JP5159604B2 - バニロイド受容体拮抗薬としての新規な化合物、その異性体又はその薬剤学的に許容される塩、及びこれを含む医薬組成物 - Google Patents

バニロイド受容体拮抗薬としての新規な化合物、その異性体又はその薬剤学的に許容される塩、及びこれを含む医薬組成物 Download PDF

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JP5159604B2
JP5159604B2 JP2008502895A JP2008502895A JP5159604B2 JP 5159604 B2 JP5159604 B2 JP 5159604B2 JP 2008502895 A JP2008502895 A JP 2008502895A JP 2008502895 A JP2008502895 A JP 2008502895A JP 5159604 B2 JP5159604 B2 JP 5159604B2
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fluoro
butyl
mmol
methanesulfonylamino
hydrogen
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JP2008538109A (ja
JP2008538109A5 (https=
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キム・ヘド
スー・ヨンガー
パク・ヒュングン
オー・ウーテク
パク・ソルリン
キム・ジョヒュン
ジャン・ミジュン
パク・ヨンホ
シン・ソンソク
キム・スンヨン
キム・ジンクワン
ジョン・ヨンス
リ・キワ
チョイ・ジンキュ
リム・キュンミン
コー・ヒュンジュ
モー・ジョヒュン
キム・スンイル
ウー・ビョンヨン
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Amorepacific Corp
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JP2008502895A 2005-03-19 2006-03-15 バニロイド受容体拮抗薬としての新規な化合物、その異性体又はその薬剤学的に許容される塩、及びこれを含む医薬組成物 Expired - Fee Related JP5159604B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
KR10-2005-0022986 2005-03-19
KR20050022986 2005-03-19
US66326905P 2005-03-21 2005-03-21
US60/663,269 2005-03-21
PCT/KR2006/000929 WO2006101318A1 (en) 2005-03-19 2006-03-15 Novel compounds, isomer thereof, or pharmaceutically acceptable salts thereof as vanilloid receptor antagonist; and pharmaceutical compositions containing the same

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JP2008538109A JP2008538109A (ja) 2008-10-09
JP2008538109A5 JP2008538109A5 (https=) 2009-04-09
JP5159604B2 true JP5159604B2 (ja) 2013-03-06

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JP2008502895A Expired - Fee Related JP5159604B2 (ja) 2005-03-19 2006-03-15 バニロイド受容体拮抗薬としての新規な化合物、その異性体又はその薬剤学的に許容される塩、及びこれを含む医薬組成物
JP2008502896A Expired - Fee Related JP5064374B2 (ja) 2005-03-19 2006-03-17 バニロイド受容体拮抗薬としての新規な化合物、その異性体またはその薬剤学的に許容される塩、及びこれを含む医薬組成物

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US (2) US7763657B2 (https=)
EP (2) EP1861357B1 (https=)
JP (2) JP5159604B2 (https=)
KR (2) KR101304981B1 (https=)
AR (2) AR053561A1 (https=)
AU (2) AU2006225496A1 (https=)
BR (2) BRPI0608714A2 (https=)
CA (2) CA2601871A1 (https=)
EA (2) EA200702020A1 (https=)
IL (2) IL185891A0 (https=)
MX (2) MX2007011466A (https=)
NO (2) NO20075353L (https=)
TW (2) TW200716523A (https=)
WO (2) WO2006101318A1 (https=)

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KR101304981B1 (ko) * 2005-03-19 2013-09-06 (주)아모레퍼시픽 바닐로이드 수용체 길항물질로서의 신규 화합물, 이의이성체 또는 이의 약학적으로 허용가능한 염, 및 이를함유하는 약학 조성물
PL2054411T3 (pl) 2006-07-27 2015-02-27 Amorepacific Corp Nowe związki, ich izomery lub ich farmaceutycznie dopuszczalne sole jako antagoniści receptora waniloidowego oraz zawierające je kompozycje farmaceutyczne
DE102007017884A1 (de) 2007-04-13 2008-10-16 Grünethal GmbH Neue Vanilloid-Rezeptor Liganden und ihre Verwendung zur Herstellung von Arzneimitteln
US20110160279A1 (en) * 2007-08-13 2011-06-30 Board Of Trustees Of Southern Illinois University METHODS FOR TREATMENT AND PREVENTION OF OTOTOXICITY BY siRNA
US8557872B2 (en) 2008-01-28 2013-10-15 Amorepacific Corporation Compounds, isomer thereof, or pharmaceutically acceptable salts thereof as vanilloid receptor antagonist; and pharmaceutical compositions containing the same
WO2009136625A1 (ja) * 2008-05-07 2009-11-12 大日本住友製薬株式会社 環状アミン－１－カルボン酸エステル誘導体およびそれを含有する医薬組成物
US8691855B2 (en) 2008-07-02 2014-04-08 Amorepacific Corporation Compounds, isomer thereof, or pharmaceutically acceptable salts thereof as vanilloid receptor antagonist and pharmaceutical compositions containing the same
CN103429242A (zh) * 2010-11-03 2013-12-04 夏威夷大学 用于预防和治疗心脏肥大的方法和组合物
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US20080234383A1 (en) 2008-09-25
BRPI0608624A2 (pt) 2010-01-19
EA200702020A1 (ru) 2008-02-28
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NO20075353L (no) 2007-12-18
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EP1861357A4 (en) 2011-08-31
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TW200716522A (en) 2007-05-01
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