HK1254129A1 - 给予谷氨酰胺酶抑制剂的方法 - Google Patents

给予谷氨酰胺酶抑制剂的方法 Download PDF

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Publication number
HK1254129A1
HK1254129A1 HK18113200.9A HK18113200A HK1254129A1 HK 1254129 A1 HK1254129 A1 HK 1254129A1 HK 18113200 A HK18113200 A HK 18113200A HK 1254129 A1 HK1254129 A1 HK 1254129A1
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group
substituted
alkyl
compound
independently
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HK18113200.9A
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Chinese (zh)
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Matthew I. Gross
Mark K. Bennett
Christopher Molineaux
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Calithera Biosciences, Inc.
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Publication of HK1254129A1 publication Critical patent/HK1254129A1/zh

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/433—Thidiazoles
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    • A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
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  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
HK18113200.9A 2015-03-30 2016-03-30 给予谷氨酰胺酶抑制剂的方法 HK1254129A1 (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201562139928P 2015-03-30 2015-03-30
US62/139928 2015-03-30
US201562168112P 2015-05-29 2015-05-29
US62/168112 2015-05-29
PCT/US2016/024998 WO2016160980A1 (en) 2015-03-30 2016-03-30 Methods of administering glutaminase inhibitors

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EP (1) EP3277276B1 (enExample)
JP (1) JP6768693B2 (enExample)
KR (1) KR20170131650A (enExample)
CN (1) CN107921031A (enExample)
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BR (1) BR112017020780A2 (enExample)
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HUE056078T2 (hu) 2012-11-16 2022-01-28 Calithera Biosciences Inc Heterociklusos glutamináz inhibitorok
HRP20192056T1 (hr) 2014-04-30 2020-02-21 Pfizer Inc. Derivati diheterocikla vezani na cikloalkil
JP6889101B2 (ja) 2014-08-07 2021-06-18 キャリセラ バイオサイエンシーズ， インコーポレイテッド グルタミナーゼ阻害剤の結晶形態
BR112017021312A2 (pt) * 2015-04-06 2018-06-26 Calithera Biosciences Inc tratamento de câncer de pulmão com inibidores de glutaminase
SG11201802830QA (en) 2015-10-05 2018-05-30 Calithera Biosciences Inc Combination therapy with glutaminase inhibitors and immuno-oncology agents
WO2018039441A1 (en) 2016-08-25 2018-03-01 Calithera Biosciences, Inc. Combination therapy with glutaminase inhibitors
WO2018039544A1 (en) 2016-08-25 2018-03-01 Calithera Biosciences, Inc. Combination therapy with glutaminase inhibitors
WO2018102715A1 (en) * 2016-12-02 2018-06-07 Indiana University Research And Technology Corporation Compositions and methods for treating and/or reducing corneal dystrophy
WO2020086440A1 (en) * 2018-10-22 2020-04-30 Beth Israel Deaconess Medical Center Immunomodulatory compounds
US20240016775A1 (en) * 2020-02-24 2024-01-18 Fukang (Shanghai) Health Technology Co., Ltd Anti-coronavirus application of poly adp ribose polymerase inhibitor
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