JP2021519271A5 - - Google Patents
Info
- Publication number
- JP2021519271A5 JP2021519271A5 JP2020551349A JP2020551349A JP2021519271A5 JP 2021519271 A5 JP2021519271 A5 JP 2021519271A5 JP 2020551349 A JP2020551349 A JP 2020551349A JP 2020551349 A JP2020551349 A JP 2020551349A JP 2021519271 A5 JP2021519271 A5 JP 2021519271A5
- Authority
- JP
- Japan
- Prior art keywords
- disorder
- agonists
- compound
- free
- formula
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2024102491A JP2024123211A (ja) | 2018-03-23 | 2024-06-26 | 有機化合物 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862647482P | 2018-03-23 | 2018-03-23 | |
| US62/647,482 | 2018-03-23 | ||
| PCT/US2019/023687 WO2019183546A1 (en) | 2018-03-23 | 2019-03-22 | Organic compounds |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024102491A Division JP2024123211A (ja) | 2018-03-23 | 2024-06-26 | 有機化合物 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2021519271A JP2021519271A (ja) | 2021-08-10 |
| JP2021519271A5 true JP2021519271A5 (enExample) | 2022-02-17 |
Family
ID=67987581
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020551349A Pending JP2021519271A (ja) | 2018-03-23 | 2019-03-22 | 有機化合物 |
| JP2024102491A Pending JP2024123211A (ja) | 2018-03-23 | 2024-06-26 | 有機化合物 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024102491A Pending JP2024123211A (ja) | 2018-03-23 | 2024-06-26 | 有機化合物 |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US20210008065A1 (enExample) |
| EP (1) | EP3768271B1 (enExample) |
| JP (2) | JP2021519271A (enExample) |
| CN (1) | CN112088004A (enExample) |
| AU (2) | AU2019236860B2 (enExample) |
| BR (1) | BR112020019181A2 (enExample) |
| CA (1) | CA3095101A1 (enExample) |
| DK (1) | DK3768271T3 (enExample) |
| FI (1) | FI3768271T3 (enExample) |
| IL (2) | IL277509B2 (enExample) |
| MX (1) | MX2020009929A (enExample) |
| WO (1) | WO2019183546A1 (enExample) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR102373288B1 (ko) * | 2013-12-03 | 2022-03-10 | 인트라-셀룰라 써래피스, 인코퍼레이티드. | 신규한 방법 |
| PL3838274T3 (pl) | 2016-01-26 | 2024-04-02 | Intra-Cellular Therapies, Inc. | Pochodna pirydo[3',4':4,5]pirolo[1,2,3-DE]chinoksaliny do zastosowania w leczeniu zaburzeń OUN |
| RU2767410C2 (ru) | 2017-03-24 | 2022-03-17 | Интра-Селлулар Терапиз, Инк. | Новые композиции и способы |
| EP3658144B1 (en) | 2017-07-26 | 2022-01-26 | Intra-Cellular Therapies, Inc. | Pyridopyrroloquinoxaline compounds, their compositions and uses in therapy |
| US11440911B2 (en) | 2017-09-26 | 2022-09-13 | Intra-Cellular Therapies, Inc. | Salts and crystals |
| WO2019178484A1 (en) | 2018-03-16 | 2019-09-19 | Intra-Cellular Therapies, Inc. | Novel methods |
| CN112040940A (zh) | 2018-03-23 | 2020-12-04 | 细胞内治疗公司 | 有机化合物 |
| CA3240552A1 (en) | 2018-06-11 | 2019-12-19 | Intra-Cellular Therapies, Inc. | Substituted heterocycle fused gamma-carbolines synthesis |
| WO2020047408A1 (en) | 2018-08-31 | 2020-03-05 | Intra-Cellular Therapies, Inc. | Novel methods |
| BR112021003655A2 (pt) | 2018-08-31 | 2021-05-18 | Intra-Cellular Therapies, Inc. | métodos novos |
| JP7520013B2 (ja) | 2018-12-17 | 2024-07-22 | イントラ－セルラー・セラピーズ・インコーポレイテッド | 置換複素環縮合γ－カルボリンの合成 |
| JP7649743B2 (ja) | 2018-12-21 | 2025-03-21 | イントラ－セルラー・セラピーズ・インコーポレイテッド | 有機化合物 |
| WO2021007245A1 (en) | 2019-07-07 | 2021-01-14 | Intra-Cellular Therapies, Inc. | Novel methods |
| US12478623B2 (en) | 2019-09-25 | 2025-11-25 | Intra-Cellular Therapies, Inc. | Methods of treating central nervous system disorders comprising administering lumateperone and a nitric oxide donor |
| EP4072554A4 (en) | 2019-12-11 | 2023-12-20 | Intra-Cellular Therapies, Inc. | ORGANIC CONNECTION |
| JP7533361B2 (ja) * | 2021-05-26 | 2024-08-14 | 株式会社三洋物産 | 遊技機 |
| US12414948B2 (en) | 2022-05-18 | 2025-09-16 | Intra-Cellular Therapies, Inc. | Methods |
| CN119486738A (zh) | 2022-05-18 | 2025-02-18 | 细胞内治疗公司 | 新方法 |
| WO2024173901A1 (en) | 2023-02-17 | 2024-08-22 | Intra-Cellular Therapies, Inc. | Lumateperone and derivatives thereof for modulating the nervous system |
| WO2025111568A1 (en) | 2023-11-22 | 2025-05-30 | Intra-Cellular Therapies, Inc. | Lumateperone and analogues, as 5-ht2a or 5-ht2a/d2 receptor modulators, for use in the treatment of psychiatric disorders caused by viral, bacterial, or autoimmune encephalitis, and of psychiatric symptoms thereof |
