JP5159604B2 - バニロイド受容体拮抗薬としての新規な化合物、その異性体又はその薬剤学的に許容される塩、及びこれを含む医薬組成物 - Google Patents

バニロイド受容体拮抗薬としての新規な化合物、その異性体又はその薬剤学的に許容される塩、及びこれを含む医薬組成物 Download PDF

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JP5159604B2
JP5159604B2 JP2008502895A JP2008502895A JP5159604B2 JP 5159604 B2 JP5159604 B2 JP 5159604B2 JP 2008502895 A JP2008502895 A JP 2008502895A JP 2008502895 A JP2008502895 A JP 2008502895A JP 5159604 B2 JP5159604 B2 JP 5159604B2
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fluoro
butyl
mmol
methanesulfonylamino
hydrogen
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JP2008538109A (ja
JP2008538109A5 (enExample
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キム・ヘド
スー・ヨンガー
パク・ヒュングン
オー・ウーテク
パク・ソルリン
キム・ジョヒュン
ジャン・ミジュン
パク・ヨンホ
シン・ソンソク
キム・スンヨン
キム・ジンクワン
ジョン・ヨンス
リ・キワ
チョイ・ジンキュ
リム・キュンミン
コー・ヒュンジュ
モー・ジョヒュン
キム・スンイル
ウー・ビョンヨン
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Amorepacific Corp
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  • Hydrogenated Pyridines (AREA)
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JP2008502895A 2005-03-19 2006-03-15 バニロイド受容体拮抗薬としての新規な化合物、その異性体又はその薬剤学的に許容される塩、及びこれを含む医薬組成物 Expired - Fee Related JP5159604B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
KR20050022986 2005-03-19
KR10-2005-0022986 2005-03-19
US66326905P 2005-03-21 2005-03-21
US60/663,269 2005-03-21
PCT/KR2006/000929 WO2006101318A1 (en) 2005-03-19 2006-03-15 Novel compounds, isomer thereof, or pharmaceutically acceptable salts thereof as vanilloid receptor antagonist; and pharmaceutical compositions containing the same

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JP2008538109A JP2008538109A (ja) 2008-10-09
JP2008538109A5 JP2008538109A5 (enExample) 2009-04-09
JP5159604B2 true JP5159604B2 (ja) 2013-03-06

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JP2008502895A Expired - Fee Related JP5159604B2 (ja) 2005-03-19 2006-03-15 バニロイド受容体拮抗薬としての新規な化合物、その異性体又はその薬剤学的に許容される塩、及びこれを含む医薬組成物
JP2008502896A Expired - Fee Related JP5064374B2 (ja) 2005-03-19 2006-03-17 バニロイド受容体拮抗薬としての新規な化合物、その異性体またはその薬剤学的に許容される塩、及びこれを含む医薬組成物

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US (2) US7763657B2 (enExample)
EP (2) EP1861357B1 (enExample)
JP (2) JP5159604B2 (enExample)
KR (2) KR101304981B1 (enExample)
AR (2) AR056943A1 (enExample)
AU (2) AU2006225496A1 (enExample)
BR (2) BRPI0608714A2 (enExample)
CA (2) CA2601871A1 (enExample)
EA (2) EA200702020A1 (enExample)
IL (2) IL185891A0 (enExample)
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MX2007011466A (es) 2005-03-19 2008-01-16 Amorepacific Corp Compuestos novedosos, isomeros de los mismos, o sales farmaceuticamente aceptables de los mismos como antagonistas de receptor de vaniloides, y composiciones farmaceuticas que contienen los mismos.
PL2054411T3 (pl) 2006-07-27 2015-02-27 Amorepacific Corp Nowe związki, ich izomery lub ich farmaceutycznie dopuszczalne sole jako antagoniści receptora waniloidowego oraz zawierające je kompozycje farmaceutyczne
DE102007017884A1 (de) * 2007-04-13 2008-10-16 Grünethal GmbH Neue Vanilloid-Rezeptor Liganden und ihre Verwendung zur Herstellung von Arzneimitteln
WO2009023025A1 (en) * 2007-08-13 2009-02-19 Board Of Trustees Of Southern Illinois University Methods for treatment and prevention of ototoxicity by sirna
CN101925575B (zh) 2008-01-28 2014-06-18 株式会社爱茉莉太平洋 作为香草酸受体拮抗剂的化合物、其异构体或其药物学可接受的盐、及包含这些化合物的药物组合物
US8367835B2 (en) 2008-05-07 2013-02-05 Dainippon Sumitomo Pharma Co., Ltd. Cyclic amine-1-carboxylic acid ester derivative and pharmaceutical composition containing the same
EP2307394B1 (en) 2008-07-02 2012-09-26 Amorepacific Corporation Sulphonamides as vanilloid receptor antagonist
EP3348267B1 (en) * 2010-11-03 2024-01-10 University Of Hawaii Trpv1 inhibitor for prevention and treatment of cardiac hypertrophy
AR085509A1 (es) 2011-03-09 2013-10-09 Bayer Cropscience Ag Indol- y bencimidazolcarboxamidas como insecticidas y acaricidas
DK3738434T3 (da) 2011-12-28 2023-12-04 Global Blood Therapeutics Inc Mellemprodukter til opnåelse af substituerede benzaldehydforbindelser og fremgangsmåder til anvendelse deraf ved øgning af vævsoxygenering
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CA2601871A1 (en) 2006-09-28
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US7960584B2 (en) 2011-06-14
EA200702020A1 (ru) 2008-02-28
NO20075354L (no) 2007-12-18
TW200716522A (en) 2007-05-01
EP1861358A4 (en) 2011-08-31
KR101304981B1 (ko) 2013-09-06
EP1861358A1 (en) 2007-12-05
BRPI0608714A2 (pt) 2010-01-26
US20080234383A1 (en) 2008-09-25
KR20080007329A (ko) 2008-01-18
NO20075353L (no) 2007-12-18
AU2006225434A1 (en) 2006-09-28
US20090105258A1 (en) 2009-04-23
JP2008538109A (ja) 2008-10-09
EP1861357A1 (en) 2007-12-05
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AR056943A1 (es) 2007-11-07
AU2006225496A1 (en) 2006-09-28
IL185892A0 (en) 2008-02-09
BRPI0608624A2 (pt) 2010-01-19
JP5064374B2 (ja) 2012-10-31
WO2006101318A1 (en) 2006-09-28
KR20070114821A (ko) 2007-12-04
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CA2601873A1 (en) 2006-09-28
EP1861357A4 (en) 2011-08-31
IL185891A0 (en) 2008-02-09
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