JP5837732B2 - ピルフェニドンおよび薬学的に受容可能な賦形剤のカプセル処方物 - Google Patents

ピルフェニドンおよび薬学的に受容可能な賦形剤のカプセル処方物 Download PDF

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JP5837732B2
JP5837732B2 JP2008532431A JP2008532431A JP5837732B2 JP 5837732 B2 JP5837732 B2 JP 5837732B2 JP 2008532431 A JP2008532431 A JP 2008532431A JP 2008532431 A JP2008532431 A JP 2008532431A JP 5837732 B2 JP5837732 B2 JP 5837732B2
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capsule
pirfenidone
months
capsule according
capsules
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JP2009509962A5 (enExample
JP2009509962A (ja
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ラマチャンドラン ラダクリシュナン,
ラマチャンドラン ラダクリシュナン,
ロナルド ブラディーカ,
ロナルド ブラディーカ,
ケニス サルズボー,
ケニス サルズボー,
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インターミューン, インコーポレイテッド
インターミューン, インコーポレイテッド
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4418Non condensed pyridines; Hydrogenated derivatives thereof having a carbocyclic group directly attached to the heterocyclic ring, e.g. cyproheptadine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4412Non condensed pyridines; Hydrogenated derivatives thereof having oxo groups directly attached to the heterocyclic ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4858Organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/48Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/4841Filling excipients; Inactive ingredients
    • A61K9/4866Organic macromolecular compounds
    • AHUMAN NECESSITIES
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    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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    • A61P17/02Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
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    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/04Drugs for skeletal disorders for non-specific disorders of the connective tissue
    • AHUMAN NECESSITIES
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • AHUMAN NECESSITIES
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    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
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    • A61P27/16Otologicals
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    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
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    • A61P41/00Drugs used in surgical methods, e.g. surgery adjuvants for preventing adhesion or for vitreum substitution
    • AHUMAN NECESSITIES
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • A61P7/10Antioedematous agents; Diuretics
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    • AHUMAN NECESSITIES
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    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Epidemiology (AREA)
  • Pulmonology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Otolaryngology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Surgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Hematology (AREA)
  • Vascular Medicine (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
JP2008532431A 2005-09-22 2006-09-22 ピルフェニドンおよび薬学的に受容可能な賦形剤のカプセル処方物 Active JP5837732B2 (ja)

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Application Number Priority Date Filing Date Title
US72025705P 2005-09-22 2005-09-22
US60/720,257 2005-09-22
PCT/US2006/037057 WO2007038315A2 (en) 2005-09-22 2006-09-22 Capsule formulation of pirfenidone and pharmaceutically acceptable excipients

Related Child Applications (1)

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JP2012180913A Division JP5715101B2 (ja) 2005-09-22 2012-08-17 ピルフェニドンおよび薬学的に受容可能な賦形剤のカプセル処方物

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JP2009509962A JP2009509962A (ja) 2009-03-12
JP2009509962A5 JP2009509962A5 (enExample) 2015-11-05
JP5837732B2 true JP5837732B2 (ja) 2015-12-24

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JP2008532431A Active JP5837732B2 (ja) 2005-09-22 2006-09-22 ピルフェニドンおよび薬学的に受容可能な賦形剤のカプセル処方物
JP2012180913A Active JP5715101B2 (ja) 2005-09-22 2012-08-17 ピルフェニドンおよび薬学的に受容可能な賦形剤のカプセル処方物
JP2014129551A Pending JP2014169341A (ja) 2005-09-22 2014-06-24 ピルフェニドンおよび薬学的に受容可能な賦形剤のカプセル処方物

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JP2012180913A Active JP5715101B2 (ja) 2005-09-22 2012-08-17 ピルフェニドンおよび薬学的に受容可能な賦形剤のカプセル処方物
JP2014129551A Pending JP2014169341A (ja) 2005-09-22 2014-06-24 ピルフェニドンおよび薬学的に受容可能な賦形剤のカプセル処方物

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US (5) US7988994B2 (enExample)
EP (2) EP1940364B2 (enExample)
JP (3) JP5837732B2 (enExample)
KR (3) KR101645069B1 (enExample)
CN (3) CN101267810A (enExample)
AP (2) AP2012006231A0 (enExample)
AU (2) AU2006295440B2 (enExample)
BR (1) BRPI0616324A2 (enExample)
CA (2) CA2762013C (enExample)
CU (1) CU20080043A7 (enExample)
CY (1) CY1115544T1 (enExample)
DK (1) DK1940364T4 (enExample)
EA (1) EA030093B1 (enExample)
EC (1) ECSP088394A (enExample)
ES (1) ES2496144T5 (enExample)
GE (1) GEP20115303B (enExample)
IL (2) IL189273A (enExample)
MA (1) MA29875B1 (enExample)
MX (1) MX2008003882A (enExample)
NO (1) NO345131B1 (enExample)
NZ (3) NZ591443A (enExample)
PL (1) PL1940364T5 (enExample)
PT (1) PT1940364E (enExample)
SI (1) SI1940364T2 (enExample)
TN (1) TNSN08136A1 (enExample)
UA (2) UA115861C2 (enExample)
WO (1) WO2007038315A2 (enExample)
ZA (1) ZA200802237B (enExample)

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