HK1254129A1 - 給予谷氨酰胺酶抑制劑的方法 - Google Patents
給予谷氨酰胺酶抑制劑的方法Info
- Publication number
- HK1254129A1 HK1254129A1 HK18113200.9A HK18113200A HK1254129A1 HK 1254129 A1 HK1254129 A1 HK 1254129A1 HK 18113200 A HK18113200 A HK 18113200A HK 1254129 A1 HK1254129 A1 HK 1254129A1
- Authority
- HK
- Hong Kong
- Prior art keywords
- administering
- methods
- glutaminase inhibitors
- glutaminase
- inhibitors
- Prior art date
Links
- 102000009127 Glutaminase Human genes 0.000 title 1
- 108010073324 Glutaminase Proteins 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/433—Thidiazoles
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- A—HUMAN NECESSITIES
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
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- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
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- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
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Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
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- Immunology (AREA)
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- Hematology (AREA)
- Molecular Biology (AREA)
- Communicable Diseases (AREA)
- Diabetes (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Virology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Coloring Foods And Improving Nutritive Qualities (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201562139928P | 2015-03-30 | 2015-03-30 | |
US201562168112P | 2015-05-29 | 2015-05-29 | |
PCT/US2016/024998 WO2016160980A1 (en) | 2015-03-30 | 2016-03-30 | Methods of administering glutaminase inhibitors |
Publications (1)
Publication Number | Publication Date |
---|---|
HK1254129A1 true HK1254129A1 (zh) | 2019-07-12 |
Family
ID=57007550
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HK18113200.9A HK1254129A1 (zh) | 2015-03-30 | 2018-10-16 | 給予谷氨酰胺酶抑制劑的方法 |
Country Status (14)
Country | Link |
---|---|
US (1) | US20160287564A1 (zh) |
EP (1) | EP3277276B1 (zh) |
JP (1) | JP6768693B2 (zh) |
KR (1) | KR20170131650A (zh) |
CN (1) | CN107921031A (zh) |
AU (1) | AU2016243631B2 (zh) |
BR (1) | BR112017020780A2 (zh) |
CA (1) | CA2981499A1 (zh) |
EA (1) | EA037152B1 (zh) |
HK (1) | HK1254129A1 (zh) |
IL (1) | IL254779A0 (zh) |
MX (1) | MX2017012408A (zh) |
SG (1) | SG11201708034SA (zh) |
WO (1) | WO2016160980A1 (zh) |
Families Citing this family (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8604016B2 (en) | 2011-11-21 | 2013-12-10 | Calithera Biosciences Inc. | Heterocyclic inhibitors of glutaminase |
EP2920168B1 (en) | 2012-11-16 | 2021-07-21 | Calithera Biosciences, Inc. | Heterocyclic glutaminase inhibitors |
JP6574203B2 (ja) | 2014-04-30 | 2019-09-11 | ファイザー・インク | シクロアルキル結合ジヘテロ環誘導体 |
EA037738B1 (ru) | 2014-08-07 | 2021-05-17 | Калитера Байосайенсиз, Инк. | Кристаллические формы ингибиторов глутаминазы |
US10441587B2 (en) * | 2015-04-06 | 2019-10-15 | Calithera Biosciences, Inc. | Treatment of lung cancer with inhibitors of glutaminase |
SG11201802830QA (en) | 2015-10-05 | 2018-05-30 | Calithera Biosciences Inc | Combination therapy with glutaminase inhibitors and immuno-oncology agents |
JP2019524852A (ja) | 2016-08-25 | 2019-09-05 | キャリセラ バイオサイエンシーズ, インコーポレイテッド | グルタミナーゼ阻害剤を用いる併用療法 |
AU2017315446A1 (en) | 2016-08-25 | 2019-03-07 | Calithera Biosciences, Inc. | Combination therapy with glutaminase inhibitors |
WO2018102715A1 (en) * | 2016-12-02 | 2018-06-07 | Indiana University Research And Technology Corporation | Compositions and methods for treating and/or reducing corneal dystrophy |
