JP5885670B2 - 黄斑変性の処置のための組成物および方法 - Google Patents

黄斑変性の処置のための組成物および方法 Download PDF

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Publication number
JP5885670B2
JP5885670B2 JP2012543284A JP2012543284A JP5885670B2 JP 5885670 B2 JP5885670 B2 JP 5885670B2 JP 2012543284 A JP2012543284 A JP 2012543284A JP 2012543284 A JP2012543284 A JP 2012543284A JP 5885670 B2 JP5885670 B2 JP 5885670B2
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compound
composition
cyclodextrin
pharmaceutically acceptable
composition according
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JP2013513612A (ja
JP2013513612A5 (https=
Inventor
トーマス エー． ジョーダン，
トーマス エー． ジョーダン，
ジョン クリフォード キャバラ，
ジョン クリフォード キャバラ，
ジェラルド ディー． ケイグル，
ジェラルド ディー． ケイグル，
Original Assignee
アルデイラ セラピューティクス， インコーポレイテッド
アルデイラ セラピューティクス， インコーポレイテッド
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/423—Oxazoles condensed with carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/40—Cyclodextrins; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0048—Eye, e.g. artificial tears
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Inorganic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
JP2012543284A 2009-12-11 2010-12-09 黄斑変性の処置のための組成物および方法 Active JP5885670B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US28574509P 2009-12-11 2009-12-11
US61/285,745 2009-12-11
PCT/US2010/059719 WO2011072141A1 (en) 2009-12-11 2010-12-09 Compositions and methods for the treatment of macular degeneration

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2014255880A Division JP6063916B2 (ja) 2009-12-11 2014-12-18 黄斑変性の処置のための組成物および方法

Publications (3)

Publication Number Publication Date
JP2013513612A JP2013513612A (ja) 2013-04-22
JP2013513612A5 JP2013513612A5 (https=) 2014-01-30
JP5885670B2 true JP5885670B2 (ja) 2016-03-15

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JP2012543284A Active JP5885670B2 (ja) 2009-12-11 2010-12-09 黄斑変性の処置のための組成物および方法
JP2014255880A Active JP6063916B2 (ja) 2009-12-11 2014-12-18 黄斑変性の処置のための組成物および方法
JP2016083344A Active JP6378242B2 (ja) 2009-12-11 2016-04-19 黄斑変性の処置のための組成物および方法
JP2016245212A Pending JP2017052799A (ja) 2009-12-11 2016-12-19 黄斑変性の処置のための組成物および方法

Family Applications After (3)

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JP2014255880A Active JP6063916B2 (ja) 2009-12-11 2014-12-18 黄斑変性の処置のための組成物および方法
JP2016083344A Active JP6378242B2 (ja) 2009-12-11 2016-04-19 黄斑変性の処置のための組成物および方法
JP2016245212A Pending JP2017052799A (ja) 2009-12-11 2016-12-19 黄斑変性の処置のための組成物および方法

Country Status (4)

Country Link
US (4) US9814701B2 (https=)
JP (4) JP5885670B2 (https=)
CA (1) CA2782015C (https=)
WO (1) WO2011072141A1 (https=)

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