JP2020529472A - ペプチド化合物の環化放出関連する出願の相互参照 - Google Patents

ペプチド化合物の環化放出関連する出願の相互参照 Download PDF

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JP2020529472A
JP2020529472A JP2020527859A JP2020527859A JP2020529472A JP 2020529472 A JP2020529472 A JP 2020529472A JP 2020527859 A JP2020527859 A JP 2020527859A JP 2020527859 A JP2020527859 A JP 2020527859A JP 2020529472 A JP2020529472 A JP 2020529472A
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group
formula
compound
alkyl
acid
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JP2020529472A5 (https=
Inventor
ラマセシャン マヘシュ
ラマセシャン マヘシュ
ボックス アンドリュー
ボックス アンドリュー
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サークル ファーマ，インコーポレイティド
サークル ファーマ，インコーポレイティド
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Publication of JP2020529472A publication Critical patent/JP2020529472A/ja
Publication of JP2020529472A5 publication Critical patent/JP2020529472A5/ja
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/04—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
    • C07K1/042—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers characterised by the nature of the carrier
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/107—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length by chemical modification of precursor peptides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/64—Cyclic peptides containing only normal peptide links

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Analytical Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Peptides Or Proteins (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
JP2020527859A 2017-07-28 2018-07-27 ペプチド化合物の環化放出関連する出願の相互参照 Pending JP2020529472A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201762538477P 2017-07-28 2017-07-28
US62/538,477 2017-07-28
PCT/US2018/044182 WO2019023634A1 (en) 2017-07-28 2018-07-27 CYCLATIVE RELEASE OF PEPTIDE COMPOUNDS

Publications (2)

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JP2020529472A true JP2020529472A (ja) 2020-10-08
JP2020529472A5 JP2020529472A5 (https=) 2021-09-09

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Family Applications (1)

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JP2020527859A Pending JP2020529472A (ja) 2017-07-28 2018-07-27 ペプチド化合物の環化放出関連する出願の相互参照

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Country Link
US (1) US11299513B2 (https=)
EP (1) EP3658567A1 (https=)
JP (1) JP2020529472A (https=)
WO (1) WO2019023634A1 (https=)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN112592382A (zh) * 2020-11-27 2021-04-02 安徽大学 一种树脂及其制备方法以及其在制备头尾环肽中的应用

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN121248729A (zh) * 2025-06-12 2026-01-02 杭州湃肽生化科技有限公司 一种全保护环肽及其制备方法

Citations (1)

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JP2002525376A (ja) * 1998-09-25 2002-08-13 ザ ユニバーシティ オブ クイーンズランド アミド結合形成のための補助基

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US20050153894A1 (en) 1999-11-30 2005-07-14 Cyclacel Limited p21 peptides
US20040053849A1 (en) 2000-12-20 2004-03-18 Bair Kenneth Walter Inhibitors of the E2F-1/cyclin interaction for cancer therapy
BR0116330A (pt) 2000-12-20 2004-02-25 Novartis Ag Inibidores da interação e2f-1/ciclina para terapia de câncer
US20040077549A1 (en) 2000-12-20 2004-04-22 Bair Kenneth Walter Inhibitors of the E2F-1/cyclin interaction for cancer therapy
JP2004269357A (ja) 2002-01-25 2004-09-30 Marine Biotechnol Inst Co Ltd 鉄と高い結合能を有する化合物およびその製造方法
WO2006105386A1 (en) 2005-03-30 2006-10-05 Genentech, Inc. Cdk2 inhibitors
WO2008000870A1 (es) 2006-06-19 2008-01-03 Fundación De La Comunidad Valenciana, Centro De Investigación Principe Felipe Compuestos orgánicos que inhiben la actividad catalítica del complejo ciclina a/kinasa 2 dependiente de ciclina mediante su unión a un nuevo sitio farmacofórico en la molécula de ciclina
US20110039763A1 (en) 2009-01-06 2011-02-17 C3 Jian, Inc. Targeted antimicrobial moieties
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US20140296484A1 (en) 2013-03-27 2014-10-02 University Of South Carolina Cyclin Based Inhibitors of CDK2 and CDK4
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WO2017046226A2 (en) 2015-09-17 2017-03-23 Histide Ag Pharmaceutical association for converting a neoplastic cell into a non-neoplastic cell and uses thereof.
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JP6890836B2 (ja) 2015-09-17 2021-06-18 ヒスタイド アクツィエンゲゼルシャフト 腫瘍細胞を非腫瘍細胞に変換するための医薬的連合体及びその使用
WO2017046229A1 (en) 2015-09-17 2017-03-23 Histide Ag Pharmaceutical association of growth factor receptor agonist and adhesion protein inhibitor for converting a neoplastic cell into a non-neoplastic cell and uses thereof
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JP2002525376A (ja) * 1998-09-25 2002-08-13 ザ ユニバーシティ オブ クイーンズランド アミド結合形成のための補助基

Non-Patent Citations (6)

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BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS (2008) VOL.18, PP.4731-4735, JPN6022021031, ISSN: 0004959467 *
J. AM. CHEM. SOC. (1999) VOL.121, PP.3311-3320, JPN6022021028, ISSN: 0004959466 *
ORGANIC LETTERS (2005) VOL.7, NO.13, PP.2647-2650, JPN6022021026, ISSN: 0004959465 *
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Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN112592382A (zh) * 2020-11-27 2021-04-02 安徽大学 一种树脂及其制备方法以及其在制备头尾环肽中的应用

Also Published As

Publication number Publication date
EP3658567A1 (en) 2020-06-03
WO2019023634A1 (en) 2019-01-31
US11299513B2 (en) 2022-04-12
US20200207803A1 (en) 2020-07-02

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