JP2021511342A5 - - Google Patents

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JP2021511342A5
JP2021511342A5 JP2020540426A JP2020540426A JP2021511342A5 JP 2021511342 A5 JP2021511342 A5 JP 2021511342A5 JP 2020540426 A JP2020540426 A JP 2020540426A JP 2020540426 A JP2020540426 A JP 2020540426A JP 2021511342 A5 JP2021511342 A5 JP 2021511342A5
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JP2020540426A 2018-01-22 2019-01-22 癌処置のためのbcl-2タンパク質分解剤 Active JP7385284B2 (ja)

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US201862620219P 2018-01-22 2018-01-22
US62/620,219 2018-01-22
PCT/US2019/014545 WO2019144117A1 (en) 2018-01-22 2019-01-22 Bcl-2 proteins degraders for cancer treatment

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JP2021511342A JP2021511342A (ja) 2021-05-06
JP2021511342A5 true JP2021511342A5 (enExample) 2022-01-31
JP7385284B2 JP7385284B2 (ja) 2023-11-22

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US (1) US12118414B2 (enExample)
EP (1) EP3743069B1 (enExample)
JP (1) JP7385284B2 (enExample)
CN (1) CN112105360B (enExample)
CA (1) CA3088253A1 (enExample)
ES (1) ES3041854T3 (enExample)
WO (1) WO2019144117A1 (enExample)

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TW202430522A (zh) * 2022-09-30 2024-08-01 大陸商江蘇恆瑞醫藥股份有限公司 一種用於bcl-2蛋白靶向降解的嵌合體化合物、其製備方法及其在醫藥上的應用
CN120659777A (zh) * 2022-10-03 2025-09-16 佛罗里达大学研究基金公司 募集Cereblon的Bcl-xL/Bcl-2双重降解剂
WO2024078581A1 (en) * 2022-10-12 2024-04-18 Appicine Therapeutics (Hk) Limited Selective bcl-xl protac compounds and uses thereof
WO2024153185A1 (zh) * 2023-01-18 2024-07-25 苏州宜联生物医药有限公司 包含bcl-2家族蛋白降解剂的抗体药物偶联物及其制备方法和用途
JP2026507476A (ja) * 2023-02-17 2026-03-04 チア タイ ティエンチン ファーマシューティカル グループ カンパニー リミテッド トリフルオロメタンスルホニル基を含む化合物
WO2024179577A1 (zh) * 2023-03-01 2024-09-06 西藏海思科制药有限公司 一种Bcl-2家族蛋白降解剂的药物组合物
CN118724870B (zh) * 2023-03-28 2026-04-28 暨南大学 蛋白降解靶向嵌合体及其应用
TW202535872A (zh) 2023-11-07 2025-09-16 美商樹線生物科學公司 四氫異喹啉異雙功能bcl-xl降解劑
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