1) | JPH08500110A (enExample) |
| KR (1) | KR100294154B1 (enExample) |
| AT (1) | ATE161422T1 (enExample) |
| AU (1) | AU677595B2 (enExample) |
| CA (1) | CA2142320C (enExample) |
| CY (1) | CY2143B1 (enExample) |
| DE (1) | DE69316015T2 (enExample) |
| ES (1) | ES2111168T3 (enExample) |
| GB (1) | GB9217295D0 (enExample) |
| GR (1) | GR3025794T3 (enExample) |
| HK (1) | HK1004323A1 (enExample) |
| IL (1) | IL106693A (enExample) |
| LU (1) | LU90656I2 (enExample) |
| MX (1) | MX9304967A (enExample) |
| NZ (1) | NZ254947A (enExample) |
| SG (1) | SG43911A1 (enExample) |
| TW (1) | TW260607B (enExample) |
| WO (1) | WO1994004138A1 (enExample) |
| ZA (1) | ZA935942B (enExample) |
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2001517625A (ja) * | 1997-09-25 | 2001-10-09 | バイエル・アクチエンゲゼルシヤフト | 活性成分放出制御薬物製剤 |
| JP2002537319A (ja) * | 1999-02-26 | 2002-11-05 | アンドルックス ファーマスーティカルズ インコーポレーテッド | 放出制御されたブプロピオン製剤 |
| JP2023516404A (ja) * | 2020-03-05 | 2023-04-19 | アッヴィ・インコーポレイテッド | エラゴリクスの投与方法 |
Families Citing this family (225)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5541231A (en) * | 1993-07-30 | 1996-07-30 | Glaxo Wellcome Inc. | Stabilized Pharmaceutical |
| GB9315856D0 (en) * | 1993-07-30 | 1993-09-15 | Wellcome Found | Stabilized pharmaceutical |
| US5616344A (en) * | 1994-06-14 | 1997-04-01 | Fuisz Technologies Ltd. | Apparatus and process for strengthening low density compression dosage units and product therefrom |
| US6221917B1 (en) | 1997-12-30 | 2001-04-24 | American Home Products Corporation | Pharmaceutical composition containing bupropion hydrochloride and a stabilizer |
| US5968553A (en) * | 1997-12-30 | 1999-10-19 | American Home Products Corporation | Pharmaceutical composition containing bupropion hydrochloride and an inorganic acid stabilizer |
| US7098206B2 (en) * | 1998-01-21 | 2006-08-29 | Smithkline Beecham Corporation | Pharmaceutically active morpholinol |
| US6998400B2 (en) * | 1998-01-22 | 2006-02-14 | Smithkline Beecham Corporation | Pharmaceutically active morpholinol |
| AU2349999A (en) | 1998-01-29 | 1999-08-16 | Sepracor, Inc. | Pharmacological uses of pure (+) -bupropion |
| CA2318960A1 (en) * | 1998-01-29 | 1999-08-05 | Sepracor Inc. | Pharmaceutical uses of optically pure (+)-bupropion |
| JP2002501888A (ja) * | 1998-01-29 | 2002-01-22 | セプラコア インコーポレーテッド | 光学的に純粋な(−)−ビュープロピオンを用いて禁煙を支援するためのまたは疼痛や他の障害を治療するための方法および組成物 |
| JP2002501892A (ja) * | 1998-01-29 | 2002-01-22 | セプラコア インコーポレーテッド | 光学的に純粋な(−)−ビュープロピオンの薬学的使用 |
| US6150420A (en) * | 1998-06-01 | 2000-11-21 | Theramax, Inc. | Method for enhanced brain delivery of bupropion |
| US6153223A (en) * | 1998-06-05 | 2000-11-28 | Watson Pharmaceuticals, Inc. | Stabilized pharmaceutical compositions |
| US6096341A (en) * | 1998-10-30 | 2000-08-01 | Pharma Pass Llc | Delayed release tablet of bupropion hydrochloride |
| US6033686A (en) * | 1998-10-30 | 2000-03-07 | Pharma Pass Llc | Controlled release tablet of bupropion hydrochloride |
| US6238697B1 (en) * | 1998-12-21 | 2001-05-29 | Pharmalogix, Inc. | Methods and formulations for making bupropion hydrochloride tablets using direct compression |
