JP2025508971A5 - - Google Patents

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Publication number
JP2025508971A5
JP2025508971A5 JP2024552216A JP2024552216A JP2025508971A5 JP 2025508971 A5 JP2025508971 A5 JP 2025508971A5 JP 2024552216 A JP2024552216 A JP 2024552216A JP 2024552216 A JP2024552216 A JP 2024552216A JP 2025508971 A5 JP2025508971 A5 JP 2025508971A5
Authority
JP
Japan
Prior art keywords
heterocycloalkyl
cycloalkyl
alkyl
pharmaceutically acceptable
heteroaryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024552216A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025508971A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/CN2023/078948 external-priority patent/WO2023165504A1/en
Publication of JP2025508971A publication Critical patent/JP2025508971A/ja
Publication of JP2025508971A5 publication Critical patent/JP2025508971A5/ja
Pending legal-status Critical Current

Links

JP2024552216A 2022-03-01 2023-03-01 ジアシルグリセロールキナーゼ(DGK)α阻害剤及びその使用 Pending JP2025508971A (ja)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
CN2022078653 2022-03-01
CNPCT/CN2022/078653 2022-03-01
CN2022091497 2022-05-07
CNPCT/CN2022/091497 2022-05-07
CNPCT/CN2022/127020 2022-10-24
CN2022127020 2022-10-24
CNPCT/CN2023/071857 2023-01-12
CN2023071857 2023-01-12
PCT/CN2023/078948 WO2023165504A1 (en) 2022-03-01 2023-03-01 Diacylglycerol kinase (dgk) alpha inhibitors and uses thereof

Publications (2)

Publication Number Publication Date
JP2025508971A JP2025508971A (ja) 2025-04-10
JP2025508971A5 true JP2025508971A5 (https=) 2026-03-09

Family

ID=87883011

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024552216A Pending JP2025508971A (ja) 2022-03-01 2023-03-01 ジアシルグリセロールキナーゼ(DGK)α阻害剤及びその使用

Country Status (12)

Country Link
US (2) US20240051958A1 (https=)
EP (1) EP4486741A4 (https=)
JP (1) JP2025508971A (https=)
KR (1) KR20240156394A (https=)
CN (1) CN118871438A (https=)
AR (1) AR128669A1 (https=)
AU (1) AU2023227010A1 (https=)
CA (1) CA3244501A1 (https=)
IL (1) IL315015A (https=)
MX (1) MX2024010648A (https=)
TW (1) TW202342477A (https=)
WO (1) WO2023165504A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4486741A4 (en) 2022-03-01 2026-04-08 Insilico Medicine Ip Ltd Diacylglycerol Kinase (DGK) Alpha Inhibitors and Their Uses
EP4661869A1 (en) 2023-02-06 2025-12-17 Bayer Aktiengesellschaft Combinations of dgk (diacylglycerol kinase) inhibitors and immune checkpoint inhibitors and modulators
WO2025051110A1 (en) * 2023-09-04 2025-03-13 Insilico Medicine Ip Limited Combinations treatments of diacylglycerol kinase (dgk) alpha inhibitors and other therapies

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