JP4707389B2 - プロテインキナーゼ依存性疾患の処置における１Ｈ−イミダゾ［４，５−ｃ］キノリン誘導体 - Google Patents

プロテインキナーゼ依存性疾患の処置における１Ｈ−イミダゾ［４，５−ｃ］キノリン誘導体 Download PDF

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JP4707389B2
JP4707389B2 JP2004505373A JP2004505373A JP4707389B2 JP 4707389 B2 JP4707389 B2 JP 4707389B2 JP 2004505373 A JP2004505373 A JP 2004505373A JP 2004505373 A JP2004505373 A JP 2004505373A JP 4707389 B2 JP4707389 B2 JP 4707389B2
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phenyl
chloro
formula
imidazo
compounds
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JP2005534636A5 (https=
JP2005534636A (ja
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カルロス・ガルシア−エチェベリア
ハンス−ゲオルク・カプラロ
パスカル・フュレ
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ノバルティス アーゲー
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP2004505373A 2002-05-21 2003-05-20 プロテインキナーゼ依存性疾患の処置における１Ｈ−イミダゾ［４，５−ｃ］キノリン誘導体 Expired - Fee Related JP4707389B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0211649.9 2002-05-21
GBGB0211649.9A GB0211649D0 (en) 2002-05-21 2002-05-21 Organic compounds
PCT/EP2003/005291 WO2003097641A2 (en) 2002-05-21 2003-05-20 1h-imidazo[4,5-c] quinoline derivatives in the treatment of protein kinase dependent diseases

Publications (3)

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JP2005534636A JP2005534636A (ja) 2005-11-17
JP2005534636A5 JP2005534636A5 (https=) 2010-05-06
JP4707389B2 true JP4707389B2 (ja) 2011-06-22

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JP2004505373A Expired - Fee Related JP4707389B2 (ja) 2002-05-21 2003-05-20 プロテインキナーゼ依存性疾患の処置における１Ｈ−イミダゾ［４，５−ｃ］キノリン誘導体

Country Status (15)

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US (1) US7998972B2 (https=)
EP (1) EP1509521B8 (https=)
JP (1) JP4707389B2 (https=)
CN (1) CN100475207C (https=)
AT (1) ATE405564T1 (https=)
AU (1) AU2003240680A1 (https=)
BR (1) BR0311221A (https=)
CA (1) CA2485012A1 (https=)
DE (1) DE60323090D1 (https=)
DK (1) DK1509521T3 (https=)
ES (1) ES2312783T3 (https=)
GB (1) GB0211649D0 (https=)
PT (1) PT1509521E (https=)
SI (1) SI1509521T1 (https=)
WO (1) WO2003097641A2 (https=)

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