JP5820269B2 - Ｓｇｌｔ２阻害剤を使用する高尿酸血症の治療方法およびｓｇｌｔ２阻害剤を含有する組成物 - Google Patents

Ｓｇｌｔ２阻害剤を使用する高尿酸血症の治療方法およびｓｇｌｔ２阻害剤を含有する組成物 Download PDF

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JP5820269B2
JP5820269B2 JP2011510594A JP2011510594A JP5820269B2 JP 5820269 B2 JP5820269 B2 JP 5820269B2 JP 2011510594 A JP2011510594 A JP 2011510594A JP 2011510594 A JP2011510594 A JP 2011510594A JP 5820269 B2 JP5820269 B2 JP 5820269B2
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sglt2 inhibitor
sglt2
inhibitor
uric acid
hyperuricemia
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JP2011520965A (ja
JP2011520965A5 (enExample
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ブルース・ロバート・レスリー
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AstraZeneca AB
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/351—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom not condensed with another ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7004—Monosaccharides having only carbon, hydrogen and oxygen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H7/00—Compounds containing non-saccharide radicals linked to saccharide radicals by a carbon-to-carbon bond
    • C07H7/04—Carbocyclic radicals

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Organic Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pyrane Compounds (AREA)
JP2011510594A 2008-05-22 2009-05-15 Ｓｇｌｔ２阻害剤を使用する高尿酸血症の治療方法およびｓｇｌｔ２阻害剤を含有する組成物 Expired - Fee Related JP5820269B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US5535208P 2008-05-22 2008-05-22
US61/055,352 2008-05-22
PCT/US2009/044156 WO2009143020A1 (en) 2008-05-22 2009-05-15 Method for treating hyperuricemia employing an sglt2 inhibitor and composition containing same

Related Child Applications (1)

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JP2014128550A Division JP2014205700A (ja) 2008-05-22 2014-06-23 Ｓｇｌｔ２阻害剤を使用する高尿酸血症の治療方法およびｓｇｌｔ２阻害剤を含有する組成物

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JP2011520965A JP2011520965A (ja) 2011-07-21
JP2011520965A5 JP2011520965A5 (enExample) 2012-06-14
JP5820269B2 true JP5820269B2 (ja) 2015-11-24

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JP2011510594A Expired - Fee Related JP5820269B2 (ja) 2008-05-22 2009-05-15 Ｓｇｌｔ２阻害剤を使用する高尿酸血症の治療方法およびｓｇｌｔ２阻害剤を含有する組成物
JP2014128550A Pending JP2014205700A (ja) 2008-05-22 2014-06-23 Ｓｇｌｔ２阻害剤を使用する高尿酸血症の治療方法およびｓｇｌｔ２阻害剤を含有する組成物

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US (1) US8791077B2 (enExample)
EP (2) EP2668953A1 (enExample)
JP (2) JP5820269B2 (enExample)
CN (1) CN102105153B (enExample)
BR (1) BRPI0913129A2 (enExample)
CA (1) CA2725047A1 (enExample)
ES (1) ES2526930T3 (enExample)
MX (1) MX2010012656A (enExample)
WO (1) WO2009143020A1 (enExample)

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EP2291189A1 (en) 2011-03-09
CN102105153B (zh) 2014-03-05
JP2011520965A (ja) 2011-07-21
MX2010012656A (es) 2010-12-20
WO2009143020A1 (en) 2009-11-26
US8791077B2 (en) 2014-07-29
BRPI0913129A2 (pt) 2016-01-05
CA2725047A1 (en) 2009-11-26
EP2291189B1 (en) 2014-10-01
US20110065658A1 (en) 2011-03-17
ES2526930T3 (es) 2015-01-16
CN102105153A (zh) 2011-06-22
JP2014205700A (ja) 2014-10-30
EP2668953A1 (en) 2013-12-04

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