JP2025513882A5 - - Google Patents

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Publication number
JP2025513882A5
JP2025513882A5 JP2024560672A JP2024560672A JP2025513882A5 JP 2025513882 A5 JP2025513882 A5 JP 2025513882A5 JP 2024560672 A JP2024560672 A JP 2024560672A JP 2024560672 A JP2024560672 A JP 2024560672A JP 2025513882 A5 JP2025513882 A5 JP 2025513882A5
Authority
JP
Japan
Prior art keywords
alkyl
heterocycloalkyl
cycloalkyl
heteroaryl
aryl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024560672A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025513882A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2023/018508 external-priority patent/WO2023200964A1/en
Publication of JP2025513882A publication Critical patent/JP2025513882A/ja
Publication of JP2025513882A5 publication Critical patent/JP2025513882A5/ja
Pending legal-status Critical Current

Links

JP2024560672A 2022-04-14 2023-04-13 タンパク質チロシンホスファターゼ阻害剤およびその使用 Pending JP2025513882A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US202263331073P 2022-04-14 2022-04-14
US63/331,073 2022-04-14
US202363486559P 2023-02-23 2023-02-23
US63/486,559 2023-02-23
PCT/US2023/018508 WO2023200964A1 (en) 2022-04-14 2023-04-13 Protein tyrosine phosphatase inhibitors and uses thereof

Publications (2)

Publication Number Publication Date
JP2025513882A JP2025513882A (ja) 2025-04-30
JP2025513882A5 true JP2025513882A5 (https=) 2026-04-20

Family

ID=88330255

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024560672A Pending JP2025513882A (ja) 2022-04-14 2023-04-13 タンパク質チロシンホスファターゼ阻害剤およびその使用

Country Status (6)

Country Link
US (1) US20250257059A1 (https=)
EP (1) EP4508050A4 (https=)
JP (1) JP2025513882A (https=)
CN (1) CN119365452A (https=)
TW (1) TW202404964A (https=)
WO (1) WO2023200964A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4522594A4 (en) * 2022-05-13 2026-04-22 Mondego Bio Lda A Limited Liability Company By Quotas Soc Por Quotas PTPN2 INHIBITORS
JP2025539027A (ja) * 2022-11-09 2025-12-03 ブリストル-マイヤーズ スクイブ カンパニー タンパク質チロシンホスファターゼの阻害剤、組成物、および使用方法
PE20252789A1 (es) 2023-05-24 2025-12-22 Kumquat Biosciences Inc Compuestos heterociclicos y usos de estos
WO2025030008A1 (en) * 2023-08-02 2025-02-06 Nerio Therapeutics, Inc. Protein tyrosine phosphatase inhibitor combinations
CN119707953A (zh) * 2024-04-19 2025-03-28 中国药科大学 噻二唑烷酮衍生物及其制备方法和应用
WO2026037253A1 (zh) * 2024-08-10 2026-02-19 杭州英创医药科技有限公司 作为ptpn抑制剂的化合物
CN121591722A (zh) * 2024-08-22 2026-03-03 武汉人福创新药物研发中心有限公司 作为蛋白质酪氨酸磷酸酶抑制剂的含双键取代的化合物及其应用

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2630448A1 (en) * 2005-12-08 2007-06-14 Novartis Ag 1,1,3-trioxo-1,2,5-thiadiazolidines and their use as ptp-ases inhibitors
CA2647472A1 (en) * 2006-03-31 2007-10-11 Novartis Ag Organic compounds
IL286373B2 (en) * 2019-03-14 2026-03-01 Calico Life Sciences Llc Protein tyrosine phosphate inhibitor compounds and uses thereof
EP4351558A4 (en) * 2021-06-10 2025-05-07 Ness Therapeutics, Inc. Compounds containing 5-(2-fluoro-6-hydroxyphenyl)-1,2,5-thiazolidin-3-one 1,1-dioxide as inhibitors of protein kinase phosphatase enzymes

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