JP2020529472A5 - - Google Patents

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Publication number
JP2020529472A5
JP2020529472A5 JP2020527859A JP2020527859A JP2020529472A5 JP 2020529472 A5 JP2020529472 A5 JP 2020529472A5 JP 2020527859 A JP2020527859 A JP 2020527859A JP 2020527859 A JP2020527859 A JP 2020527859A JP 2020529472 A5 JP2020529472 A5 JP 2020529472A5
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JP
Japan
Prior art keywords
group
formula
compound
alkyl
cycloalkyl
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Pending
Application number
JP2020527859A
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English (en)
Japanese (ja)
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JP2020529472A (ja
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Priority claimed from PCT/US2018/044182 external-priority patent/WO2019023634A1/en
Publication of JP2020529472A publication Critical patent/JP2020529472A/ja
Publication of JP2020529472A5 publication Critical patent/JP2020529472A5/ja
Pending legal-status Critical Current

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JP2020527859A 2017-07-28 2018-07-27 ペプチド化合物の環化放出関連する出願の相互参照 Pending JP2020529472A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201762538477P 2017-07-28 2017-07-28
US62/538,477 2017-07-28
PCT/US2018/044182 WO2019023634A1 (en) 2017-07-28 2018-07-27 CYCLATIVE RELEASE OF PEPTIDE COMPOUNDS

Publications (2)

Publication Number Publication Date
JP2020529472A JP2020529472A (ja) 2020-10-08
JP2020529472A5 true JP2020529472A5 (https=) 2021-09-09

Family

ID=63312461

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2020527859A Pending JP2020529472A (ja) 2017-07-28 2018-07-27 ペプチド化合物の環化放出関連する出願の相互参照

Country Status (4)

Country Link
US (1) US11299513B2 (https=)
EP (1) EP3658567A1 (https=)
JP (1) JP2020529472A (https=)
WO (1) WO2019023634A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN112592382B (zh) * 2020-11-27 2022-10-04 安徽大学 一种树脂及其制备方法以及其在制备头尾环肽中的应用
CN120309693B (zh) * 2025-06-12 2025-09-16 杭州湃肽生化科技有限公司 一类环肽化合物及其制备方法和应用

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AUPP616598A0 (en) * 1998-09-25 1998-10-15 University Of Queensland, The Auxiliary for amide bond formation
GB9928323D0 (en) 1999-11-30 2000-01-26 Cyclacel Ltd Peptides
GB2369823B (en) 1999-11-30 2003-06-04 Cyclacel Ltd Assays for cyclin-interacting compounds
US20050153894A1 (en) 1999-11-30 2005-07-14 Cyclacel Limited p21 peptides
EP1345957A2 (en) 2000-12-20 2003-09-24 Novartis AG Inhibitors of the e2f-1/cyclin interaction for cancer therapy
US20040077549A1 (en) 2000-12-20 2004-04-22 Bair Kenneth Walter Inhibitors of the E2F-1/cyclin interaction for cancer therapy
US20040053849A1 (en) 2000-12-20 2004-03-18 Bair Kenneth Walter Inhibitors of the E2F-1/cyclin interaction for cancer therapy
JP2004269357A (ja) 2002-01-25 2004-09-30 Marine Biotechnol Inst Co Ltd 鉄と高い結合能を有する化合物およびその製造方法
WO2006105386A1 (en) 2005-03-30 2006-10-05 Genentech, Inc. Cdk2 inhibitors
WO2008000870A1 (es) 2006-06-19 2008-01-03 Fundación De La Comunidad Valenciana, Centro De Investigación Principe Felipe Compuestos orgánicos que inhiben la actividad catalítica del complejo ciclina a/kinasa 2 dependiente de ciclina mediante su unión a un nuevo sitio farmacofórico en la molécula de ciclina
US20100184684A1 (en) 2009-01-06 2010-07-22 C3 Jian, Inc. Antibacterial and antifungal peptides
US9376465B2 (en) 2012-03-27 2016-06-28 University Of South Carolina Cyclin based inhibitors of CDK2 and CDK4
US20140296484A1 (en) 2013-03-27 2014-10-02 University Of South Carolina Cyclin Based Inhibitors of CDK2 and CDK4
US10011635B2 (en) 2013-09-27 2018-07-03 H. Lee Moffitt Cancer Center And Research Institute, Inc. Cyclic peptide conjugates and methods of use
US20190224279A1 (en) 2015-09-17 2019-07-25 Histide Ag Pharmaceutical association comprising a growth factor receptor agonist conjugated to a bioactive carrier for converting a neoplastic cell into a non-neoplastic cell and uses thereof
DK3349778T3 (da) 2015-09-17 2021-11-22 Histide Ag Farmaceutisk association af vækstfaktorreceptoragonist og adhæsionsproteininhibitor til omdannelse af en neoplastisk celle til en ikke-neoplastisk celle og anvendelser deraf
AU2016323407A1 (en) 2015-09-17 2018-04-19 Histide Ag Pharmaceutical association of growth factor receptor agonist and adhesion protein inhibitor for converting a neoplastic cell into a non-neoplastic cell and uses thereof
WO2017046226A2 (en) 2015-09-17 2017-03-23 Histide Ag Pharmaceutical association for converting a neoplastic cell into a non-neoplastic cell and uses thereof.
WO2017046229A1 (en) 2015-09-17 2017-03-23 Histide Ag Pharmaceutical association of growth factor receptor agonist and adhesion protein inhibitor for converting a neoplastic cell into a non-neoplastic cell and uses thereof
SG10201913355RA (en) 2015-09-17 2020-02-27 Histide Ag Pharmaceutical association for converting a neoplastic cell into a non-neoplastic cell and uses thereof

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