ATE405564T1 - 1h-imidazoä4,5-cüchinolinderivate zur behandlung von protein kinase-abhängigen krankheiten - Google Patents

1h-imidazoä4,5-cüchinolinderivate zur behandlung von protein kinase-abhängigen krankheiten

Info

Publication number
ATE405564T1
ATE405564T1 AT03730079T AT03730079T ATE405564T1 AT E405564 T1 ATE405564 T1 AT E405564T1 AT 03730079 T AT03730079 T AT 03730079T AT 03730079 T AT03730079 T AT 03730079T AT E405564 T1 ATE405564 T1 AT E405564T1
Authority
AT
Austria
Prior art keywords
treatment
protein kinase
imidazoä4
cuchinolin
derivatives
Prior art date
Application number
AT03730079T
Other languages
English (en)
Inventor
Carlos Garcia-Echeverria
Hans-Georg Capraro
Pascal Furet
Original Assignee
Novartis Pharma Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Pharma Gmbh filed Critical Novartis Pharma Gmbh
Application granted granted Critical
Publication of ATE405564T1 publication Critical patent/ATE405564T1/de

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/06—Antipsoriatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Enzymes And Modification Thereof (AREA)
AT03730079T 2002-05-21 2003-05-20 1h-imidazoä4,5-cüchinolinderivate zur behandlung von protein kinase-abhängigen krankheiten ATE405564T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GBGB0211649.9A GB0211649D0 (en) 2002-05-21 2002-05-21 Organic compounds

Publications (1)

Publication Number Publication Date
ATE405564T1 true ATE405564T1 (de) 2008-09-15

Family

ID=9937093

Family Applications (1)

Application Number Title Priority Date Filing Date
AT03730079T ATE405564T1 (de) 2002-05-21 2003-05-20 1h-imidazoä4,5-cüchinolinderivate zur behandlung von protein kinase-abhängigen krankheiten

Country Status (16)

Country Link
US (1) US7998972B2 (de)
EP (1) EP1509521B8 (de)
JP (1) JP4707389B2 (de)
CN (1) CN100475207C (de)
AT (1) ATE405564T1 (de)
AU (1) AU2003240680A1 (de)
BR (1) BR0311221A (de)
CA (1) CA2485012A1 (de)
DE (1) DE60323090D1 (de)
DK (1) DK1509521T3 (de)
ES (1) ES2312783T3 (de)
GB (1) GB0211649D0 (de)
HK (1) HK1074837A1 (de)
PT (1) PT1509521E (de)
SI (1) SI1509521T1 (de)
WO (1) WO2003097641A2 (de)

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EP1509521B8 (de) 2009-02-18
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ES2312783T3 (es) 2009-03-01
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US7998972B2 (en) 2011-08-16
AU2003240680A1 (en) 2003-12-02
EP1509521B1 (de) 2008-08-20
JP4707389B2 (ja) 2011-06-22
WO2003097641A3 (en) 2004-05-06
US20050245562A1 (en) 2005-11-03
HK1074837A1 (en) 2005-11-25
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