JP6768693B2 - グルタミナーゼ阻害剤を投与する方法 - Google Patents

グルタミナーゼ阻害剤を投与する方法 Download PDF

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JP6768693B2
JP6768693B2 JP2017550897A JP2017550897A JP6768693B2 JP 6768693 B2 JP6768693 B2 JP 6768693B2 JP 2017550897 A JP2017550897 A JP 2017550897A JP 2017550897 A JP2017550897 A JP 2017550897A JP 6768693 B2 JP6768693 B2 JP 6768693B2
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cancer
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JP2018510175A (ja
JP2018510175A5 (enExample
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マシュー アイ． グロス，
マシュー アイ． グロス，
マーク ケー． ベネット，
マーク ケー． ベネット，
クリストファー モリニュー，
クリストファー モリニュー，
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キャリセラ バイオサイエンシーズ， インコーポレイテッド
キャリセラ バイオサイエンシーズ， インコーポレイテッド
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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JP2017550897A 2015-03-30 2016-03-30 グルタミナーゼ阻害剤を投与する方法 Expired - Fee Related JP6768693B2 (ja)

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US201562139928P 2015-03-30 2015-03-30
US62/139,928 2015-03-30
US201562168112P 2015-05-29 2015-05-29
US62/168,112 2015-05-29
PCT/US2016/024998 WO2016160980A1 (en) 2015-03-30 2016-03-30 Methods of administering glutaminase inhibitors

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JP2018510175A JP2018510175A (ja) 2018-04-12
JP2018510175A5 JP2018510175A5 (enExample) 2019-05-09
JP6768693B2 true JP6768693B2 (ja) 2020-10-14

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US (1) US20160287564A1 (enExample)
EP (1) EP3277276B1 (enExample)
JP (1) JP6768693B2 (enExample)
KR (1) KR20170131650A (enExample)
CN (1) CN107921031A (enExample)
AU (1) AU2016243631B2 (enExample)
BR (1) BR112017020780A2 (enExample)
CA (1) CA2981499A1 (enExample)
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HK (1) HK1254129A1 (enExample)
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Families Citing this family (16)

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Publication number Priority date Publication date Assignee Title
US8604016B2 (en) 2011-11-21 2013-12-10 Calithera Biosciences Inc. Heterocyclic inhibitors of glutaminase
HUE056078T2 (hu) 2012-11-16 2022-01-28 Calithera Biosciences Inc Heterociklusos glutamináz inhibitorok
HRP20192056T1 (hr) 2014-04-30 2020-02-21 Pfizer Inc. Derivati diheterocikla vezani na cikloalkil
JP6889101B2 (ja) 2014-08-07 2021-06-18 キャリセラ バイオサイエンシーズ， インコーポレイテッド グルタミナーゼ阻害剤の結晶形態
BR112017021312A2 (pt) * 2015-04-06 2018-06-26 Calithera Biosciences Inc tratamento de câncer de pulmão com inibidores de glutaminase
SG11201802830QA (en) 2015-10-05 2018-05-30 Calithera Biosciences Inc Combination therapy with glutaminase inhibitors and immuno-oncology agents
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