| US6855820B2 (en) * | 1999-01-20 | 2005-02-15 | Smithkline Beecham Corporation | Pharmaceutically active morpholinol |
| US6734213B2 (en) | 1999-01-20 | 2004-05-11 | Smithkline Beecham Corporation | Pharmaceutically active morpholinol |
| US8545880B2 (en) * | 1999-02-26 | 2013-10-01 | Andrx Pharmaceuticals, Llc | Controlled release oral dosage form |
| US6589553B2 (en) * | 2001-02-08 | 2003-07-08 | Andrx Pharmaceuticals, Inc. | Controlled release oral dosage form |
| US6342496B1 (en) * | 1999-03-01 | 2002-01-29 | Sepracor Inc. | Bupropion metabolites and methods of use |
| US6337328B1 (en) * | 1999-03-01 | 2002-01-08 | Sepracor, Inc. | Bupropion metabolites and methods of use |
| USD430285S (en) * | 1999-04-16 | 2000-08-29 | Merck & Co., Inc. | Tablet |
| US6280763B1 (en) | 1999-05-10 | 2001-08-28 | Pierce Management, Llc | Apparatus and method for transdermal delivery of bupropion |
| AU781718B2 (en) * | 1999-11-02 | 2005-06-09 | Depomed, Inc. | Pharmacological inducement of the fed mode for enhanced drug administration to the stomach |
| US6306436B1 (en) | 2000-04-28 | 2001-10-23 | Teva Pharmaceuticals Usa, Inc. | Stabilized, acid-free formulation for sustained release of bupropion hydrochloride |
| CA2685214C (en) * | 2001-02-08 | 2013-01-22 | Andrx Pharmaceuticals, Inc. | Improved controlled release oral dosage form |
| ITMI20011457A1 (it) * | 2001-07-09 | 2003-01-09 | Valpharma Sa | Composizione farmaceutica a rilascio modificato contenente bupropionehc1 come sostanza attiva |
| US20030044462A1 (en) * | 2001-08-20 | 2003-03-06 | Kali Laboratories, Inc. | Sustained release tablets containing bupropion hydrochloride |
| EP2316469A1 (en) | 2002-02-22 | 2011-05-04 | Shire LLC | Delivery system and methods for protecting and administering dextroamphetamine |
| US20050215552A1 (en) * | 2002-05-17 | 2005-09-29 | Gadde Kishore M | Method for treating obesity |
| CA2483464C (en) * | 2002-05-17 | 2011-12-20 | Duke University | Method for treating obesity |
| US7776314B2 (en) | 2002-06-17 | 2010-08-17 | Grunenthal Gmbh | Abuse-proofed dosage system |
| AU2003284942A1 (en) * | 2002-10-30 | 2004-06-07 | Pharmacia Corporation | Oral extended release tablets and methods of making and using the same |
| US20040096497A1 (en) * | 2002-11-19 | 2004-05-20 | Ponder Garratt W. | Methods of providing controlled-release pharmaceutical compositions and controlled-release pharmaceutical compositions |
| US6893660B2 (en) * | 2002-11-21 | 2005-05-17 | Andrx Pharmaceuticals, Inc. | Stable pharmaceutical compositions without a stabilizer |
| ES2639579T3 (es) | 2003-04-29 | 2017-10-27 | Orexigen Therapeutics, Inc. | Composiciones para afectar la pérdida de peso que comprende un antagonista opioide y bupropión |
| DE102004032051A1 (de) * | 2004-07-01 | 2006-01-19 | Grünenthal GmbH | Verfahren zur Herstellung einer gegen Missbrauch gesicherten, festen Darreichungsform |
| DE10336400A1 (de) | 2003-08-06 | 2005-03-24 | Grünenthal GmbH | Gegen Missbrauch gesicherte Darreichungsform |
| US20070048228A1 (en) * | 2003-08-06 | 2007-03-01 | Elisabeth Arkenau-Maric | Abuse-proofed dosage form |