| US20250352469A1 (en) | 2024-05-16 | 2025-11-20 | Intra-Cellular Therapies, Inc. | Novel compositions, devices, and methods |
| WO2025257090A1 (en) | 2024-06-10 | 2025-12-18 | Interquim, S.A. | Process for the preparation of synthesis intermediates of lumateperone and lumateperone analogues |
Family Cites Families (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4389330A (en) | 1980-10-06 | 1983-06-21 | Stolle Research And Development Corporation | Microencapsulation process |
| IE52535B1 (en) | 1981-02-16 | 1987-12-09 | Ici Plc | Continuous release pharmaceutical compositions |
| US4530840A (en) | 1982-07-29 | 1985-07-23 | The Stolle Research And Development Corporation | Injectable, long-acting microparticle formulation for the delivery of anti-inflammatory agents |
| CH656884A5 (de) | 1983-08-26 | 1986-07-31 | Sandoz Ag | Polyolester, deren herstellung und verwendung. |
| US5538739A (en) | 1989-07-07 | 1996-07-23 | Sandoz Ltd. | Sustained release formulations of water soluble peptides |
| CN1074923C (zh) | 1993-11-19 | 2001-11-21 | 詹森药业有限公司 | 微囊密封的3-哌啶基取代的1,2-苯并异唑类和1,2-苯并异噻唑类 |
| PT1140012E (pt) | 1998-12-17 | 2004-05-31 | Alza Corp | Conversao de capsulas de gelatina cheias com liquido em sistemas de libertacao controlada por camadas multiplas |
| ATE277048T1 (de) | 1999-06-15 | 2004-10-15 | Bristol Myers Squibb Pharma Co | Substituierte hetercyclisch kondensierte gamma carboline |
| US7071186B2 (en) | 1999-06-15 | 2006-07-04 | Bristol-Myers Squibb Pharma Co. | Substituted heterocycle fused gamma-carbolines |
| US6713471B1 (en) | 1999-06-15 | 2004-03-30 | Bristol-Myers Squibb Pharma Company | Substituted heterocycle fused gamma-carbolines |
| US20050232995A1 (en) | 2002-07-29 | 2005-10-20 | Yam Nyomi V | Methods and dosage forms for controlled delivery of paliperidone and risperidone |
| NZ570198A (en) | 2002-07-29 | 2010-01-29 | Alza Corp | Methods and dosage forms for controlled delivery of paliperidone or risperidone |
| KR102107954B1 (ko) | 2007-03-12 | 2020-05-07 | 인트라-셀룰라 써래피스, 인코퍼레이티드. | 치환된 헤테로환 융합 감마-카르볼린 합성 |
| AU2009223701B2 (en) | 2008-03-12 | 2015-04-16 | Intra-Cellular Therapies, Inc. | Substituted heterocycle fused gamma-carbolines solid |
| EP3085231A1 (en) | 2008-05-27 | 2016-10-26 | Intra-Cellular Therapies, Inc. | Method and compositions for sleep disorders and other disorders |
| CA2796756A1 (en) | 2010-04-22 | 2011-10-27 | Intra-Cellular Therapies, Inc. | Substituted pyrido(3',4':4,5)pyrrolo(1,2,3-de)quinoxalines for the treatment of central nervous system disorders |
| KR20140146192A (ko) | 2012-04-14 | 2014-12-24 | 인트라-셀룰라 써래피스, 인코퍼레이티드. | 유기 화합물 |
| AR092568A1 (es) * | 2012-09-14 | 2015-04-22 | Abbvie Deutschland | Derivados triciclicos de quinolinas y de quinoxalinas |
| CA2944755A1 (en) * | 2014-04-04 | 2015-10-08 | Intra-Cellular Therapies, Inc. | Organic compounds |
| US10077267B2 (en) | 2014-04-04 | 2018-09-18 | Intra-Cellular Therapies, Inc. | Organic compounds |
| WO2017117514A1 (en) * | 2015-12-31 | 2017-07-06 | Tung Roger D | Deuterated iti-007 |
| DK3407889T3 (da) * | 2016-03-25 | 2021-08-09 | Intra Cellular Therapies Inc | Organiske forbindelser og deres anvendelse til behandling og forebyggelse af lidelser i centralnervesystemet |
-
2019
- 2019-03-22 US US17/040,893 patent/US20210008065A1/en active Pending
- 2019-03-22 AU AU2019236860A patent/AU2019236860B2/en active Active
- 2019-03-22 WO PCT/US2019/023687 patent/WO2019183546A1/en not_active Ceased
- 2019-03-22 MX MX2020009929A patent/MX2020009929A/es unknown
- 2019-03-22 FI FIEP19771617.8T patent/FI3768271T3/fi active
- 2019-03-22 DK DK19771617.8T patent/DK3768271T3/da active
- 2019-03-22 CN CN201980028290.1A patent/CN112088004A/zh active Pending
- 2019-03-22 IL IL277509A patent/IL277509B2/en unknown
- 2019-03-22 EP EP19771617.8A patent/EP3768271B1/en active Active
- 2019-03-22 JP JP2020551349A patent/JP2021519271A/ja active Pending
- 2019-03-22 IL IL303857A patent/IL303857B2/en unknown
- 2019-03-22 BR BR112020019181-7A patent/BR112020019181A2/pt unknown
- 2019-03-22 CA CA3095101A patent/CA3095101A1/en active Pending
-
2024
- 2024-06-26 JP JP2024102491A patent/JP2024123211A/ja active Pending
-
2025
- 2025-02-07 AU AU2025200857A patent/AU2025200857A1/en active Pending
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