WO2020086440A1 (en) * | 2018-10-22 | 2020-04-30 | Beth Israel Deaconess Medical Center | Immunomodulatory compounds |
CA3169303A1 (en) * | 2020-02-24 | 2021-09-02 | Xiaokun SHEN | Application of poly adp-ribose polymerase inhibitors in corona virus resistance |
CN111643669A (zh) * | 2020-06-30 | 2020-09-11 | 广东省中医院(广州中医药大学第二附属医院、广州中医药大学第二临床医学院、广东省中医药科学院) | 谷氨酰胺酶抑制剂在制备治疗银屑病的药物中的应用 |
CN113633642A (zh) * | 2021-08-26 | 2021-11-12 | 山东第一医科大学附属青岛眼科医院(山东省眼科研究所、青岛眼科医院) | Abt-263在制备抑制角膜移植免疫排斥反应的药物中的应用 |
CN114748482B (zh) * | 2022-04-29 | 2023-09-26 | 广东龙帆生物科技有限公司 | 一种pf-04691502在制备用于抗腺病毒感染的药物中的用途 |
Family Cites Families (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN103030597B (zh) * | 2011-09-30 | 2014-10-01 | 南昌滨西科技有限公司 | 肾脏型谷氨酰胺酶抑制剂及其制备方法和用途 |
US8604016B2 (en) * | 2011-11-21 | 2013-12-10 | Calithera Biosciences Inc. | Heterocyclic inhibitors of glutaminase |
PL2782570T3 (pl) * | 2011-11-21 | 2020-04-30 | Calithera Biosciences Inc. | Heterocykliczne inhibitory glutaminazy |
EP2920168B1 (en) * | 2012-11-16 | 2021-07-21 | Calithera Biosciences, Inc. | Heterocyclic glutaminase inhibitors |
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WO2016004418A1 (en) * | 2014-07-03 | 2016-01-07 | Board Of Regents, University Of Texas System | Glutaminase inhibitor therapy |
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EA037738B1 (ru) * | 2014-08-07 | 2021-05-17 | Калитера Байосайенсиз, Инк. | Кристаллические формы ингибиторов глутаминазы |
WO2016054388A1 (en) * | 2014-10-03 | 2016-04-07 | University Of Pittsburgh - Of The Commonwealth System Of Higher Education | Glutaminase inhibitors |
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-
2016
- 2016-03-30 AU AU2016243631A patent/AU2016243631B2/en not_active Ceased
- 2016-03-30 US US15/085,451 patent/US20160287564A1/en not_active Abandoned
- 2016-03-30 KR KR1020177031129A patent/KR20170131650A/ko not_active Application Discontinuation
- 2016-03-30 MX MX2017012408A patent/MX2017012408A/es unknown
- 2016-03-30 EP EP16774100.8A patent/EP3277276B1/en active Active
- 2016-03-30 SG SG11201708034SA patent/SG11201708034SA/en unknown
- 2016-03-30 CN CN201680031557.9A patent/CN107921031A/zh active Pending
- 2016-03-30 CA CA2981499A patent/CA2981499A1/en not_active Abandoned
- 2016-03-30 BR BR112017020780A patent/BR112017020780A2/pt not_active IP Right Cessation
- 2016-03-30 EA EA201792162A patent/EA037152B1/ru not_active IP Right Cessation
- 2016-03-30 WO PCT/US2016/024998 patent/WO2016160980A1/en active Application Filing
- 2016-03-30 JP JP2017550897A patent/JP6768693B2/ja not_active Expired - Fee Related
-
2017
- 2017-09-28 IL IL254779A patent/IL254779A0/en unknown
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2018
- 2018-10-16 HK HK18113200.9A patent/HK1254129A1/zh unknown
Also Published As
Publication number | Publication date |
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KR20170131650A (ko) | 2017-11-29 |
EA037152B1 (ru) | 2021-02-11 |
EA201792162A1 (ru) | 2018-04-30 |
AU2016243631B2 (en) | 2021-07-29 |
JP2018510175A (ja) | 2018-04-12 |
MX2017012408A (es) | 2018-04-26 |
CA2981499A1 (en) | 2016-10-06 |
BR112017020780A2 (pt) | 2018-06-26 |
EP3277276A4 (en) | 2019-02-06 |
EP3277276B1 (en) | 2020-11-04 |
US20160287564A1 (en) | 2016-10-06 |
CN107921031A (zh) | 2018-04-17 |
IL254779A0 (en) | 2017-12-31 |
AU2016243631A1 (en) | 2017-10-26 |
EP3277276A1 (en) | 2018-02-07 |
SG11201708034SA (en) | 2017-10-30 |
WO2016160980A1 (en) | 2016-10-06 |
JP6768693B2 (ja) | 2020-10-14 |
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