| DE102005005446A1 (de) | 2005-02-04 | 2006-08-10 | Grünenthal GmbH | Bruchfeste Darreichungsformen mit retardierter Freisetzung |
| DE10361596A1 (de) | 2003-12-24 | 2005-09-29 | Grünenthal GmbH | Verfahren zur Herstellung einer gegen Missbrauch gesicherten Darreichungsform |
| US8075872B2 (en) | 2003-08-06 | 2011-12-13 | Gruenenthal Gmbh | Abuse-proofed dosage form |
| EP1575565B1 (en) * | 2003-08-08 | 2010-01-06 | Biovail Laboratories International Srl | Modified-release tablet of bupropion hydrochloride |
| US7713959B2 (en) * | 2004-01-13 | 2010-05-11 | Duke University | Compositions of an anticonvulsant and mirtazapine to prevent weight gain |
| US20060160750A1 (en) * | 2004-01-13 | 2006-07-20 | Krishnan K R R | Compositions of an anticonvulsant and an antipsychotic drug and methods of using the same for affecting weight loss |
| KR20060128995A (ko) | 2004-01-13 | 2006-12-14 | 듀크 유니버시티 | 체중감량에 영향을 미치는 항경련제와 항정신병 약물의조성물 |
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| US8586085B2 (en) | 2004-11-08 | 2013-11-19 | Biokey, Inc. | Methods and formulations for making pharmaceutical compositions containing bupropion |
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- 1993-08-13 EP EP93918020A patent/EP0656775B1/en not_active Expired - Lifetime
- 1993-08-13 SG SG1996005086A patent/SG43911A1/en unknown
- 1993-08-13 AT AT93918020T patent/ATE161422T1/de active
- 1993-08-13 NZ NZ254947A patent/NZ254947A/en not_active IP Right Cessation
- 1993-08-13 KR KR1019950700497A patent/KR100294154B1/ko not_active Expired - Lifetime
- 1993-08-16 MX MX9304967A patent/MX9304967A/es unknown
-
1997
- 1997-12-30 GR GR970403389T patent/GR3025794T3/el unknown
-
1999
- 1999-11-29 CY CY9900040A patent/CY2143B1/xx unknown
-
2000
- 2000-10-18 LU LU90656C patent/LU90656I2/fr unknown
Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2001517625A (ja) * | 1997-09-25 | 2001-10-09 | バイエル・アクチエンゲゼルシヤフト | 活性成分放出制御薬物製剤 |
| JP2002537319A (ja) * | 1999-02-26 | 2002-11-05 | アンドルックス ファーマスーティカルズ インコーポレーテッド | 放出制御されたブプロピオン製剤 |
| JP2023516404A (ja) * | 2020-03-05 | 2023-04-19 | アッヴィ・インコーポレイテッド | エラゴリクスの投与方法 |
Also Published As
| Publication number | Publication date |
|---|---|
| WO1994004138A1 (en) | 1994-03-03 |
| KR100294154B1 (ko) | 2001-09-17 |
| ES2111168T3 (es) | 1998-03-01 |
| EP0656775A1 (en) | 1995-06-14 |
| CA2142320A1 (en) | 1994-03-03 |
| MX9304967A (es) | 1994-05-31 |
| KR950702827A (ko) | 1995-08-23 |
| ZA935942B (en) | 1995-02-13 |
| AU4725893A (en) | 1994-03-15 |
| GR3025794T3 (en) | 1998-03-31 |
| US5427798A (en) | 1995-06-27 |
| DE69316015D1 (de) | 1998-02-05 |
| LU90656I2 (fr) | 2001-01-15 |
| IL106693A0 (en) | 1993-12-08 |
| GB9217295D0 (en) | 1992-09-30 |
| AU677595B2 (en) | 1997-05-01 |
| CA2142320C (en) | 2001-10-09 |
| DE69316015T2 (de) | 1998-04-16 |
| EP0656775B1 (en) | 1997-12-29 |
| HK1004323A1 (en) | 1998-11-20 |
| TW260607B (enExample) | 1995-10-21 |
| CY2143B1 (en) | 2002-06-21 |
| IL106693A (en) | 1997-06-10 |
| SG43911A1 (en) | 1997-11-14 |
| ATE161422T1 (de) | 1998-01-15 |
| NZ254947A (en) | 1996-04-26 |
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