JPH03176460A - グルタル酸誘導体およびその製法 - Google Patents

グルタル酸誘導体およびその製法

Info

Publication number
JPH03176460A
JPH03176460A JP2311242A JP31124290A JPH03176460A JP H03176460 A JPH03176460 A JP H03176460A JP 2311242 A JP2311242 A JP 2311242A JP 31124290 A JP31124290 A JP 31124290A JP H03176460 A JPH03176460 A JP H03176460A
Authority
JP
Japan
Prior art keywords
formula
salt
compound
optically pure
substantially optically
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2311242A
Other languages
English (en)
Japanese (ja)
Other versions
JPH0585538B2 (https=
Inventor
Ian T Barnish
イアン・トンプソン・バーニッシュ
Keith James
キース・ジェームズ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Inc
Original Assignee
Pfizer Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Inc filed Critical Pfizer Inc
Publication of JPH03176460A publication Critical patent/JPH03176460A/ja
Publication of JPH0585538B2 publication Critical patent/JPH0585538B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C227/30—Preparation of optical isomers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
    • C07C229/46—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino or carboxyl groups bound to carbon atoms of rings other than six-membered aromatic rings of the same carbon skeleton
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/06—Systems containing only non-condensed rings with a five-membered ring
    • C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicinal Preparation (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Lubricants (AREA)
  • Peptides Or Proteins (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
JP2311242A 1989-11-16 1990-11-16 グルタル酸誘導体およびその製法 Granted JPH03176460A (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB898925933A GB8925933D0 (en) 1989-11-16 1989-11-16 Glutaric acid derivatives and preparation thereof
GB8925933.7 1989-11-16

Publications (2)

Publication Number Publication Date
JPH03176460A true JPH03176460A (ja) 1991-07-31
JPH0585538B2 JPH0585538B2 (https=) 1993-12-07

Family

ID=10666416

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2311242A Granted JPH03176460A (ja) 1989-11-16 1990-11-16 グルタル酸誘導体およびその製法

Country Status (29)

Country Link
US (1) US5087732A (https=)
EP (1) EP0432898B1 (https=)
JP (1) JPH03176460A (https=)
KR (1) KR940005958B1 (https=)
CN (2) CN1028361C (https=)
AT (1) ATE104270T1 (https=)
AU (1) AU623814B2 (https=)
BR (1) BR9005746A (https=)
CA (1) CA2029785C (https=)
CZ (1) CZ284374B6 (https=)
DE (1) DE69008130T2 (https=)
DK (1) DK0432898T3 (https=)
EG (1) EG19319A (https=)
ES (1) ES2062410T3 (https=)
FI (1) FI107148B (https=)
GB (1) GB8925933D0 (https=)
HU (1) HU207711B (https=)
IE (1) IE63684B1 (https=)
IL (1) IL96299A (https=)
MX (1) MX23335A (https=)
MY (1) MY104782A (https=)
NO (1) NO179072C (https=)
NZ (1) NZ236080A (https=)
PH (1) PH27369A (https=)
PL (2) PL164610B1 (https=)
PT (1) PT95889B (https=)
RU (1) RU2002734C1 (https=)
SK (1) SK282272B6 (https=)
ZA (1) ZA909161B (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5208236A (en) * 1992-09-23 1993-05-04 Schering Corporation N-(acylaminomethyl)glutaryl amino acids and use
FR2890069B1 (fr) * 2005-08-31 2011-03-04 Senn Chemicals Internat Intermediaires de synthese pour la preparation de b2-aminoacides et leurs procedes de preparation
PT2380871E (pt) * 2010-04-15 2013-03-07 Indena Spa Um processo para a preparação de derivados de isoserina

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2460891C2 (de) * 1974-12-21 1982-09-23 Gödecke AG, 1000 Berlin 1-Aminomethyl-1-cycloalkanessigsäuren und deren Ester, Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel
KR880007441A (ko) * 1986-12-11 1988-08-27 알렌 제이.스피겔 스피로-치환된 글루타르아미드 이뇨제
GB8820844D0 (en) * 1988-09-05 1988-10-05 Pfizer Ltd Therapeutic agents

Also Published As

Publication number Publication date
CN1107135A (zh) 1995-08-23
IL96299A0 (en) 1991-08-16
ES2062410T3 (es) 1994-12-16
DE69008130D1 (de) 1994-05-19
NO904961L (no) 1991-05-21
JPH0585538B2 (https=) 1993-12-07
US5087732A (en) 1992-02-11
CZ568590A3 (cs) 1998-08-12
DE69008130T2 (de) 1994-07-21
FI107148B (fi) 2001-06-15
NO904961D0 (no) 1990-11-15
BR9005746A (pt) 1991-07-30
CN1051991C (zh) 2000-05-03
HU907179D0 (en) 1991-05-28
KR940005958B1 (ko) 1994-06-25
CN1028361C (zh) 1995-05-10
KR910009635A (ko) 1991-06-28
IL96299A (en) 1997-11-20
HU207711B (en) 1993-05-28
HUT56536A (en) 1991-09-30
CA2029785A1 (en) 1991-05-17
CZ284374B6 (cs) 1998-11-11
CA2029785C (en) 1995-03-28
NO179072B (no) 1996-04-22
PL287759A1 (en) 1991-11-04
ZA909161B (en) 1992-06-24
PL164543B1 (pl) 1994-08-31
GB8925933D0 (en) 1990-01-04
ATE104270T1 (de) 1994-04-15
SK568590A3 (en) 2001-12-03
IE63684B1 (en) 1995-05-31
NZ236080A (en) 1992-04-28
MX23335A (es) 1993-09-01
FI905664L (fi) 1991-05-17
AU6668490A (en) 1991-05-23
RU2002734C1 (ru) 1993-11-15
FI905664A0 (fi) 1990-11-15
PT95889A (pt) 1991-09-13
EP0432898B1 (en) 1994-04-13
PH27369A (en) 1993-06-21
PL164610B1 (pl) 1994-08-31
EG19319A (en) 1994-09-29
NO179072C (no) 1996-07-31
EP0432898A3 (en) 1991-09-11
DK0432898T3 (da) 1994-05-16
IE904121A1 (en) 1991-05-22
CN1051725A (zh) 1991-05-29
MY104782A (en) 1994-05-31
PT95889B (pt) 1997-06-30
AU623814B2 (en) 1992-05-21
EP0432898A2 (en) 1991-06-19
SK282272B6 (sk) 2001-12-03

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Legal Events

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LAPS Cancellation because of no payment of annual fees