JP5290964B2 - 新規1,4−ジアザ−ビシクロ[3.2.2]ノニルオキサジアゾリル誘導体及びそれらの医学的使用 - Google Patents

新規1,4−ジアザ−ビシクロ[3.2.2]ノニルオキサジアゾリル誘導体及びそれらの医学的使用 Download PDF

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JP5290964B2
JP5290964B2 JP2009512569A JP2009512569A JP5290964B2 JP 5290964 B2 JP5290964 B2 JP 5290964B2 JP 2009512569 A JP2009512569 A JP 2009512569A JP 2009512569 A JP2009512569 A JP 2009512569A JP 5290964 B2 JP5290964 B2 JP 5290964B2
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pain
diaza
bicyclo
disease
disorder
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ペータース、ダン
オルセン、グンナー、エム.
ニールセン、エルセベット、オステルガード
ティンマーマン、ダニエル、ビー.
ロッヘル、スティーブン、チャールズ
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ノイロサーチ アクティーゼルスカブ
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    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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JP2009512569A 2006-05-30 2007-05-29 新規1,4−ジアザ−ビシクロ[3.2.2]ノニルオキサジアゾリル誘導体及びそれらの医学的使用 Expired - Fee Related JP5290964B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US80902406P 2006-05-30 2006-05-30
DKPA200600731 2006-05-30
US60/809,024 2006-05-30
DKPA200600731 2006-05-30
PCT/EP2007/055169 WO2007138038A1 (en) 2006-05-30 2007-05-29 Novel 1,4-diaza-bicyclo[3.2.2]nonyl oxadiazolyl derivatives and their medical use

Publications (3)

Publication Number Publication Date
JP2009538867A JP2009538867A (ja) 2009-11-12
JP2009538867A5 JP2009538867A5 (https=) 2010-05-27
JP5290964B2 true JP5290964B2 (ja) 2013-09-18

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JP2009512569A Expired - Fee Related JP5290964B2 (ja) 2006-05-30 2007-05-29 新規1,4−ジアザ−ビシクロ[3.2.2]ノニルオキサジアゾリル誘導体及びそれらの医学的使用
JP2009512568A Pending JP2009538866A (ja) 2006-05-30 2007-05-29 新規1,4−ジアザ−ビシクロ[3.2.2]ノニルオキサジアゾリル誘導体及びそれらの医学的使用

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US (4) US8158619B2 (https=)
EP (3) EP2194056B1 (https=)
JP (2) JP5290964B2 (https=)
KR (1) KR101458194B1 (https=)
CN (2) CN101432286A (https=)
AT (3) ATE463497T1 (https=)
AU (2) AU2007267174B2 (https=)
BR (1) BRPI0708843A2 (https=)
CA (2) CA2653769A1 (https=)
DE (2) DE602007005802D1 (https=)
DK (2) DK2032574T3 (https=)
ES (1) ES2342334T3 (https=)
IL (1) IL193925A (https=)
MX (2) MX2008014887A (https=)
MY (1) MY147764A (https=)
NO (1) NO20085398L (https=)
NZ (1) NZ571288A (https=)
PL (1) PL2032575T3 (https=)
PT (1) PT2032575E (https=)
RU (1) RU2427581C2 (https=)
UA (1) UA95946C2 (https=)
WO (2) WO2007138038A1 (https=)
ZA (1) ZA200807756B (https=)

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CA2718194A1 (en) 2008-03-11 2009-09-17 Neurosearch A/S Novel 1,4-diaza-bicyclo[3.2.2]nonyl oxadiazolyl derivatives useful as modulator of nicotinic acetylcholine receptors
WO2009150138A1 (en) * 2008-06-10 2009-12-17 Neurosearch A/S Novel oxadiazolyl-diazabicyclononane derivatives and their medical use
US20110263577A1 (en) * 2008-10-13 2011-10-27 Neurosearch A/S Novel oxadiazolyl-diazabicyclononane derivatives and their medical use
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WO2010086279A1 (en) 2009-01-27 2010-08-05 Neurosearch A/S Novel dibenzofuranyl-oxadiazolyl-diazabicyclononane derivatives and their medical use
WO2010086280A1 (en) 2009-01-27 2010-08-05 Neurosearch A/S Novel n-oxides of furanyl-oxadiazolyl-diazabicyclononane derivatives and their medical use
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JO3250B1 (ar) 2009-09-22 2018-09-16 Novartis Ag إستعمال منشطات مستقبل نيكوتينيك أسيتيل كولين ألفا 7
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WO2011073296A1 (en) 2009-12-18 2011-06-23 Neurosearch A/S Diazabicyclononyl oxadiazole compounds and their use as nicotinic acetylcholine receptor modulators
US8986654B2 (en) 2011-04-15 2015-03-24 Danpet Ab Labelled and un-labelled methyl-pyrrolyl-oxadiazolyl-diazabicyclononane derivatives and their medical use
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WO2020163248A1 (en) 2019-02-04 2020-08-13 Skyhawk Therapeutics, Inc. Methods and compositions for modulating splicing
JP2022519294A (ja) * 2019-02-04 2022-03-22 スカイホーク・セラピューティクス・インコーポレーテッド スプライシングを調節するための方法および組成物
EP3920915A4 (en) 2019-02-05 2022-10-05 Skyhawk Therapeutics, Inc. METHODS AND COMPOSITIONS FOR MODULATING SPLICE
CN114126613A (zh) 2019-02-05 2022-03-01 斯基霍克疗法公司 用于调节剪接的方法和组合物
CN113661162A (zh) 2019-02-06 2021-11-16 斯基霍克疗法公司 用于调节剪接的方法和组合物
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US8372832B2 (en) 2013-02-12
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